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N-[2-(piperidin-1-yl)ethyl]-3-[(pyridin-3-ylmethyl)sulfamoyl]benzamide
(4aR,8aR)-2-methanesulfonyl-7-[(6-methyl-2H-1,3-benzodioxol-5-yl)methyl]-decahydro-2,7-naphthyridin-4a-ol
(3aS,6aR)-3-cyclopentyl-5-(2,3-dihydro-1H-inden-2-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-{4-hydroxy-4-[2-(4-phenylazepane-1-carbonyl)-1-benzofuran-5-yl]piperidin-1-yl}butan-1-one
[(2,2-difluoro-2H-1,3-benzodioxol-5-yl)methyl](methyl){[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
6-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,2,3,4-tetrahydroquinoxaline-2,3-dione
(2S,4R)-1-[(2,3-dimethoxyphenyl)methyl]-N-(propan-2-yl)-4-({[3-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
N-(1-benzylpyrrolidin-3-yl)-3-cyclohexyl-N-methyl-1H-pyrazole-4-carboxamide
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
3-(1H-1,2,3,4-tetrazol-1-yl)-1-{3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}propan-1-one
methyl (2S)-2-cyclopropyl-2-(3-{[2-(methylsulfanyl)phenyl]carbamoyl}propanamido)acetate
2-[2-(4-chlorophenoxy)ethyl]-2,7-diazaspiro[4.5]decan-6-one
3-[(3aS,6aS)-3a-(hydroxymethyl)-octahydrocyclopenta[c]pyrrole-2-carbonyl]-6-phenyl-1,2-dihydropyridin-2-one
2-[4-(1-benzyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]-N-(1,3-dimethyl-1H-pyrazol-4-yl)acetamide
N-[3-(1H-imidazol-1-yl)propyl]-2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
(3S,9aR)-8-(2-chlorobenzoyl)-3-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-(benzyloxy)-1-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]butan-1-one
1-ethyl-8-methyl-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(5-{[1-(2-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}thiophen-2-yl)acetamide
(2S,4R)-N-(1,1-dioxo-1λ6-thiolan-3-yl)-4-[(4-methoxyphenyl)sulfanyl]-1-{[4-(trifluoromethoxy)phenyl]methyl}pyrrolidine-2-carboxamide
4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperidine
4-cyclopropanecarbonyl-6-[(3-fluorophenyl)methoxy]-1-(2-phenylethyl)-1,4-diazepan-2-one
N-[2-({[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)ethyl]acetamide
N-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-N-methyloxolan-3-amine
(2S,4S)-4-amino-1-(2,3-dihydro-1H-inden-2-yl)-N,N-diethylpyrrolidine-2-carboxamide
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-1-methylpiperidine-2-carboxamide
N2-[1,3-dimethyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-N1-(3-methylpyridin-4-yl)ethane-1,2-diamine
(3R,5S)-5-[(4-methylpiperazin-1-yl)methyl]-N-(2-methylpropyl)-1-(2-phenylethyl)piperidine-3-carboxamide
1-[4-(4-aminopiperidin-1-yl)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
[(1-ethyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)[(3-methylthiophen-2-yl)methyl]amine
2-methoxy-5-oxo-6-[2-(pyrazin-2-yl)ethyl]-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-3-yl]piperazine
N-(3-hydroxy-3-phenylpropyl)-N,3,5-trimethyl-1-benzofuran-2-carboxamide
(2E)-3-(2-chlorophenyl)-1-[3-(4-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}phenoxymethyl)piperidin-1-yl]prop-2-en-1-one
N-[(3S,4R)-1-{[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-4-propylpyrrolidin-3-yl]methanesulfonamide
2-(2-methoxyethyl)-9-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
7-methoxy-4-methyl-2-(1H-pyrazol-4-yl)quinoline
4-(2-methoxyphenyl)-2-[5-methyl-4-(4-methylpiperazine-1-carbonyl)-1H-pyrazol-1-yl]pyrimidine
N-benzyl[(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)amino]sulfonamide
2-{9-[(3,5-difluorophenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
ethyl 1-(2,4-dimethyl-6-oxo-1,6-dihydropyridin-3-yl)-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylate
N-{1-[7-(but-2-ynoyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-3-methylbutyl}-3-methoxypropanamide
(3aS,6aR)-3-[3-(4-methoxyphenyl)propyl]-5-[2-(methylsulfanyl)pyrimidin-4-yl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-[(4-chlorophenyl)methyl]-4-[2,2-dimethyl-3-(pyrrolidin-1-yl)propyl]piperazine
2-(4-{[4-(3-methoxyphenyl)piperazin-1-yl]methyl}phenyl)-6-methyl-3,4-dihydropyrimidin-4-one
2-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]-1H-1,3-benzodiazole
1-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-(pyridin-3-yl)ethane-1,2-dione
3-(3-methoxypropyl)-3-(1-methylpiperidin-4-yl)-1-[2-(methylsulfanyl)phenyl]urea
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
1-[1-(2-aminopyrimidin-4-yl)piperidin-4-yl]-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide