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1-(1-cyclopropanecarbonylpiperidin-3-yl)-4-[3-(trifluoromethyl)phenyl]piperazine
2-[3-(cyclopropylmethyl)-5-[2-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)ethyl]-1H-1,2,4-triazol-1-yl]benzoic acid
{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[(1-methyl-1H-imidazol-2-yl)methyl]amine
1-(cyclobutylmethyl)-3-hydroxy-3-({[(5-methylfuran-2-yl)methyl]amino}methyl)piperidin-2-one
3-[(prop-2-en-1-yl)({[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl})amino]-1λ6-thiolane-1,1-dione
1-(2,2-dimethylpropyl)-4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidine
6-(4-fluorophenyl)-N-methyl-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}imidazo[2,1-b][1,3]thiazole-3-carboxamide
5-(2,6-difluoro-4-methoxyphenyl)-3-[2-(methylsulfanyl)ethyl]-1-propyl-1H-1,2,4-triazole
3-[N-(2-phenylethyl)-1-quinoxalin-5-ylformamido]propanamide
3-methyl-1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)piperidin-3-ol
N-(3-acetylphenyl)-4-[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
methyl (2S,4R)-1-[(3-methoxyphenyl)methyl]-4-{2-[4-(trifluoromethyl)phenyl]benzamido}pyrrolidine-2-carboxylate
3-[4-(3-methylphenyl)piperazin-1-yl]-N-(1-propanoylazepan-3-yl)propanamide
1-[2-(dimethylamino)ethyl]-N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-5-oxopyrrolidine-3-carboxamide
(3E)-1-{1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}pent-3-en-1-one
4-(2-methoxy-2-phenylacetyl)-1-(2-methoxyphenyl)piperazin-2-one
N-(2H-1,3-benzodioxol-5-yl)-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carboxamide
3-(5-{[4-(4-amino-5-methylpyrimidin-2-yl)piperazin-1-yl]methyl}thiophen-2-yl)prop-2-yn-1-ol
1-(4-methylphenyl)-3-(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)urea
2-(3-{7-ethyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl}phenoxy)acetamide
N-[2-({2-amino-3-ethyl-3H-imidazo[4,5-b]pyridin-6-yl}formamido)ethyl]-4-fluorobenzamide
6-cyclopropyl-N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]pyrimidin-4-amine
5-{[benzyl(methyl)amino]methyl}-N-{spiro[2.5]octan-1-ylmethyl}-1,2-oxazole-3-carboxamide
6-fluoro-N,N-dimethyl-2-[1-(2-methylpyridin-4-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
N-[(1-benzylpiperidin-4-yl)methyl]-N-methylspiro[2.3]hexane-1-carboxamide
6-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-N-propylpyridine-3-carboxamide
8-[3-(1H-1,2,3-benzotriazol-1-yl)propanoyl]-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
(2R,3S,6R)-3-phenyl-5-(pyridine-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-{5-[1-(1-methyl-1H-imidazole-2-carbonyl)pyrrolidin-2-yl]thiophene-2-carbonyl}piperidin-4-ol
4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)-1-pentylpiperidine
ethyl 1-(2-methoxy-5-methylbenzenesulfonyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
5-[(4-{octahydro-1H-pyrido[1,2-a]piperazine-2-carbonyl}-1,3-oxazol-2-yl)methoxy]isoquinoline
methyl (2S,4S,5R)-2-ethyl-5-(4-fluorophenyl)-1-methyl-4-(1,2-oxazinane-2-carbonyl)pyrrolidine-2-carboxylate
3-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
1-[(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)sulfonyl]-4-(hydroxymethyl)piperidin-4-ol
(2S,4S)-1-{[4-(benzyloxy)-3-methoxyphenyl]methyl}-N-[2-(2-methoxyphenyl)ethyl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
4-({3-[5-(trifluoromethyl)-1H-1,2,4-triazol-3-yl]phenyl}methyl)morpholine
8-(3-methyl-4-oxo-3,4-dihydroquinazoline-7-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
3-fluoro-5-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine-1-carbonyl)pyridine
1-methyl-4-(morpholine-4-sulfonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(2-fluoro-6-methoxyphenyl)-1,3-thiazole-4-carboxamide
2-{4-[4-methyl-2-(methylamino)-1,3-thiazole-5-carbonyl]morpholin-3-yl}-N-phenylacetamide
1-(2-aminoethyl)-N-[(1-propyl-1H-imidazol-2-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
5-({[(3-{2-[4-(3,4-difluorobenzenesulfonyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)amino}methyl)pyrrolidin-2-one
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylcyclopent-1-ene-1-carboxamide
3-(5-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)-1-(pyrrolidin-1-yl)propan-1-one
1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-methylpiperidin-3-ol
N-[3-({[2-(2-ethyl-1H-imidazol-1-yl)ethyl]carbamoyl}amino)-2-methylphenyl]-2-methoxyacetamide
2-[2-(4-fluorophenyl)morpholin-4-yl]-N-(pyridin-2-ylmethyl)acetamide
4-(4-fluoro-3-methylbenzoyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one