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1-(2-chlorophenyl)-4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-one
1-cyclopentyl-4-(4-phenyl-1,4-diazepane-1-carbonyl)pyrrolidin-2-one
8-(1-benzofuran-2-ylmethyl)-1-benzyl-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}pyrimidin-4-yl)piperidin-3-ol
8-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
N-benzyl-N-ethyl-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
2-chloro-4-[4-(4-methylpiperazin-1-yl)quinazolin-6-yl]benzamide
methyl 2-[({1-[(3,4-difluorophenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)(methyl)amino]acetate
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
1-methyl-4-(2-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}pyridine-4-carbonyl)piperazine
2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-1-[4-(1H-pyrazol-1-yl)butan-2-yl]-1H-imidazole
{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}(methyl){[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
3-{[(4-benzyl-5-{1-[(2-fluorophenyl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)sulfanyl]methyl}pyridine
2-[(2-butoxyacetamido)methyl]-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
N-{2-[(2-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-2-oxoethyl)sulfanyl]phenyl}acetamide
1-(methoxymethyl)-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}cyclobutane-1-carboxamide
(3S,4R)-4-methyl-1-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}piperidine-3,4-diol
(4aS,8aR)-6-(5-chloropyridine-3-carbonyl)-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
(3S,4R)-1-(4-ethyl-5-methylthiophene-3-carbonyl)-4-(3-methylthiophen-2-yl)piperidin-3-ol
5-chloro-2-methoxy-N-{3-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]propyl}benzene-1-sulfonamide
(4aS,8aR)-1-[3-(methylsulfanyl)propyl]-6-(pyrazin-2-yl)-decahydro-1,6-naphthyridin-2-one
4-(1H-imidazol-1-ylmethyl)-1-(2-propyl-1,3-thiazole-4-carbonyl)piperidin-4-ol
2-(3,4-dimethoxyphenyl)-N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]acetamide
2-[(4aS,7aR)-4-(2-methoxyacetyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N-(thiophen-2-ylmethyl)acetamide
2-[(2-{[(2-methylphenyl)(pyridin-4-yl)methyl]carbamoyl}phenyl)amino]acetic acid
[3-(2-phenylethyl)-1-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl]methanol
(1S,4S)-2-{5-ethyl-6-methylthieno[2,3-d]pyrimidin-4-yl}-2,5-diazabicyclo[2.2.1]heptane
2-{[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]amino}-N-[5-(oxolan-2-yl)-1,3,4-thiadiazol-2-yl]acetamide
6-oxo-N-[3-(3-phenylpropanamido)phenyl]-1,6-dihydropyridine-2-carboxamide
2-cyclopropyl-N-[3-(methylsulfanyl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
methyl 2-[N-methyl-1-(3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}phenyl)formamido]acetate
N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-2-[(prop-2-en-1-yl)amino]benzamide
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
N-[1-methyl-3-(pyridin-2-yl)-1H-pyrazol-5-yl]-4-(3-methylpyridin-2-yl)piperazine-1-carboxamide
N-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-N-[(2-methoxyphenyl)methyl]cyclopropanamine
1-[(3-fluorophenyl)methyl]-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
1-(2-{4-[2-(trifluoromethyl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethyl)piperazine
1-(cyclopropylmethyl)-5-[4-(1H-pyrazol-1-yl)benzoyl]-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
[1-(2-chlorobenzenesulfonyl)-3-ethylpiperidin-3-yl]methanol
N-(2,1,3-benzoxadiazol-4-ylmethyl)-N-methyl-2,3-dihydro-1H-inden-2-amine
(3S,4R)-3-methoxy-1-(7-methyl-2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidin-4-amine
(1S,5R)-6-(cyclopropylmethyl)-3-[4-(3,5-dimethyl-1H-pyrazol-1-yl)butanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
[(3R,4S)-1-[(2,4-dimethoxyphenyl)methyl]-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
(2S)-1-[(6,8-dimethyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-N-ethylpyrrolidine-2-carboxamide
4-{3-hexyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decane-8-carbonyl}benzonitrile
3-{[1-(quinoxaline-5-carbonyl)pyrrolidin-3-yl]methyl}benzoic acid
1-cyclopentyl-N-{2-[4-(dimethylamino)phenyl]ethyl}-5-oxopyrrolidine-3-carboxamide
[(3R,4R)-1-(8-methoxy-4-methylquinolin-2-yl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
N-[(2-fluorophenyl)methyl]-3-{1-[3-(pyridin-2-yl)propanoyl]piperidin-3-yl}propanamide
1-[4-(dimethylamino)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-hydroxyethan-1-one