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ethyl 4-[(4-chlorophenyl)methyl]-1-cyclopentylpiperidine-4-carboxylate
N-{1-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]piperidin-4-yl}methanesulfonamide
1-[(4-ethylphenyl)methyl]-4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
4-[(5-cyclohexylthiophen-2-yl)methyl]morpholine-2-carboxamide
N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-5-propylthiophene-3-carboxamide
N-(1,4-dioxan-2-ylmethyl)-4-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
1-{4-[5-(azepan-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(propan-2-yloxy)ethan-1-one
2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-4-methylphenyl]-5-methylpyrimidin-4-amine
(3aR,6aR)-2-cyclopentyl-5-[(2-hydroxy-6-methoxyphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-ethyl-N-(pyridin-4-ylmethyl)benzamide
2-{5-[2-(6-methylpyridin-2-yl)-1H-imidazol-1-yl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
3-methyl-1-{4-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}butan-1-one
1-(4-{1H-pyrazolo[3,4-b]pyridin-1-yl}thiophen-2-yl)ethan-1-one
ethyl 1-benzyl-5-(quinoxalin-5-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-3-methyl-1H-pyrazole-4-carboxamide
5-[5-methyl-2-(4H-1,2,4-triazol-4-yl)pyridin-3-yl]-1,2,3,4-tetrahydroisoquinoline
N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-2-methoxyacetamide
{1-[1-(1-benzothiophene-2-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methanol
8-(1H-indol-2-ylmethyl)-1-methyl-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{2-methoxy-4-[3-(1H-pyrazol-3-yl)phenyl]phenyl}acetamide
3-(2-{2-azabicyclo[2.2.1]heptan-2-yl}-2-oxoethyl)-3-phenyl-1-[3-(pyridin-3-yloxy)propyl]pyrrolidine-2,5-dione
(5S)-5-[({[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(pyridin-4-ylmethyl)amino)methyl]pyrrolidin-2-one
1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-4-(1H-imidazol-1-ylmethyl)piperidine
[(3R,4R)-1-(2-methoxy-5-methylbenzoyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
1-(2-methoxyethyl)-N3-methyl-4-oxo-N5-[(1-phenylcyclopentyl)methyl]-N3-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-(2-methoxy-5-phenylphenyl)acetamide
[(3R,4R)-1-(5-chloropyridine-3-carbonyl)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}pyrrolidin-3-yl]methanol
1-[2-(dimethylamino)ethyl]-5-oxo-N-[(3-phenylphenyl)methyl]pyrrolidine-3-carboxamide
5-ethyl-2-(4-{imidazo[1,2-b]pyridazin-6-yl}piperazin-1-yl)pyrimidine
2-{4-[(3,5-dimethoxyphenyl)methyl]-1-(1-methylpiperidin-4-yl)piperazin-2-yl}ethan-1-ol
[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl](propyl)(pyridin-3-ylmethyl)amine
[(3R,5R)-5-[(dimethylamino)methyl]-1-(3-phenoxybenzoyl)piperidin-3-yl]methanol
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(quinolin-8-ylmethyl)piperidin-3-yl]propanamide
2-methoxy-1-{4-[(1-methyl-1H-imidazol-5-yl)methyl]-1,4-diazepan-1-yl}ethan-1-one
N-[(2R,3R)-2-(2-methoxyethoxy)-1'-[2-(thiophen-3-yl)acetyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
N,3-diethyl-5-hydroxy-N-(pyridin-4-ylmethyl)adamantane-1-carboxamide
1-[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
N-[(3S,7S,8aS)-3-[(4-methoxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-methoxybenzamide
diethyl({[5-methyl-4-(3-methyl-1H-1,2,4-triazol-5-yl)furan-2-yl]methyl})amine
ethyl 1-[3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanoyl]-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylate
(1S,5R)-3-benzoyl-6-(2-methoxypyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(propan-2-yl)-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
7-[(2,3-difluorophenyl)methyl]-2-(thiophene-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-(1-ethylpiperidin-4-yl)-4-(naphthalen-2-yloxy)piperidine-4-carboxylic acid
1-(1-benzoxepine-4-carbonyl)-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
4-[(2,6-dimethylhept-5-en-1-yl)amino]adamantan-1-ol
3-({[4-(pyridin-2-yl)pyrimidin-2-yl]amino}methyl)benzoic acid
N-[(3R,4S)-4-cyclopropyl-1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]pyrrolidin-3-yl]-2-hydroxyacetamide
1-[2-(4-methoxyphenoxy)ethyl]-2-(1,3-thiazol-2-yl)piperidine
2-{[6-(methoxymethyl)pyrimidin-4-yl]amino}-1-[3-(trifluoromethyl)phenyl]ethan-1-ol