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N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-6-methylpyridazin-3-amine
N-{2-[1-(furan-2-ylmethyl)piperidin-3-yl]ethyl}pyrimidine-5-carboxamide
N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
1-cyclohexyl-N3,N5-dimethyl-4-oxo-N3-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
4-[1-(2-hydroxyethyl)-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-5-yl]-N,N-dimethylpiperidine-1-carboxamide
5-chloro-N-{2-[(pyridin-3-yl)amino]ethyl}pyridine-2-carboxamide
(3S)-1-(4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzoyl)pyrrolidin-3-amine
6-fluoro-N,2-dimethyl-N-(prop-2-yn-1-yl)quinoline-4-carboxamide
1-(1H-indazol-5-yl)-3-[3-(2-oxopyrrolidin-1-yl)propyl]urea
(2E)-3-(pyridin-2-yl)-1-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}prop-2-en-1-one
3-(3-chloro-5-fluorophenyl)-1-{3-[3-(hydroxymethyl)piperidin-1-yl]propyl}urea
4-{2-[3-cyclopropyl-1-(3-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
3-methoxy-N-[1-(2-phenylethyl)piperidin-3-yl]propanamide
1-(1-cyclopentylpiperidin-3-yl)-4-(2-methoxyphenyl)piperazine
5-methyl-2-(3-{[4-(pyrrolidin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)pyrimidin-4-amine
8-[(3-methoxyphenyl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-tert-butyl-4-{6-[(propan-2-yl)amino]pyridazin-3-yl}benzene-1-sulfonamide
3-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}benzonitrile
4-benzyl-1-(2-chloropyridine-4-carbonyl)-3-ethyl-1,4-diazepan-5-one
(4aS,8aS)-2-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}-decahydroisoquinolin-4a-ol
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-(naphthalen-1-yl)pyridine-3-carboxamide
(3S,5S)-1-(2,3-dihydro-1H-inden-2-yl)-5-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-N-[(4-methoxy-2,5-dimethylphenyl)methyl]pyrrolidin-3-amine
N-benzyl[(2-fluoro-5-methylphenyl)amino]sulfonamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N-methylpiperidin-3-amine
(3aR,6aS)-5-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(2S)-3-(1H-imidazol-4-yl)-1-[4-(morpholin-4-ylmethyl)piperidin-1-yl]-1-oxopropan-2-yl]acetamide
(1R,3S)-3-(2-aminoethoxy)-7-(4-ethyl-5-methylthiophene-3-carbonyl)-7-azaspiro[3.5]nonan-1-ol
1-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperidine-4-carboxamide
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-ethyl-N-(2-methylprop-2-en-1-yl)acetamide
N4-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-N1,N1-dimethylpiperidine-1,4-dicarboxamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-(1-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-4-yl)propanamide
3-{[1-(1,4-dioxan-2-ylmethyl)-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-4-methyl-1,2,5-oxadiazole
3-(4-ethyl-1,3-dimethyl-1H-pyrazol-5-yl)-1-(pyridin-4-ylmethyl)urea
4-(2-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethyl)morpholine
2-[2-({2-amino-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}amino)ethyl]-6-phenyl-2,3,4,5-tetrahydropyridazin-3-one
4-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl}-1-(2-methylpropyl)piperidine
1-[4-(4-methoxybenzoyl)piperazin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
2-{2-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
2-[4-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl]ethan-1-ol
1-methyl-3-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]-1,2-dihydroquinolin-2-one
N-[(4-methoxyphenyl)methyl]-4-methyl-5-{1-[3-(6-methylpyridin-2-yl)propyl]-1H-pyrazol-3-yl}-1,3-thiazol-2-amine
5-[(isoquinolin-5-yloxy)methyl]-N-(2-methoxyethyl)-N-methyl-1,2-oxazole-3-carboxamide
1-{2-[methyl(pyridin-2-ylmethyl)amino]acetyl}-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
N,N-dimethyl-3-[4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]aniline
(3S,4R)-1-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
1-(1H-1,2,3-triazole-5-carbonyl)-4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazine
3-{[4-fluoro-3-(trifluoromethyl)phenyl]methyl}-1,3-oxazolidin-2-one
2-(2-fluorophenyl)-2-(4-hydroxy-4-phenylpiperidin-1-yl)acetic acid
1-(2-{2-[2-(pyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}phenyl)ethan-1-one
[(3R,5R)-1-[1-(methoxymethyl)cyclopropanecarbonyl]-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol