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(1R,5R)-6-[(1-ethyl-1H-indol-4-yl)methyl]-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
{7-methyl-2-[3-(pyridin-4-yl)azetidin-1-yl]quinolin-3-yl}methanol
3-(4-methoxy-2-methylbenzoyl)-1-(oxane-4-carbonyl)piperidine
6-(3-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-3-oxopropyl)-2,3,4,5-tetrahydropyridazin-3-one
4-({2-[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}methyl)pyridine
(4aR,8aS)-1-(2-cyclohexylethyl)-6-[4-(piperidin-1-yl)benzoyl]-decahydro-1,6-naphthyridin-2-one
(1R,5R)-3-(1-ethyl-1H-pyrazole-5-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane
3-{2-[4-(6-aminopyrimidin-4-yl)-6-hydroxy-1,4-diazepan-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
2-acetamido-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}acetamide
1-[2-(4-chlorophenyl)ethyl]-6-oxo-N-(3-phenylpropyl)piperidine-3-carboxamide
(4aR,7aS)-1-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]pyrimidin-4-yl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(diethylamino)-3-(2-methoxy-4-{[methyl(pyrimidin-4-ylmethyl)amino]methyl}phenoxy)propan-2-ol
N,4-dimethyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
methyl (2S,4S)-1-methyl-4-(1-methyl-3-phenyl-1H-pyrazole-5-amido)pyrrolidine-2-carboxylate
3-(diethylamino)-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)propanamide
2,6-dimethoxy-3-[3-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyridine
3-(pyrimidin-4-yl)-N-(1,3,6-trimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)piperidine-1-carboxamide
(1S,5R)-6-(dimethyl-1,2-oxazole-4-carbonyl)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}pyrrolidin-3-yl]acetamide
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-{1-[1-(2-aminoacetyl)piperidin-4-yl]-1H-pyrazol-5-yl}pyridine-3-carboxamide
1-(2-methoxyethyl)-6-oxo-N-(1-phenylcyclopropyl)piperidine-3-carboxamide
5-fluoro-N4-methyl-N2-[1-(2-phenylethyl)piperidin-3-yl]pyrimidine-2,4-diamine
2-(3,4-difluorophenyl)-1-(7-{[ethyl(pyridin-4-ylmethyl)amino]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
4-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
1-(oxan-4-ylmethyl)-4-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
N-cyclopropyl-5-(2-fluorophenoxymethyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-3-carboxamide
7-fluoro-4-{2-[2-(pyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}-1,2-dihydroquinolin-2-one
4-({5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-yl}amino)butan-1-ol
1-(3-chlorophenyl)-5-methyl-4-(naphthalene-1-carbonyl)piperazin-2-one
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-2-(pyridin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[(3R,4S)-1-cyclopentyl-4-propylpyrrolidin-3-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propanamide
1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine
1-methyl-3-(propan-2-yl)-N-{[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H-pyrazole-5-carboxamide
methyl (2S)-1-{[4-(1-methyl-1H-indole-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}pyrrolidine-2-carboxylate
N-benzyl-3-[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]-N-methylpropanamide
1-{2-[7-(2,6-dimethoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}-4-phenylpyrrolidin-2-one
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-{2-[4-(hydroxymethyl)piperidin-1-yl]ethyl}-5-methylpiperidin-2-one
1-[5-methyl-6-(pyrrolidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-yl]piperidine
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-(thiophen-3-ylmethyl)-1H-pyrazole-4-carboxamide
1-(1,3-thiazol-2-ylmethyl)-4-(4H-1,2,4-triazol-3-yl)piperidine
4-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}morpholine
1-(3-{4-[2-(methoxymethyl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidine-1-carbonyl}phenyl)imidazolidin-2-one
2-({[(3R,4R)-1-(2,6-difluoro-3-methoxybenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
(2,1,3-benzoxadiazol-4-ylmethyl)(methyl)[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]amine
(benzylsulfamoyl)[(5-methylpyrazin-2-yl)methyl]amine
1-(2-{4-[3-(4-fluorophenoxy)propyl]piperazin-1-yl}-2-oxoethyl)-1,2-dihydropyrimidin-2-one
1-{2-[({2-methylthieno[2,3-d]pyrimidin-4-yl}amino)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}ethan-1-one
N-cyclopropyl-3-[5-(9H-purin-6-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanamide
1-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-methyl-1,4-dihydroquinolin-4-one