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5-{[benzyl(methyl)amino]methyl}-N,N-dimethyl-1,2-oxazole-3-carboxamide
(3S,4S)-4-(1H-imidazol-2-yl)-1-(3,4,7-trimethyl-1H-indole-2-carbonyl)pyrrolidine-3-carboxylic acid
2,2-diphenyl-1-{4-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}ethan-1-ol
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-N-methyl-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
methyl 3-(2-methoxyacetamido)-5-[(5-methylhex-5-en-2-yl)amino]-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-(hydroxymethyl)-1-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-3-ol
4,6-dimethyl-3-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
methyl 1-[6-(2-methylphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperidine-2-carboxylate
N,N-diethyl-2-[3-(furan-2-yl)-1-(2-methoxyphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]acetamide
methyl 3-(2-cyclopentylacetamido)-6-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-ylmethyl)thieno[2,3-b]pyridine-2-carboxylate
1-[4-(6-methylpyridin-2-yl)piperazin-1-yl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
({4-[(8-methoxyquinolin-2-yl)methyl]-1,4-oxazepan-6-yl}methyl)dimethylamine
5-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-2-methyl-1,4-dihydropyridin-4-one
4-(5-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl)morpholine
[(3-methyl-1-{2-[4-(pyrrolidin-1-yl)piperidin-1-yl]ethyl}-1H-pyrazol-4-yl)methyl](2-methylprop-2-en-1-yl)amine
1-cyclopentyl-4-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}piperazin-2-one
2-(1,4-dimethylpiperazin-2-yl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}acetamide
N-(thiophen-3-ylmethyl)-1H-indazole-3-carboxamide
1-(carbamoylmethyl)-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]piperidine-3-carboxamide
1-(3-methylbutyl)-3-(propan-2-yl)-8-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(3-fluorophenyl)-3-{2-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]-2-oxoethyl}-1-(pyridin-3-ylmethyl)pyrrolidine-2,5-dione
N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
1-cyclopropanecarbonyl-4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
4-{4-[(4-methylpyrimidin-2-yl)amino]piperidin-1-yl}-1λ6-thiane-1,1-dione
[2-methoxy-1-(pyridin-2-yl)ethyl](methyl)(quinolin-4-ylmethyl)amine
1-{1-[(2-chlorophenyl)methyl]piperidin-4-yl}-4-(pyrrolidine-1-carbonyl)piperidine
4-{[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}thiomorpholine
N-{[1-(3,5-dimethylphenyl)cyclopentyl]methyl}-5-methoxy-4-oxo-1,4-dihydropyridine-2-carboxamide
2-cyclopropyl-N-[1-(pyridin-3-yl)propan-2-yl]-1,3-benzoxazole-6-carboxamide
(3R,4R)-N-cyclohexyl-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidine-1-carboxamide
5-(1-{4-[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]-1H-1,2,3-triazol-1-yl}ethyl)-1,3,4-thiadiazol-2-amine
1-(4-fluorophenyl)-N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}cyclopropane-1-carboxamide
3-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propanamide
2-(2-{5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-6-yl}ethyl)-6-phenyl-2,3,4,5-tetrahydropyridazin-3-one
5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1,2-oxazole-3-carboxamide
3-{4-[(dimethylamino)methyl]-4-hydroxyazepane-1-carbonyl}-4,6-dimethyl-1,2-dihydropyridin-2-one
1-{1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-3-yl}-4-(4-methoxyphenyl)piperazine
1-{2-[3-(2-fluorophenoxy)azetidin-1-yl]-2-oxoethyl}-3-methyl-1,2-dihydroquinoxalin-2-one
N-phenyl-5-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)pyridin-2-amine
2-methyl-N-[(4-sulfamoylphenyl)methyl]-1,3-benzoxazole-6-carboxamide
4-[4-(piperidine-1-carbonyl)phenoxy]-1-(1,3-thiazol-2-ylmethyl)piperidine
ethyl 4-{[3-(2-hydroxyethyl)-4-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-1-yl]methyl}-1H-pyrazole-3-carboxylate
1-{2-[2-(dimethylamino)ethyl]morpholin-4-yl}-4,4,4-trifluorobutan-1-one
3-(4-fluorophenyl)-4-(thiophen-3-ylmethyl)piperazin-2-one
N-(2-methoxyethyl)-2-{2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}-N-(thiophen-3-ylmethyl)acetamide
2-(methylamino)-N-[(2E)-3-phenylprop-2-en-1-yl]-N-propylpyridine-4-carboxamide
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-(3-chloro-1,2-oxazol-5-yl)propanamide
N-[(3R,5S)-5-(ethylcarbamoyl)-1-[(2E)-3-phenylprop-2-en-1-yl]pyrrolidin-3-yl]-1H-pyrrole-2-carboxamide
1-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-(pyridin-4-yl)propan-1-one
4-(1,3-dimethyl-1H-indole-2-carbonyl)-1-(4-methylphenyl)piperazin-2-one