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2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]-1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidine
1-phenyl-4-{2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidine-1-carbonyl}-1H-1,2,3-triazole
1-[(2-fluorophenyl)methyl]-3-hydroxy-3-({methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)piperidin-2-one
N,N-dimethyl-2-[4-(1,2,3,4-tetrahydroisoquinolin-5-yl)phenyl]acetamide
methyl (2R)-2-(4-hydroxyphenyl)-2-{5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-6-yl}acetate
7-(3-cyclopropyl-1,2-oxazole-5-carbonyl)-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-2-(naphthalen-2-yloxy)propanamide
3-methyl-8-{[1-(3-methylbutyl)-1H-1,3-benzodiazol-2-yl]methyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
3-[1-(1-benzyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]-N-cyclopropylpropanamide
3,5-dimethyl-N-{3-methyl-1-[7-(4-methyl-1,3-oxazole-5-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]butyl}benzamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-1-cyclopentyl-N-methyl-5-oxopyrrolidine-3-carboxamide
1'-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
N-{[1-(8-chloroquinolin-2-yl)piperidin-4-yl]methyl}acetamide
N-{[1-(furan-2-ylmethyl)pyrrolidin-3-yl]methyl}-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
N-[2-(4-{[4-(4-fluorophenyl)-4-oxobutanamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]pyridine-2-carboxamide
2-(2H-1,3-benzodioxol-5-yloxy)-N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}propanamide
methyl 6-(2-methylbutanoyl)-2-[(3-methylphenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-methyl-2-oxo-8-[4-(trifluoromethyl)benzoyl]-1,8-diazaspiro[4.5]decane-4-carboxylic acid
(5S)-5-[1-benzyl-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]pyrrolidin-2-one
ethyl 4-[4-(4-{[2-(3-chlorophenyl)ethyl]amino}piperidin-1-yl)benzoyl]piperazine-1-carboxylate
cyclohexyl[4-(pyridin-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methanol
1-[3-(2-methylphenyl)benzoyl]-3-(1H-pyrazol-5-yl)piperidine
1-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
1-{1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carbonyl}piperidin-4-amine
1-(3-methoxybenzoyl)-4-(2,4,5-trimethylbenzoyl)piperazine
5-({2-[(3-fluorophenyl)methyl]morpholin-4-yl}methyl)-N-propylpyrimidin-2-amine
9-(3-methylbut-2-enoyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-({[(3-ethyl-1,2-oxazol-5-yl)methyl](methyl)amino}methyl)-6-methoxyphenol
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methyloxolane-3-carboxamide
1-{3-[(3-fluorophenyl)amino]piperidin-1-yl}-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
4-[(3R,4S)-3-amino-4-cyclopropylpyrrolidine-1-carbonyl]-6-(2-methylpropyl)-1,2-dihydropyrimidin-2-one
1-(furan-2-ylmethyl)-N-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}piperidine-3-carboxamide
N-{2-methyl-1-[3-(3-methylpyridin-2-yl)-1,2,4-oxadiazol-5-yl]propyl}acetamide
1-[4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-2-(2H-indazol-2-yl)ethan-1-one
N-(1-{1-[4-(2-methylpropyl)benzoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide
N-[2-(1-benzylpyrrolidin-3-yl)ethyl]-4-chloro-1,3-dimethyl-1H-pyrazole-5-carboxamide
4-ethyl-3-{1-[2-(pyridin-2-yl)pyrimidine-5-carbonyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3,4,7-trimethyl-N-[(3S)-pyrrolidin-3-yl]-1H-indole-2-carboxamide
1-benzyl-4-(5-{[(4-fluorophenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)piperidine
8-chloro-3-(pyrrolidin-3-yl)-3,4-dihydroquinazolin-4-one
2-{[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]amino}-N-(pyrazin-2-yl)acetamide
ethyl(1H-indol-7-ylmethyl)[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amine
1-(5-chloro-3-fluoropyridin-2-yl)-4-[(3-methylpyridin-2-yl)methyl]piperazine
(2S,4R)-N,N-diethyl-1-(3-hydroxypropanoyl)-4-(2-methylfuran-3-amido)pyrrolidine-2-carboxamide
2-(5-tert-butyl-1,3,4-oxadiazol-2-yl)-9-oxa-2-azaspiro[5.5]undecane
3-[3-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]-4,5,6,7-tetrahydro-1H-indazole
3-[4-ethyl-5-oxo-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]-2,3-dihydro-1λ6-thiophene-1,1-dione
N-tert-butyl-7-[(3-methylphenyl)methyl]-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
N-butyl-4-{[2-(4-methoxyphenyl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-[3-(4-chloro-1H-pyrazol-1-yl)propyl]-2-ethylpyrimidine-5-carboxamide