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N-[(2-chloropyridin-3-yl)methyl]-N-methyl-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
N-[(3S,7S,8aS)-3-ethyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-methylbenzamide
4-chloro-1-methyl-N-[2-(3-methylthiophen-2-yl)ethyl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
4-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-6-methylpyrimidin-2-amine
N-(3-chloro-5-fluorophenyl)-4-(3-hydroxypiperidin-1-yl)piperidine-1-carboxamide
N'-cycloheptyl-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}butanediamide
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-6-methyl-1-(propan-2-yl)-1H-pyrazolo[3,4-b]pyridine-4-carboxamide
1-(cyclopropylmethyl)-3-[(2-methylphenyl)methyl]-6-(thiolan-3-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
(2R,6R)-11-methoxy-4-[3-(methylsulfanyl)propyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-methyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-(pyridin-2-ylmethyl)piperazin-2-yl}ethan-1-ol
1-[3-(dimethylamino)benzoyl]-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
N-{[4-(2-methylpropyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}furan-2-carboxamide
1,5-dimethyl-2-phenyl-4-(1-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1H-1,2,3-triazol-4-yl)-2,3-dihydro-1H-pyrazol-3-one
N-[(2-methoxynaphthalen-1-yl)methyl]-1-methyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[(3-methoxyphenyl)methyl]-4-(6-methylpyridine-3-carbonyl)piperazin-2-one
2-methoxy-5-{4-phenyl-1-[2-(trimethyl-1H-pyrazol-1-yl)ethyl]-1H-imidazol-5-yl}pyrimidine
ethyl 1-[2-(4-methoxyphenyl)ethyl]-5-(quinolin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-ethyl-8-(2-methyl-1,3-benzothiazole-6-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
6-(methoxymethyl)-N-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}pyrimidin-4-amine
ethyl 1-[(3,7-dimethyl-1H-indol-2-yl)methyl]-4-(2-methoxyethyl)piperidine-4-carboxylate
N-methyl-N-{2-[(oxan-3-ylmethyl)carbamoyl]phenyl}thiophene-2-carboxamide
2,4-dimethoxy-N-{[4-(2-methylpropyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}benzamide
N-(4-acetylphenyl)-3-(naphthalene-2-carbonyl)piperidine-1-carboxamide
5-methyl-1'-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[2-(azepan-1-yl)ethyl]-3-[(2-fluorophenyl)formamido]-N-methylpropanamide
(2S,4S)-4-(4-{2-[(3-methylthiophen-2-yl)formamido]propan-2-yl}-1H-1,2,3-triazol-1-yl)pyrrolidine-2-carboxylic acid
N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide
3-{1-[3-(prop-2-en-1-yloxy)benzoyl]piperidin-3-yl}-1-(pyrrolidin-1-yl)propan-1-one
(1R,2S)-N-butyl-2-(5,6,7,8-tetrahydro-1,6-naphthyridine-6-carbonyl)cyclohexane-1-carboxamide
1-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(piperidine-1-carbonyl)piperidine
2-{4-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}-5-ethylpyrimidine
1-{3-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-3-oxopropyl}azepan-2-one
1-{2-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
(4aS,8aR)-6-(ethanesulfonyl)-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-1H-1,2,3-triazole-5-carboxamide
8-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3aR,7aS)-2-[6-(morpholine-4-carbonyl)pyrazin-2-yl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
1-[4-(2-methoxyphenoxy)piperidin-1-yl]-3-(methylsulfanyl)propan-1-one
7-cyclohexyl-2-[(2-methyl-1,3-thiazol-4-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
2-{3-[1-(2-hydroxyethyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]piperidin-1-yl}acetamide
N-({3-[(3-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)-3-(furan-2-yl)-3-phenylpropanamide
1-cyclopentyl-5-[2-({[3-(trifluoromethyl)phenyl]methyl}amino)ethyl]pyrrolidin-2-one
N-[1-(2-phenylethyl)piperidin-3-yl]thiophene-2-carboxamide
2-cyclopropyl-9-(1,2,4-oxadiazol-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-cyclopropyl-7-(2,3-dihydro-1-benzofuran-5-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(1R,5R)-N,N-dimethyl-6-{pyrazolo[1,5-a]pyridine-3-carbonyl}-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
(1R,5R)-6-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
3-{[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-methyl-1H-1,2,4-triazol-5-yl]methyl}-1λ6-thiolane-1,1-dione
2-[4-(5-methylpyrimidin-4-yl)piperidine-1-carbonyl]-5-(1H-1,2,3,4-tetrazol-1-yl)phenol