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3-{[1-(2-amino-5,6,7,8-tetrahydroquinazoline-4-carbonyl)pyrrolidin-3-yl]methyl}benzamide
1-(2,2-dimethylpropyl)-3-hydroxy-3-[({2-[(4-methylpyridin-2-yl)amino]ethyl}amino)methyl]piperidin-2-one
4-{3-[1-ethyl-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]phenyl}morpholine
2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]-N-[(5-phenyl-4H-1,2,4-triazol-3-yl)methyl]acetamide
2-({[(3R,4R)-1-[3-(4-fluorophenyl)benzoyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
2-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]pyridine-3-carboxamide
5-oxo-1-[4-(propan-2-yl)phenyl]-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}pyrrolidine-3-carboxamide
(1R,9aR)-1-{[2-(pyridin-3-yl)-1H-imidazol-1-yl]methyl}-octahydro-1H-quinolizin-1-ol
1-[(1-propyl-1H-imidazol-2-yl)methyl]-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
2-hydroxy-3-methyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]butanamide
N-(1,3-dihydro-2-benzofuran-5-yl)-4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carboxamide
1-(3,5-dimethylphenyl)-N-[(4-methanesulfonylmorpholin-2-yl)methyl]piperidin-4-amine
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-2-(pyridin-3-yl)acetamide
{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}[(1-ethyl-1H-pyrazol-4-yl)methyl]amine
(1-{[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
(3S,4S)-1-[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl]-4-propylpyrrolidine-3-carboxylic acid
N-{1-[1-(2H-1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-2-(2-fluorophenyl)ethyl}-N-methylthiophene-2-carboxamide
5-{[(4-methoxynaphthalen-1-yl)oxy]methyl}-N-methyl-N-(1-methylpyrrolidin-3-yl)-1,2-oxazole-3-carboxamide
3-chloro-6-[4-(3,5-dimethylphenyl)-3-oxopiperazin-1-yl]pyridine-2-carboxylic acid
(1R,5S)-6-{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}-6-azabicyclo[3.2.1]octane
4-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyridine
N-[3-chloro-2-(4-ethylpiperazin-1-yl)phenyl]-1,2,3-thiadiazole-4-carboxamide
methyl 2-[({2-[2-hydroxy-3-(piperidin-1-yl)propoxy]phenyl}methyl)(methyl)amino]acetate
2-methyl-4-{3-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]phenyl}but-3-yn-2-ol
5-(2-chlorophenyl)-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]furan-2-carboxamide
1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-N-methylpiperidine-3-carboxamide
7-fluoro-2-methyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]quinoline-4-carboxamide
(3R,4R)-1-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
methyl 3-(furan-3-amido)-1-(2-methylpropyl)-5-[(thiophen-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(2R,6R)-4-(dimethylsulfamoyl)-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-(cyclohexylmethyl)-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-6-oxopiperidine-3-carboxamide
7-methyl-2-(pyrrolidine-1-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
3-[3-(3-methoxybenzoyl)piperidin-1-yl]propanamide
1-methyl-9-[2-(trifluoromethyl)benzoyl]-1,4,9-triazaspiro[5.5]undecan-5-one
1-[(4aR,8aR)-4a-hydroxy-7-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
N-[2-(1H-indol-3-yl)ethyl]-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-(3-{1-[2-(dimethylamino)ethyl]-4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)pyridine-2-carbonitrile
1-(1-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-4-yl)propan-1-ol
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[3-(1H-1,2,4-triazol-1-yl)propanoyl]pyrrolidine-3-carboxylic acid
9-(cyclopropylmethyl)-4-(6-methoxypyrimidin-4-yl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
7-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-(furan-2-ylmethyl)-N,2,6-trimethylquinoline-4-carboxamide
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-1-(2-ethoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-1-[4-(quinazolin-4-yl)piperazin-1-yl]ethan-1-one
1-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(propan-2-yloxy)ethan-1-one
1-[2-(methylamino)pyridine-4-carbonyl]-4-phenoxypiperidine-4-carboxylic acid
7-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
8-{[3-(morpholin-4-yl)phenyl]methyl}-2,8-diazaspiro[4.5]decan-3-one
6-ethoxy-3-{[4-(pyridin-4-yl)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
4-(3-methyl-1,2,4-oxadiazol-5-yl)-2-(pyridin-4-yl)quinoline