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N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
[1-({1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidin-3-yl}methyl)-1H-1,2,3-triazol-4-yl]methanol
1-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pentan-1-one
methyl 4-(5-{[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
3-(2-oxooxolan-3-yl)-N-[(2E)-3-phenylprop-2-en-1-yl]-N-propylpropanamide
1-acetyl-N-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-3-carboxamide
N-[2-(1H-imidazol-4-yl)ethyl]pyrazolo[1,5-a]pyridine-7-carboxamide
1-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-3-(cyclopropylmethyl)piperidine-3-carboxylic acid
2-[(4-methoxyphenyl)methyl]-4-(4,4,4-trifluorobutyl)morpholine
4-(4,6-dimethylpyrimidin-2-yl)-N-[3-(1H-imidazol-5-yl)phenyl]piperazine-1-carboxamide
{[(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-3-yl)methyl]sulfamoyl}dimethylamine
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-({1-[2-methyl-3-(1H-1,2,4-triazol-1-yl)propanoyl]piperidin-4-yl}methyl)benzoic acid
N,N-dimethyl-2-[(1S,5R)-6-{2-[4-(methylsulfanyl)phenyl]acetyl}-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
ethyl 4-[(3-methoxyphenyl)methyl]-1-[(3-methylquinoxalin-2-yl)methyl]piperidine-4-carboxylate
6-(benzyloxy)-4-[(2E)-3-(4-hydroxy-3-methoxyphenyl)prop-2-en-1-yl]-1-(oxan-4-ylmethyl)-1,4-diazepan-2-one
6-(2-fluoro-4-methoxyphenyl)-N-(2-hydroxyethyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
5-(2-chloro-4-methoxyphenoxymethyl)-N-methyl-N-(pyrazin-2-ylmethyl)-1,2-oxazole-3-carboxamide
5-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]-4-methyl-2-(4-methylpiperazin-1-yl)pyrimidine
N-tert-butyl-4-[(3-methoxypropyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
(3R,4R)-3,4-dimethyl-1-(2-phenylmethanesulfonylbenzoyl)pyrrolidin-3-ol
7-methyl-3-({4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}methyl)quinolin-2-ol
2-(2,5-dimethoxyphenyl)-2-(4-hydroxy-4-phenylpiperidin-1-yl)acetic acid
N-(4-{5-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}phenyl)acetamide
{[6-chloro-2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}bis(prop-2-en-1-yl)amine
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-(oxan-4-yl)piperazin-2-yl}ethan-1-ol
{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[3-(1H-pyrazol-1-yl)propyl]amine
N-[2-(dimethylamino)ethyl]-1,3-dimethyl-2,6-dioxo-N-(oxolan-2-ylmethyl)-1,2,3,6-tetrahydropyrimidine-4-carboxamide
(3S,5R)-1-cyclohexyl-5-[(6-methylpyridin-3-yl)carbamoyl]piperidine-3-carboxylic acid
N-{[3-(difluoromethoxy)phenyl]methyl}-2-(dimethylamino)-2-(3-methylphenyl)acetamide
4-[1-(2,3-dihydro-1-benzofuran-2-carbonyl)piperidin-4-yl]-5-(3-methylphenyl)-2-(pyridin-4-yl)pyrimidine
N5,N5,N6-trimethyl-N6-[(1-methyl-1H-pyrazol-4-yl)methyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
2-(4-{6-amino-5-cyano-4-[5-(hydroxymethyl)furan-2-yl]-3-methylpyridin-2-yl}phenoxy)acetic acid
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[(3,4-dimethoxyphenyl)methyl]-1-[(4-hydroxyphenyl)methyl]piperidine-3,5-dicarboxamide
2-[2-(pyridin-3-ylmethyl)pyrrolidin-1-yl]-4-(trimethyl-1H-pyrazol-4-yl)pyrimidine
(3S,4R)-4-(4-methoxyphenyl)-N,N-dimethyl-1-(2-methylquinolin-4-yl)pyrrolidin-3-amine
3-(2-chlorophenoxy)-1-{[5-(oxan-2-yl)furan-2-yl]methyl}azetidine
2-[5-(5-methoxy-3-methyl-1H-indol-2-yl)-3-methyl-1H-1,2,4-triazol-1-yl]acetic acid
2-amino-4-(2,2-dimethyloxan-4-yl)-6-(3-hydroxyphenyl)pyridine-3-carbonitrile
4-methyl-7-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)-3,4-dihydro-2H-1,4-benzoxazin-3-one
N-[(3S,4R)-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-4-propylpyrrolidin-3-yl]acetamide
1-methyl-4-{[4-phenyl-5-(2,4,6-trimethylphenyl)-1H-imidazol-1-yl]methyl}piperidin-4-ol
3-(2,5-dimethoxyphenyl)-5-[(2-methoxyethyl)sulfamoyl]benzoic acid
8-{[6-(trifluoromethyl)pyridin-3-yl]methyl}-2,8-diazaspiro[4.5]decan-3-one
3-chloro-5-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
3-[2-(4-acetyl-1,4-diazepan-1-yl)-2-oxoethyl]-4-[(3,5-dimethoxyphenyl)methyl]piperazin-2-one
2-{5-[5-(methoxymethyl)furan-2-yl]-1-(2-methoxyphenyl)-1H-1,2,4-triazol-3-yl}acetamide
5-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-5-oxopentanamide
N'-(2,3-dimethylphenyl)-N-methyl-N-(1H-pyrazol-5-ylmethyl)propanediamide
5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]pyridin-2-amine