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N-(2H-1,3-benzodioxol-5-ylmethyl)-1-(6-ethoxy-4-methylquinazolin-2-yl)pyrrolidine-2-carboxamide
N-[2-(dimethylamino)ethyl]-1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-N-methylpiperidin-3-amine
4-(4-methoxybenzoyl)-9-[(1-methylpiperidin-3-yl)methoxy]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-{cyclopropyl[(trimethyl-1H-pyrazol-4-yl)methyl]amino}-1-(3-methylbutyl)azepan-2-one
5-(methoxymethyl)-N-methyl-N-{[2-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazole-2-carboxamide
N-[(4-fluorophenyl)methyl]-N-(3-hydroxypropyl)-4-(1H-pyrazol-3-yl)benzamide
1-(5-amino-4-chloro-1H-pyrazole-3-carbonyl)-N,N-dimethylazepan-4-amine
2-{3-[2-(furan-2-yl)azepan-1-yl]-3-oxopropyl}-2,3-dihydro-1H-isoindol-1-one
5-(cyclohexylamino)-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(3-{4-[(cyclopentylamino)methyl]-2-methoxyphenoxy}-2-hydroxypropyl)piperidin-4-ol
6-[1-(2-chloro-6-methylbenzenesulfonyl)piperidin-4-yl]-2-methyl-3,4-dihydropyrimidin-4-one
7-cyclopentyl-2-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
9-[2-(dimethylamino)-6-methylpyrimidin-4-yl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
5,6-dimethyl-N-[1-(1,3-thiazol-2-yl)propyl]pyrimidin-4-amine
N-butyl-N-methyl-2-[3-(2-methylphenyl)-2,5-dioxo-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]acetamide
4-(1H-1,3-benzodiazol-1-yl)-1-(ethanesulfonyl)piperidine-4-carboxylic acid
1-({2-[3-(1H-pyrazol-1-yl)phenyl]phenyl}methyl)piperazine
(2R,3R)-3-[4-(4-methoxyphenyl)-1H-1,2,3-triazol-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-5-methyl-N-(oxolan-2-ylmethyl)-1,3-oxazole-4-carboxamide
4-[1-(propan-2-yl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]pyridine
7-(1,5-dimethyl-1H-indazole-3-carbonyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
2-[(1,1-dioxo-1λ6-thiolan-3-yl)(methyl)amino]-N-methyl-N-{[2-(2-methylpropoxy)phenyl]methyl}acetamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
1-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]-N-[3-(3-methylphenyl)phenyl]piperidine-3-carboxamide
3-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)propanamide
2-(4,6-dimethylpyrimidin-2-yl)-7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-4-methylpentanamide
3-chloro-N-[2-(dimethylamino)ethyl]-4-{[1-(thiolan-3-yl)piperidin-4-yl]oxy}benzamide
(2S)-2-[4-(2-cyclohexylpyrimidin-5-yl)-1H-1,2,3-triazol-1-yl]-3-hydroxypropanoic acid
{4-[(1-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)methyl]phenyl}methanol
N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-2-oxo-2H-pyran-5-carboxamide
N-(oxan-4-ylmethyl)-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carboxamide
4-{1-[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-1H-1,2,3-triazol-4-yl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
2-[(1S,5R)-3-(5-chloro-3-fluoropyridin-2-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
N-[1-(4-chlorophenyl)cyclobutyl]-1-(2-methoxyethyl)-5-oxopyrrolidine-3-carboxamide
1-(2-{1-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]piperidin-2-yl}ethyl)pyrrolidin-2-one
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-3-methoxy-N-methylpropanamide
5-phenyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
3-(2-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
1-cyclopentanecarbonyl-N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]piperidine-4-carboxamide
N-[(3S,4R)-1-{2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetyl}-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
(3R,4R)-1-{2-[cyclohexyl(methyl)amino]pyridine-3-carbonyl}-4-(hydroxymethyl)piperidin-3-ol
N-[(3S,4R)-1-[1-(2-phenylethyl)piperidin-4-yl]-4-propylpyrrolidin-3-yl]acetamide
ethyl 4-{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}piperazine-1-carboxylate
9-methyl-3-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}-3,9-diazaspiro[5.6]dodecan-10-one
1-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(methylsulfanyl)ethan-1-one
3-[(2R,3R,6R)-5-(2-methoxypyridine-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
4-{3-[2-(hydroxymethyl)piperidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
3-ethyl-8-[4-(4-hydroxyphenyl)benzoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one