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1-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(4-methyl-1H-pyrazol-1-yl)ethan-1-one
2-(3-chloro-4-methoxyphenyl)benzamide
4-{1-[1-(1H-imidazol-4-ylmethyl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
N,N-diethyl-1-({4-[(6-methylpyridin-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidine-3-carboxamide
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]acetamide
2-fluoro-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-5-sulfamoylbenzamide
1-[1-(2-methylpropyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
N-benzyl-2-(methylamino)-N-[(6-methylpyridin-2-yl)methyl]acetamide
1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
3-(5-{2-[2-(2,2-dimethyloxan-4-yl)-1H-imidazol-1-yl]ethyl}-1H-1,2,4-triazol-3-yl)pyridine
N2-[(3-methylphenyl)methyl]-N2-(propan-2-yl)pyrrolidine-1,2-dicarboxamide
2-(2-acetylphenyl)-6-methylpyridine-3-carbonitrile
5-{[(1S,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-N,N-dimethylfuran-2-carboxamide
4-(2-fluoro-5-methylphenoxy)-1-(1H-imidazol-2-ylmethyl)piperidine-4-carboxylic acid
6-fluoro-4-[2-(pyrrolidine-1-carbonyl)morpholine-4-carbonyl]-1,2-dihydroquinolin-2-one
1-cyclobutyl-4-[(4-cyclopentyl-1H-1,2,3-triazol-1-yl)methyl]piperidine
3-[(2-fluorophenyl)formamido]-N-[2-(piperidin-1-yl)ethyl]propanamide
[(3S,5S)-1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-5-[(4-methyl-1,4-diazepan-1-yl)methyl]piperidin-3-yl]methanol
6-ethyl-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methylpyrimidin-4-amine
1-ethyl-5-[methyl(thiophen-3-ylmethyl)amino]-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}acetamide
1-(4-ethylpiperazin-1-yl)-3-[3-({methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]propan-2-ol
6-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-2,3-dihydropyridazin-3-one
3-{[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]sulfonyl}-N-[2-(1H-imidazol-1-yl)ethyl]benzamide
1-benzyl-4-oxo-5-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-N-(prop-2-en-1-yl)-1,4-dihydropyridine-3-carboxamide
4-(3-methoxyphenyl)-2-methyl-1H-imidazole
1-[(4-chlorophenyl)methyl]-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-3-amine
(3aR,6aR)-2-benzyl-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[5-(1-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H-imidazol-2-yl)-1,3-thiazol-2-yl]morpholine
3-[2-(5-ethyl-1,2,4-oxadiazol-3-yl)ethyl]-1-(2-fluoro-5-methanesulfonamidophenyl)urea
methyl 2-[4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]pyridine-3-carboxylate
1-(4-{[(2,6-difluoro-3-methoxyphenyl)methyl]amino}-2-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-(pyridin-3-yl)acetamide
3-(3,4-diethyl-1-methyl-1H-pyrazol-5-yl)-1-[(dimethyl-1,2-oxazol-4-yl)methyl]-1-methylurea
1-{2-[3-methyl-1-(naphthalen-1-yl)-1H-1,2,4-triazol-5-yl]ethyl}pyrrolidin-2-one
1-(4-chlorophenyl)-N-({1-[3-(pyrazin-2-yl)propanoyl]piperidin-3-yl}methyl)cyclopropane-1-carboxamide
(1S,5R)-6-(cyclopropylmethyl)-3-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
(1R,6S)-3-[5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-9-methyl-3,9-diazabicyclo[4.2.1]nonane
2-{[(5,6-dimethylpyrimidin-4-yl)(methyl)amino]methyl}-2-ethylbutan-1-ol
2-{[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]methyl}-4,6-dimethylphenol
2-ethyl-4-[4-(1H-imidazol-1-yl)benzoyl]-1-(propan-2-yl)piperazine
(1S,4S)-5-[(2-hydroxy-3-methoxyphenyl)methyl]-2-[2-(methylsulfanyl)phenyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
(3-chlorophenyl)[1-(2-methoxyphenyl)-3-methyl-1H-1,2,4-triazol-5-yl]methanol
(4aS,8aR)-1-(2-aminoethyl)-6-[(5-fluoro-1-methyl-1H-indol-3-yl)methyl]-decahydro-1,6-naphthyridin-2-one
(1R,9aR)-1-({[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]amino}methyl)-octahydro-1H-quinolizin-1-ol
1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-4-(pyrimidin-2-yl)-1,4-diazepane
2-(5-fluoro-2-methylphenyl)-1-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
1-[2-(4-chloro-2-methylphenoxy)propanoyl]-4-[(4-methoxyphenyl)methyl]-1,4-diazepan-5-one
3-{1-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]-1H-1,2,3-triazol-4-yl}benzonitrile