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4-[(3-methylphenyl)methyl]-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{2-[4-(2-fluorophenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]ethyl}-2-(pyridin-2-ylsulfanyl)acetamide
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-(pyridin-2-ylmethyl)piperidin-4-ol
methyl 3-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]-5-methoxybenzoate
N-cyclopropyl-2-(3-methyl-2-oxoimidazolidin-1-yl)-N-(1,3-thiazol-2-ylmethyl)acetamide
(2R)-2-amino-2-[1-(2-fluorophenyl)-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]ethan-1-ol
N2-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-N4,N4,5-trimethylpyrimidine-2,4-diamine
2-(dimethylamino)-1-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}ethan-1-one
4-[(1-{1-[(2-chloro-4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-4-yl)methyl]morpholine
1-[1-(3-{1H-[1,2,3]triazolo[4,5-b]pyridin-6-yl}phenyl)ethyl]pyrrolidine
N-[(2-ethoxyphenyl)methyl]-4,6-dimethyl-2-oxo-N-(prop-2-en-1-yl)-1,2-dihydropyridine-3-carboxamide
5-{[2-(3-fluorophenyl)piperidin-1-yl]methyl}-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}(methyl)[2-(oxan-4-yl)ethyl]amine
N-{1-oxa-8-azaspiro[4.5]decan-3-yl}-2-[3-(trifluoromethyl)phenyl]acetamide
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-(thiophen-2-ylmethyl)-decahydro-1,6-naphthyridin-2-one
2-[(2,6-dichlorophenyl)methyl]-5-(thiomorpholine-4-carbonyl)pyrimidin-4-ol
N-(2,6-dimethylphenyl)-2-[3-(pyridin-3-yl)propanamido]benzamide
3-[5-(thiolan-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl]pyridine
1-(2-{[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]amino}-4-methylpyrimidin-5-yl)ethan-1-one
5-(dimethylamino)-2-{2-[4-(3-methylphenoxy)piperidin-1-yl]-2-oxoethyl}-2,3-dihydropyridazin-3-one
3-(1-methyl-1H-pyrazol-4-yl)-1-[4-(4-methylphenoxy)piperidin-1-yl]propan-1-one
5-[1-(2,2-dimethylpropyl)-4-hydroxypiperidin-4-yl]-N-[2-(2-fluorophenyl)ethyl]-1-benzofuran-2-carboxamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-ethyl-N-(2-methylprop-2-en-1-yl)piperidine-3-carboxamide
(3R,4S)-4-cyclopropyl-N,N-dimethyl-1-[(5-methylpyrazin-2-yl)methyl]pyrrolidin-3-amine
1-[(3S,4S)-3-hydroxy-4-{4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}pyrrolidin-1-yl]-2-(methylsulfanyl)ethan-1-one
N-(2-ethylphenyl)-3-[4-(2-oxopyrrolidin-1-yl)butanamido]benzamide
1-(5-methyl-2-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}benzoyl)azepane
4-[1-(1,2,5-trimethyl-1H-pyrrole-3-carbonyl)piperidin-3-yl]benzoic acid
1-[4-(adamantan-1-yl)piperazin-1-yl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]pyrazolo[1,5-a]pyridine-7-carboxamide
4-(1-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carbonyl)morpholine
ethyl 4-(3-{2-[(4-methoxy-2-methylphenyl)carbamoyl]ethyl}piperidin-1-yl)piperidine-1-carboxylate
2-{[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}-1,2-oxazinane
2-{2-[1-(4-oxo-4H-chromene-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
2,6-dimethyl-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]benzamide
8-[(2E)-2-methylbut-2-en-1-yl]-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
2-(cyclopropylmethyl)-7-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-(oxolan-3-ylmethyl)-3-(thiomorpholine-4-sulfonyl)benzamide
2-[4-(2-amino-6-methylpyrimidin-4-yl)-1H-pyrazol-1-yl]-N-(1-cyclopentyl-3-methyl-1H-pyrazol-5-yl)acetamide
ethyl 3-benzyl-1-[(2-ethoxy-2-oxoethyl)carbamoyl]piperidine-3-carboxylate
(2S,4S)-1-(2,3-dihydro-1H-inden-2-yl)-4-{[(4-methoxy-2,5-dimethylphenyl)methyl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
N-(4-methoxyphenyl)-3-oxo-3-{5-oxo-1,4,9-triazaspiro[5.5]undecan-9-yl}propanamide
2-(1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}pyrrolidin-2-yl)-4-methyl-1H-1,3-benzodiazole
N-(3-chloro-4-methoxyphenyl)-4-(hydroxymethyl)-4-(2-phenoxyethyl)piperidine-1-carboxamide
(1R,5R)-6-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
2-{4-[(4-phenoxyphenyl)methyl]morpholin-2-yl}ethan-1-amine
3-ethyl-5-hydroxy-N-methyl-N-(1,2-oxazol-5-ylmethyl)adamantane-1-carboxamide
3-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[(2-methylphenyl)(pyridin-4-yl)methyl]propanamide
N-{1-[1-(2-fluorophenyl)-1H-pyrazol-4-yl]ethyl}-1-(propan-2-yl)piperidine-4-carboxamide
3-{1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-3-yl}-N-[(5-methylfuran-2-yl)methyl]propanamide