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N-{[3-(2H-1,3-benzodioxol-5-ylmethoxy)phenyl]methyl}-3-(2-oxopyrrolidin-1-yl)-N-(pyridin-2-ylmethyl)benzamide
4-amino-1-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}butan-1-one
methyl({4-methyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)[(5-methylthiophen-2-yl)methyl]amine
3-{1-[5-(3-chlorophenyl)-1,2,4-triazin-3-yl]piperidin-3-yl}propan-1-ol
6-(2,4-dimethoxyphenyl)pyrazine-2-carboxylic acid
N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]-1-benzofuran-5-carboxamide
8-methyl-2-propyl-N-(1,3-thiazol-2-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxamide
(3S,4R)-1-[4-(prop-2-en-1-yl)benzoyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
N-[(5-ethylpyridin-2-yl)methyl]-3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-N-methylpropanamide
2-[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenoxy]-5-(trifluoromethyl)pyridine
2-(1-propyl-1H-imidazol-2-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-(2-phenylethyl)-6-(3-phenylprop-2-ynoyl)-6-azaspiro[2.5]octane-1-carboxamide
N-[2-(5-methylfuran-2-yl)ethyl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
N-cyclopropyl-1-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}piperazine-2-carboxamide
(3S,4R)-1-{[2-(benzylsulfanyl)pyrimidin-5-yl]methyl}-3-ethyl-4-methylpiperidin-4-ol
3-[1-({1-[(2-fluorophenyl)methyl]-2-(propane-2-sulfonyl)-1H-imidazol-5-yl}methyl)pyrrolidin-2-yl]-4-methyl-1,2,5-oxadiazole
N-(1,3-dihydroxy-2-methylpropan-2-yl)-2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]acetamide
methyl 3-({4-[1-(2-hydroxyethyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}methyl)benzoate
N4-methyl-N6-(propan-2-yl)-N4-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}pyrimidine-2,4,6-triamine
6-[(1R,5S,8R)-8-methoxy-3-azabicyclo[3.2.1]octane-3-carbonyl]-1,2,3,4-tetrahydroquinoxaline-2,3-dione
methyl 3-(2-chlorobenzamido)-5-{[(1-methylpiperidin-2-yl)formamido]methyl}benzoate
N-(2-methoxyethyl)-5-oxo-1-(pyridin-3-ylmethyl)-N-(thiophen-3-ylmethyl)pyrrolidine-3-carboxamide
(1-{[2-(trifluoromethoxy)phenyl]methyl}pyrrolidin-3-yl)methanamine
methyl 2-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-1-oxo-1,2-dihydroisoquinoline-7-carboxylate
2-(4-amino-3-fluorophenyl)-2-(azocan-1-yl)acetic acid
(3R,4S)-4-cyclopropyl-1-(1H-indole-6-carbonyl)pyrrolidin-3-amine
1-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
N-{[1-(2,2,6,6-tetramethylpiperidin-4-yl)pyrrolidin-3-yl]methyl}thiophene-3-carboxamide
1-[2-(2-phenylethyl)morpholine-4-carbonyl]cyclopropane-1-carboxamide
4-{9-oxo-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraene-10-carbonyl}-1λ6-thiomorpholine-1,1-dione
2-{4-[2-amino-3-cyano-6-(1-methyl-1H-pyrrol-2-yl)pyridin-4-yl]phenoxy}propanoic acid
2-{[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]methyl}phenol
1-{[({3-[2-hydroxy-3-(morpholin-4-yl)propoxy]phenyl}methyl)amino]methyl}cyclohexan-1-ol
6-fluoro-2-{[4-hydroxy-4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}quinolin-4-ol
3-{[4-hydroxy-4-(pyrrolidin-1-ylmethyl)piperidin-1-yl]methyl}-7-methoxy-1,2-dihydroquinolin-2-one
5-(methoxymethyl)-N-{[7-(quinolin-7-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}furan-2-carboxamide
5-[7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]-N-ethyl-4-methyl-1,3-thiazol-2-amine
7-chloro-4-{[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-{1-[(4,5-dimethylfuran-2-yl)methyl]piperidin-4-yl}-3-(pyrrolidine-1-carbonyl)piperidine
2-ethyl-6-[1-(1-methyl-1H-indazole-3-carbonyl)piperidin-4-yl]-3,4-dihydropyrimidin-4-one
N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]-1,2,3,4-tetrahydroisoquinoline-2-sulfonamide
methyl 4-(5-{[4-(morpholine-4-carbonyl)piperidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
(3aS,6aS)-2-acetyl-5-[(2,5-dimethylthiophen-3-yl)sulfonyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-methyl-N-(2-{4-[(4-phenylpiperidin-1-yl)methyl]phenoxy}propyl)thiophene-2-carboxamide
methyl 4-[(4-{5-[3-(trifluoromethyl)phenyl]pyrimidin-4-yl}piperidin-1-yl)methyl]benzoate
4-(1H-imidazol-2-yl)-1-(3-phenyl-1,2-oxazole-5-carbonyl)piperidine
(2S,4R)-4-amino-1-(6-chloro-2-methylquinoline-4-carbonyl)-N,N-diethylpyrrolidine-2-carboxamide
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
(2R,3R,6R)-3-phenyl-5-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
N-cyclohexyl-3-{[2-(pyridin-3-yl)pyrimidin-5-yl]formamido}propanamide