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1-(azocan-1-yl)-3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]propan-1-one
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(morpholin-2-yl)acetamide
N-(3-chloro-4-methoxyphenyl)-3-{1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-3-yl}propanamide
3-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}pyridin-2-amine
methyl 1-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-2-oxo-3-(pentan-3-yl)-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylate
(1S,5R)-6-benzyl-3-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[3-({methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
1-{5-[({imidazo[1,2-a]pyridin-3-ylmethyl}(methyl)amino)methyl]-2-methoxyphenoxy}-3-[methyl(propan-2-yl)amino]propan-2-ol
N-[cyclopropyl(3-methylpyridin-2-yl)methyl]-4-(3-hydroxy-3-methylbutyl)benzamide
3-[4-(1H-pyrazol-1-yl)phenyl]-5-(thiomorpholine-4-sulfonyl)benzoic acid
(1R,9S)-5-amino-3-(2-chloro-3,6-difluorophenyl)-6,12-diazatricyclo[7.2.1.02,7]dodeca-2(7),3,5-triene-4-carbonitrile
N-butyl-4-ethyl-N-(furan-2-ylmethyl)-2-methyl-1,3-thiazole-5-carboxamide
2,5-dimethyl-N-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
3,3-dimethyl-1-[(5-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]urea
5-{1-[1-(4-methoxyphenyl)cyclopentanecarbonyl]pyrrolidin-2-yl}-3-methyl-1H-1,2,4-triazole
N-(1-hydroxybutan-2-yl)-N-(thiophen-2-ylmethyl)furan-3-carboxamide
4-[1-(propan-2-yl)-1H-imidazol-2-yl]-1-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]piperidine
4-methyl-3-{[5-(4-phenyl-1H-imidazol-5-yl)furan-2-yl]sulfanyl}-4H-1,2,4-triazole
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-{[2-(difluoromethoxy)phenyl]methyl}piperidine
1-benzyl-N3-[3-(dimethylamino)-2,2-dimethylpropyl]-4-oxo-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
(1R,5R)-6-[(4-fluoro-3-methoxyphenyl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-{[3-(morpholin-4-yl)piperidin-1-yl]methyl}naphthalen-2-ol
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}pyrrolidine-1-sulfonamide
4-{5-[4-(oxolane-2-carbonyl)piperazine-1-carbonyl]-1H-pyrazol-3-yl}phenol
(2S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-4-{[(4-methoxynaphthalen-1-yl)methyl]amino}-N-methylpyrrolidine-2-carboxamide
{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
1-(3-methyl-1,2-oxazole-5-carbonyl)-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-ol
3-(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-4-yl)-1-(4-phenylpiperazin-1-yl)propan-1-one
6-[1-(propan-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-phenyl-3-(piperidin-4-yl)-1-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
4-{1-[(2,4-dimethoxyphenyl)methyl]piperidin-3-yl}-5-(2-methylphenyl)-2-(pyridin-4-yl)pyrimidine
8-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-[(3R,4S)-3-amino-4-phenylpyrrolidin-1-yl]ethan-1-one
1-[7-(1-benzothiophen-3-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
2-(dimethylamino)-N-methyl-N-(1-{1-[(2E)-2-methylbut-2-enoyl]piperidin-4-yl}-2-phenylethyl)acetamide
5-{1-[(1-benzyl-1H-pyrazol-4-yl)methyl]-1H-imidazol-2-yl}-2-ethylpyrimidine
N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-2-oxo-2H-chromene-3-carboxamide
2-[4-(adamantan-2-yl)-1-[(4-ethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
methyl 2-chloro-4-{[2-(2-methoxyethyl)piperidine-1-carbonyl]amino}benzoate
N-{2-[4-(4-fluorophenyl)-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl]ethyl}cyclobutanecarboxamide
2-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridin-3-ol
1,3,6-trimethyl-N-[1-(pyridin-3-yl)pentyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-{4-[4-(2-methoxyphenyl)piperazine-1-carbonyl]-5-methyl-1H-pyrazol-1-yl}-4-(thiophen-2-yl)pyrimidine
methyl 1-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxylate
7-[2-(ethylamino)pyrimidine-5-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
methyl[(3-methyl-1,2-oxazol-5-yl)methyl][3-(1-methyl-1H-imidazol-2-yl)propyl]amine
1-{2-[5-(thiophen-3-ylmethyl)-1,2,4-oxadiazol-3-yl]ethyl}pyrrolidin-2-one
1-{6-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridin-3-yl}ethan-1-one
4-amino-2-(2-chloro-4-fluorophenyl)pyrimidine-5-carbonitrile
N,N-dimethyl-4-({3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}methyl)benzene-1-sulfonamide