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9-[(2-chloro-6-fluorophenyl)methyl]-3,9-diazaspiro[5.6]dodecane
7-[(2S)-2-phenylbutanoyl]-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-(3-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}phenyl)imidazolidin-2-one
(1R,5S,8R)-8-(dimethylamino)-N-[2-methyl-3-(3-methylbutanamido)phenyl]-3-azabicyclo[3.2.1]octane-3-carboxamide
N-({1-[(4-tert-butylphenyl)methyl]piperidin-3-yl}methyl)methanesulfonamide
(4aR,6R,8aS)-8a-(methoxymethyl)-2-[(4-methyl-1,3-thiazol-5-yl)methyl]-6-(morpholin-4-yl)-decahydroisoquinoline
1-methyl-1'-(5-propyl-1,2-oxazole-4-carbonyl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
2-amino-1-[2-(furan-2-yl)-4-(1,2,3,6-tetrahydropyridin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]ethan-1-one
2-[2-oxo-4-(3-phenylbenzoyl)piperazin-1-yl]benzonitrile
4-(pyridin-2-yl)-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}pyrimidin-2-amine
1-(2-methoxyphenyl)-4-pentanoylpiperazin-2-one
6-[(2-propyl-1,3-thiazol-4-yl)methyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
methyl (1S,3S,3aR,6aS)-5-methyl-3-(4-methylphenyl)-4,6-dioxo-1-phenyl-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-(2H-1,3-benzodioxol-5-yl)-4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)piperidine-1-carboxamide
N-(2-ethoxyethyl)-3-({[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}sulfamoyl)benzamide
4-[4-({[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}amino)piperidin-1-yl]-N-cyclopentylbenzamide
N-({1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}methyl)-2,3-dimethoxybenzamide
N,1-dimethyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(benzylsulfamoyl)(furan-2-ylmethyl)(pyridin-2-ylmethyl)amine
4-[4-ethyl-6-(oxan-2-ylmethyl)pyrimidin-2-yl]morpholine
6-oxo-1-(3-phenylpropyl)-N-{[2-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-8-(thian-4-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-3-(thiophen-3-yl)propanamide
N-ethyl-5-[2-(morpholin-4-ylmethyl)phenyl]thiophene-2-carboxamide
3-[2-(dimethylamino)ethyl]-1-(3-methylbutyl)-8-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(4-tert-butyl-1,3-thiazol-2-yl)methyl]-4-(cyclohex-3-en-1-yl)-1H-1,2,3-triazole
(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-7-{[(2-methylphenyl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
[(3S,4S)-1-(6-amino-2-{[(4-methylphenyl)methyl]sulfanyl}pyrimidin-4-yl)-4-(hydroxymethyl)pyrrolidin-3-yl]methanol
(3aR,6aR)-2-benzyl-N-(2-methanesulfonylethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
4-[4-(3-methoxyphenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]-1-[(3-methylphenyl)methyl]piperidine
1-[4-(cyclopentylamino)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
5-ethyl-N-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]-1,3,4-oxadiazol-2-amine
7-[2-methyl-3-(1H-pyrazol-1-yl)propanoyl]-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-(4-methoxy-3,5-dimethylphenyl)-2-({[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}(methyl)amino)acetic acid
1-{4-[3-({[(2-phenyl-1,3-thiazol-5-yl)methyl]amino}methyl)pyridin-2-yl]piperazin-1-yl}ethan-1-one
1-{3-[(3-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}-1H-pyrazol-5-yl)methoxy]phenyl}ethan-1-one
7-[(2-fluorophenyl)methyl]-2-(isoquinolin-5-ylmethyl)-2,7-diazaspiro[4.5]decane
N-[2-(2-ethyl-1,3-thiazol-4-yl)ethyl]-7-fluoro-2-methylquinoline-4-carboxamide
1-{9-methoxy-7-[4-(methylsulfanyl)phenyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-(3,4,5-trimethoxyphenyl)ethan-1-one
7-(3,6-dimethylpyrazin-2-yl)-4-(oxan-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-(2,3-dihydro-1H-indene-1-carbonyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
3-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-6-phenylpyridazine
{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}({[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl})amine
2-[2-(benzyloxy)ethyl]-N-cyclopropylbenzamide
N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-4H-thieno[3,2-b]pyrrole-5-carboxamide
1-(furan-2-ylmethyl)-N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]piperidine-4-carboxamide
methyl({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl){[2-(3-methylphenyl)pyrimidin-5-yl]methyl}amine
3-(3-{[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl}-2,5-dimethyl-1H-pyrrol-1-yl)-4-methylbenzoic acid
N-{3-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-5-({[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]amino}methyl)phenyl}acetamide
5-methyl-3-{[5-(2-methylprop-1-en-1-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-1,2-oxazole