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1-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(pyrazin-2-yl)ethan-1-one
N-[(3R,4S)-1-acetyl-4-propylpyrrolidin-3-yl]-2-(4-fluoro-3-methylphenyl)acetamide
1-[(2-methyl-1,3-oxazol-4-yl)methyl]-4-[2-(1H-1,2,3,4-tetrazol-5-yl)acetyl]-1,4-diazepane-6-carboxylic acid
1-(2-propoxyethyl)-4-(1H-1,2,3-triazole-5-carbonyl)piperazine
4-{2-[2-(2-chloro-6-fluorophenyl)-1H-imidazol-1-yl]ethyl}-1-methylpiperidine
3-(8-chloroquinolin-5-yl)-1-(oxan-4-yl)urea
N-[(1-cyclopentylpiperidin-4-yl)methyl]-3-(1-methyl-1H-pyrazol-4-yl)-N-(pyridin-3-ylmethyl)propanamide
2-{[4-(4-oxo-3,4-dihydro-2H-1-benzopyran-7-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}acetic acid
(2E)-1-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}-3-(3,4-dimethoxyphenyl)prop-2-en-1-one
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-[4-(morpholin-4-yl)-6-oxo-1,6-dihydropyridazin-1-yl]acetamide
4-(4-chlorophenoxy)-N-(3-methoxypropyl)piperidine-4-carboxamide
7-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
1-[(2-chlorophenyl)methyl]-3-{[(2,3-dihydroxypropyl)amino]methyl}-7-methoxy-1,2-dihydroquinolin-2-one
2-[(1-acetylpiperidin-4-yl)oxy]-N-[(2-aminopyridin-3-yl)methyl]-5-methoxybenzamide
[(3S,5R)-1-(1-ethyl-1H-pyrazole-3-carbonyl)-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
9-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-methyl-4-[3-(pyridin-2-yl)azetidin-1-yl]-6-(trifluoromethyl)quinoline
N-({4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-2,5-dimethoxybenzamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-1-(4-fluorophenyl)-2,2-dimethylcyclopropane-1-carboxamide
N-[(2-aminopyridin-3-yl)methyl]-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
1-[5-(2-chlorophenyl)furan-2-carbonyl]-3-(1H-imidazol-2-yl)piperidine
8-methoxy-N-[(1-methyl-1H-indol-3-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-amine
1-[2-methoxy-6-({[2-(pyridin-2-yl)ethyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1-cyclopentylpyrrolidin-2-one
1-[(1-methyl-1H-imidazol-2-yl)methyl]-N-[4-(3-methylphenyl)phenyl]piperidine-4-carboxamide
2-{5-[1-(4-chloro-1H-pyrazole-3-carbonyl)piperidin-4-yl]-1H-pyrazol-3-yl}acetic acid
N-{2-[(2-butyl-6-methylpyrimidin-4-yl)amino]ethyl}-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
11-(2-chloro-6-fluoro-3-methylbenzoyl)-3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecane
N,3-dimethyl-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]-1-propyl-1H-pyrazole-4-carboxamide
1-[(5-{[3-(methoxymethyl)piperidin-1-yl]methyl}-2,4-dimethylphenyl)methyl]-4-methylpiperazine
N-benzyl-N-methyl-3-{1-[3-(pyridin-2-yl)propanoyl]piperidin-4-yl}propanamide
[(1-methylpiperidin-4-yl)methyl](2-phenylethyl){[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}amine
N-[2-(dimethylamino)ethyl]-N-{[7-fluoro-2-(2-methylphenyl)quinolin-3-yl]methyl}-2,3-dimethoxybenzamide
2-[(8-methoxy-2H-chromen-3-yl)methyl]-2,8-diazaspiro[4.5]decane
3-{[1-(3-fluoropyridine-4-carbonyl)piperidin-4-yl]methyl}benzoic acid
5-[5-(4-methoxyphenyl)furan-2-carbonyl]-1-methyl-N-[2-(morpholin-4-yl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[4-(benzyloxy)piperidin-1-yl]-3-(3,5-dimethyl-1H-pyrazol-1-yl)propan-1-one
2-[({3-methoxy-2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amino]-1-phenylethan-1-ol
N-{3-[(3S)-3-aminopyrrolidine-1-carbonyl]-5-methylthiophen-2-yl}-2,2-dimethylpropanamide
3-({1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidin-4-yl}oxy)pyridine
1-(3-chlorobenzenesulfonyl)-3-{[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
N-[2-(pyrazin-2-yl)ethyl]-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamide
N-[(2-methoxyphenyl)methyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
{4-[(2-chloro-4-fluorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}(pyridin-3-yl)methanol
1-ethyl-4-{[3-(2-methoxyphenoxy)azetidin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
4-{8-methyl-3-[(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]imidazo[1,2-a]pyridine-2-carbonyl}morpholine
1-[(3R,4R)-4-cyclobutyl-4-hydroxy-3-methylpiperidin-1-yl]-2-(methylsulfanyl)ethan-1-one
1-cyclopentanecarbonyl-N-[(2S)-1-methoxy-3-phenylpropan-2-yl]piperidine-4-carboxamide
2-[1-(3-methylbut-2-en-1-yl)-4-{[3-(methylsulfanyl)phenyl]methyl}piperazin-2-yl]ethan-1-ol