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3-amino-2-methyl-N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}propanamide
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-ethyl-4-{[(4-methoxy-3-methylphenyl)methyl]amino}pyrrolidine-2-carboxamide
2-{[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]amino}-N-(1,3-thiazol-2-yl)propanamide
2-fluoro-N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}-5-sulfamoylbenzamide
5-(dimethylamino)-1-methyl-N-[(5-methylfuran-2-yl)methyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[2-(1H-imidazol-1-yl)-1-phenylethyl]amine
N-[3-hydroxy-2-(thiophen-2-ylmethyl)propyl]-4-methyl-2-phenylpyrimidine-5-carboxamide
N-(furan-2-ylmethyl)-2-methyl-N-(2-phenylethyl)-1,3-thiazole-4-carboxamide
2,5-dimethyl-3-(4-{2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}piperazin-1-yl)pyrazine
1-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-(propan-2-yloxy)ethan-1-one
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-methyl-N-(pyrimidin-4-ylmethyl)-1H-pyrazole-3-carboxamide
2-benzyl-8-{[2-(2-hydroxyethoxy)phenyl]methyl}-2,8-diazaspiro[4.5]decan-3-one
(2R,6R)-4-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
4-(3-methylphenoxy)-1-[(2E)-3-phenylprop-2-en-1-yl]piperidine-4-carboxylic acid
1-[(3R,4S)-3-amino-4-(4-methoxyphenyl)pyrrolidin-1-yl]-2-[4-(methylsulfanyl)phenyl]ethan-1-one
7-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepine-3-carbonyl)-3-methyl-3,4-dihydroquinazolin-4-one
1-({2-[3-(3-methylpiperidin-1-yl)propoxy]phenyl}methyl)azetidin-3-ol
3-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]quinoline
3-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-1-(pyrrolidin-1-yl)propan-1-one
2-(3-methyl-4-{[4-(piperidine-1-carbonyl)piperidin-1-yl]methyl}-1H-pyrazol-1-yl)ethan-1-ol
1-(4-cyano-2-ethylphenyl)-3-(oxolan-3-yl)urea
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
(3S,4S)-4-(4-fluorophenyl)-1-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidin-3-ol
4-(azepan-1-yl)-5-methyl-N-(thiophen-3-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-5-(propan-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-ethyl-1-methyl-4-(3-phenylpropyl)piperazine
1-(2-methyl-1,3-thiazole-5-carbonyl)-2-[2-(thiophen-2-yl)ethyl]piperidine
1-[1'-(isoquinolin-1-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-1H-pyrrole-2-carboxamide
(2R,3R,6R)-3-(4-fluorophenyl)-5-(1-methyl-1H-pyrrole-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N4-[(1-phenylcyclopentyl)methyl]-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
3-[(1-acetylpiperidin-4-yl)oxy]-N-[(2,5-difluorophenyl)methyl]-4-methoxybenzamide
(4aR,7aS)-1-propyl-4-[3-(1H-pyrazol-1-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-methoxy-N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N-methylpyrimidin-4-amine
(1-{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)(phenyl)methanol
4-[2-(ethylamino)pyrimidin-5-yl]-1-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[2-(ethylsulfanyl)ethyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
N'-(adamantan-1-yl)-N-[1-(1H-pyrazol-1-yl)propan-2-yl]propanediamide
N-methyl-N-[(2-methylpyridin-4-yl)methyl]-4-(propan-2-yl)pyrimidin-2-amine
1-{4-[(4-chlorophenyl)methyl]piperazin-1-yl}-4-(1H-1,2,4-triazol-1-yl)butan-1-one
(2S,4S)-4-amino-N-methyl-1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)pyrrolidine-2-carboxamide
N-(3-hydroxypropyl)-N-methyl-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
7-fluoro-3-{7-oxo-1H,5H,6H,7H,8H-pyrido[3,2-f]indazol-5-yl}-1,2-dihydroquinolin-2-one
N-{[1-(morpholin-4-yl)cyclohexyl]methyl}thian-4-amine
5-[3-(1H-pyrazol-1-yl)benzoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
N-[(3-fluorophenyl)methyl]-N-[(4-methoxyphenyl)methyl]-3-(1H-pyrazol-1-yl)propanamide
3-[1-(diethylsulfamoyl)piperidin-3-yl]benzoic acid
N-[2-(dimethylamino)-2-(5-methylfuran-2-yl)ethyl]-3-(4-hydroxyphenyl)benzamide
4-(2-chlorophenoxy)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine
({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}methyl)(furan-2-ylmethyl)(prop-2-en-1-yl)amine