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[(3R,4R)-1-[(1-benzyl-1H-indol-6-yl)methyl]-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
2-{[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-5-(piperazin-1-yl)-2,3-dihydropyridazin-3-one
(1R,3S)-7-(cyclopropanesulfonyl)-3-methoxy-3-methyl-7-azaspiro[3.5]nonan-1-ol
dimethyl(1-{1-[(1-methyl-1H-indol-6-yl)methyl]piperidin-4-yl}ethyl)amine
3-(1H-1,2,3-benzotriazol-1-yl)-1-[2-(3-methoxyphenyl)pyrrolidin-1-yl]propan-1-one
3-[(4-hydroxyazepan-1-yl)sulfonyl]-N-(oxan-4-ylmethyl)benzamide
2-{[5-(1,2-oxazol-5-yl)furan-2-yl]sulfonyl}-2,8-diazaspiro[4.5]decane
3-{2-[2-(1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}-2,6-dimethylquinoline
4-hydroxy-N-[(2E)-3-phenylprop-2-en-1-yl]-N-propyl-2-(thiophen-2-yl)pyrimidine-5-carboxamide
3-ethoxy-1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
2-amino-N-methyl-4-phenyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)pyrimidine-5-carboxamide
2-[1'-(5-cyclobutyl-1,3,4-oxadiazol-2-yl)-2-oxo-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-1-yl]acetamide
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-N-(2-methoxyphenyl)piperidine-1-carboxamide
1-(4-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
(1-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}-3-(thiophen-2-yl)-1H-pyrazol-4-yl)methanol
4,6-dimethyl-2-oxo-N-[4-(pyridin-2-yl)butyl]-1,2,3,4-tetrahydropyrimidine-5-carboxamide
N-cyclohexyl-4-(4-{[(3R)-3-hydroxypyrrolidin-1-yl]methyl}-1H-1,2,3-triazol-1-yl)piperidine-1-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(propan-2-ylsulfanyl)acetamide
2-{4-[(3-fluorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}pyridine-3-carbonitrile
N-({1-[(3S,5S)-5-(ethylcarbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazol-4-yl}methyl)pyridine-4-carboxamide
2-(1H-indol-3-yl)-1-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
1-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
4-[4-(dimethylamino)phenyl]-1-phenyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-1-[3-(3-methyl-2-oxoimidazolidin-1-yl)phenyl]urea
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-(3,5-dimethyl-1H-pyrazol-4-yl)propan-1-one
9-[2-(4-methyl-1H-pyrazol-1-yl)acetyl]-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-{[2-(cyclopentanesulfonyl)-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}-4-methoxypiperidine
N-(3-ethoxyphenyl)-2-[4-(4-methylpiperazin-1-yl)-6-oxo-1,6-dihydropyridazin-1-yl]acetamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-[(2-hydroxyethyl)amino]pyridine-3-carboxamide
N-[3-(1H-imidazol-1-yl)propyl]-2-methyl-N-(pyridin-3-ylmethyl)imidazo[1,2-a]pyridine-6-carboxamide
1-(furan-3-ylmethyl)-4-[4-(oxolan-2-ylmethyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]piperidine
3-(2-methoxyethyl)-1-[4-(4-methyl-4H-1,2,4-triazol-3-yl)phenyl]-3-[(5-methylthiophen-2-yl)methyl]urea
(1R,3S)-7-[4-(dimethylamino)benzoyl]-7-azaspiro[3.5]nonane-1,3-diol
1-(morpholin-4-yl)-2-[(1R,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-({[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}methyl)piperidin-2-one
N-[3-(5-chloro-1H-1,3-benzodiazol-2-yl)propyl]-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-amine
2-[4-(2-amino-6-methylpyrimidin-4-yl)-1H-pyrazol-1-yl]-N-(1-methyl-1H-indazol-3-yl)acetamide
N-{[1-(1H-1,3-benzodiazol-2-ylmethyl)pyrrolidin-3-yl]methyl}-3-methylpyridine-4-carboxamide
1-ethyl-5-{[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1H-1,2,4-triazole
2-(2-benzyl-1,3-thiazole-4-carbonyl)-2,3-dihydro-1H-isoindole
N-benzyl-1-{2-[(2,3-dimethoxyphenyl)formamido]ethyl}-1H-1,2,3-triazole-4-carboxamide
N'-[3-(2-hydroxyphenyl)propyl]-N-[2-(propan-2-yl)phenyl]butanediamide
[2-({1-[(1,4-dimethyl-1H-pyrazol-5-yl)methyl]piperidin-4-yl}oxy)ethyl]dimethylamine
methyl 3-[(2-ethoxyphenyl)methyl]-7-oxo-9-[3-(pyridin-3-yl)propoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-(1-{1-[(2-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-phenoxypropanamide
4-(2,2-dimethyloxane-4-carbonyl)-7-{[4-(4-fluorophenyl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-(pyrrolidine-1-carbonyl)piperidine
3-(4-methoxyphenyl)-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-3-phenylpropanamide
3-(2-phenylethyl)-5-[3-(propan-2-yl)-1H-pyrazol-5-yl]-1H-1,2,4-triazole
5-[5-(2,3-dihydro-1H-inden-2-yl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine