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(2,1,3-benzothiadiazol-5-ylmethyl)(ethyl){[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}amine
3-{[(1-hydroxybutan-2-yl)(thiophen-3-ylmethyl)amino]methyl}phenol
(3R,5S)-5-{4-[3-(4-fluorophenoxy)propyl]piperazine-1-carbonyl}pyrrolidin-3-amine
3,5-dimethyl-4-{[4-phenyl-5-(1-propyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]methyl}-1,2-oxazole
7-(2-aminoethyl)-2-(furan-2-yl)-N-(3-methoxypropyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(2S)-N-[3-(3-methylphenyl)phenyl]-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]pyrrolidine-2-carboxamide
3-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-5-fluorobenzonitrile
4-amino-1-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]butan-1-one
(2R,3R,6R)-3-(2-methoxyphenyl)-5-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
1-butyl-4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperazine
3-{[(1-ethoxy-2-methylpropan-2-yl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
4-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-2-(piperidin-1-ylmethyl)-1,4-oxazepane
4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1H-imidazol-2-ylmethyl)piperidine
5-(oxolan-2-yl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}thiophene-2-carboxamide
methyl (2S)-1-(4-{[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carbonyl)pyrrolidine-2-carboxylate
(2S,4R)-N-ethyl-4-(5-methoxyfuran-2-amido)-1-(pyridin-2-ylmethyl)pyrrolidine-2-carboxamide
N,N-dimethyl-2-{[(1,3-thiazol-2-yl)amino]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
N-benzyl-3-({1-[3-(1H-pyrazol-1-yl)propyl]piperidin-4-yl}oxy)benzamide
N-{4-[4-(4-formyl-1,4-diazepan-1-yl)piperidin-1-yl]phenyl}-3-phenylpropanamide
(3aR,6aS)-5-(2,3-dihydro-1H-indene-5-carbonyl)-2-ethyl-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
methyl[(2-methyl-1,3-oxazol-4-yl)methyl]{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
N-(isoquinolin-5-ylmethyl)-N,2-dimethyl-6-(piperidin-3-yl)pyrimidin-4-amine
1-[(2-methylphenyl)methyl]-4-[2-(1H-pyrazol-1-yl)benzoyl]piperazine
dimethyl({4-[1-(1-methyl-1H-pyrazole-3-carbonyl)piperidin-2-yl]phenyl}methyl)amine
(2S,4S)-1-[(4-chlorophenyl)methyl]-4-{[(3,4-difluorophenyl)methyl]amino}-N-ethylpyrrolidine-2-carboxamide
N'1-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)cyclopropane-1,1-dicarboxamide
ethyl 4-(3-propyl-1H-pyrazole-5-carbonyl)piperazine-1-carboxylate
N-methyl-2-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyridine-3-carboxamide
5-methyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-1H-pyrazole-3-carboxamide
N-(3,4-dimethylphenyl)-1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidin-3-amine
9-(4-methoxypyrimidin-2-yl)-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[2-(1-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethyl]pyridine
(1R,5S,8S)-8-methoxy-3-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-3-azabicyclo[3.2.1]octane
methyl 6-(butan-2-yl)-2-{[(3-chlorophenyl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-{4-[1-(2H-1,3-benzodioxol-5-ylmethyl)-1H-imidazol-2-yl]phenyl}acetamide
{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}(methyl)[(1-methylpyrrolidin-2-yl)methyl]amine
4-(1-{4-[3-(pyrrolidin-1-yl)pyrazin-2-yl]phenyl}ethyl)morpholine
2-(3-fluorophenyl)-8-methoxy-5-[(6-methylpyridin-2-yl)methyl]-2,3,4,5-tetrahydro-1,5-benzothiazepine
2-amino-3-ethyl-N-{[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-3H-imidazo[4,5-b]pyridine-6-carboxamide
1-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-4-(4-phenyl-1H-pyrazol-5-yl)piperidine
(3R)-1-(5-chloro-3-phenyl-1H-indole-2-carbonyl)pyrrolidin-3-ol
N-[1-(1,3-thiazol-2-yl)ethyl]-5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
N-(1-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2,2-dimethylpropanamide
4-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-2-oxoethyl}-3,4-dihydro-2H-1,4-benzothiazin-3-one
4-(2-ethyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-7-fluoro-1,2-dihydroquinolin-2-one
methyl (2S,4R)-4-(5-chloro-3-phenyl-1H-indole-2-amido)-1-[(2-methylphenyl)methyl]pyrrolidine-2-carboxylate
methyl 1-[(3S,5S)-5-{[2-(3-chlorophenyl)ethyl]carbamoyl}-1-[(4-ethoxyphenyl)methyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-ethyl-N-methyl-6-[methyl({[4-(1H-pyrazol-1-yl)phenyl]methyl})amino]pyridine-3-carboxamide
N-ethyl-4-methyl-5-{2-[2-(thiophen-2-yl)ethyl]piperidine-1-carbonyl}-1,3-thiazol-2-amine
3-(furan-2-yl)-1-{7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}propan-1-one