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(3aS,6aS)-2-(cyclopropylmethyl)-5-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(2,4-dioxoimidazolidin-1-yl)-N-{1-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
3-[(1-acetylpiperidin-4-yl)oxy]-N-benzyl-N-(2-hydroxyethyl)-4-methoxybenzamide
1-(2-ethoxyethyl)-5-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
methyl 7-oxo-3-[5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carbonyl]-9-(propan-2-yloxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-3-[1-(4-methoxyphenyl)-3-methyl-1H-pyrazol-5-yl]urea
3-{5-[(dimethyl-1,2-oxazol-4-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1-(pyrrolidin-1-yl)propan-1-one
1-(furan-2-ylmethyl)-N-[2-(1H-indol-3-yl)ethyl]piperidine-3-carboxamide
8-(1-phenylcyclopentanecarbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-{1'-[(2R)-2-hydroxy-2-phenylacetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
2-methyl-4-{methyl[(6-methyl-2H-1,3-benzodioxol-5-yl)methyl]amino}butan-2-ol
3-[3-ethyl-4-(4-fluorophenyl)-1-methyl-1H-pyrazol-5-yl]-1-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}urea
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-4-phenyl-1H-imidazole-5-carboxamide
5-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-4-methylphenyl]-N,N-dimethylfuran-2-carboxamide
3-(6-chloro-2-methylpyridin-3-yl)-1-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)urea
7-[(2-methyl-1,3-oxazol-4-yl)methyl]-N-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-2,3-dimethyl-1H-indole-7-carboxamide
N-(cyclobutylmethyl)-N-(oxolan-2-ylmethyl)-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
(3aS,6aS)-2-(2-cyclopentylacetyl)-5-[(2-fluorophenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(2-{[(3R,5S)-5-[3-(trifluoromethyl)phenoxymethyl]piperidin-3-yl]formamido}ethyl)acetamide
3-methyl-5-{2-oxo-2-[6-oxo-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-2-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
(1-benzothiophen-2-ylmethyl)({3-[(3,4-dimethoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)methylamine
2-(1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}piperidin-4-yl)-1,2,3,4-tetrahydroisoquinoline
3-(3-methyl-1,2,4-thiadiazol-5-yl)-1-[(1-methyl-4-phenylpiperidin-4-yl)methyl]urea
N-cyclopropyl-2-[4-({[2-(pyrazin-2-yl)ethyl]carbamoyl}amino)phenyl]acetamide
N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
(4aS,8aR)-6-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-(2-phenylethyl)-decahydro-1,6-naphthyridin-2-one
N-benzyl-5-[(4-hydroxyphenyl)methyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-[3-(1H-imidazol-1-yl)propyl]-9-[3-(methylsulfanyl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
N-{[2-(diethylamino)pyridin-3-yl]methyl}-2-methylfuran-3-carboxamide
4-{[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]methyl}pyridine
3-(2-ethylphenoxy)-1-[(2R)-oxolane-2-carbonyl]azetidine
N-{1-[1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
1-(2,3-dihydro-1H-inden-5-yl)-3-methyl-3-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}urea
1-(oxan-4-ylmethyl)-6-(pyridin-3-ylmethoxy)-4-[3-(thiophen-2-yl)propanoyl]-1,4-diazepan-2-one
1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(pyridin-3-yl)piperazine
methyl 4-{[4-(hydroxymethyl)-4-(2-phenoxyethyl)piperidin-1-yl]methyl}benzoate
3-(1-butyl-1H-imidazol-2-yl)-1-(4-fluoro-3-methylbenzoyl)piperidine
1-{1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carbonyl}-1,4-diazepan-5-one
4-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-1λ6-thiomorpholine-1,1-dione
3-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-1-benzothiophene-2-carboxamide
2-[1-(3-methylbut-2-en-1-yl)-4-{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperazin-2-yl]ethan-1-ol
2-({[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-3-yl]oxy}methyl)pyridine
ethyl 4-[1-methyl-6-oxo-3-(pyridin-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl]-1H-pyrazole-3-carboxylate
5-(3-{imidazo[1,2-a]pyridin-2-yl}-1,2,4-oxadiazol-5-yl)-1-(2-phenylethyl)piperidin-2-one
1-[2-(naphthalen-1-ylmethyl)morpholin-4-yl]propan-1-one
2-ethyl-4-[1-(3-methylphenyl)-1H-imidazol-2-yl]pyrimidine
1-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propan-1-one
{1-[(8-methoxy-2H-chromen-3-yl)methyl]-3-(2-methoxyethyl)piperidin-3-yl}methanol