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2-[3-(1H-pyrazol-5-yl)piperidine-1-carbonyl]-6-(4H-1,2,4-triazol-4-yl)pyridine
3-(1H-indol-3-yl)-1-[4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]propan-1-one
1-{[3-(cyclopentyloxy)phenyl]methyl}-3-(4H-1,2,4-triazol-3-yl)piperidine
1-{[3-methoxy-4-(3-methoxyphenoxy)phenyl]methyl}pyrrolidine
2-(4-methoxy-3-methylphenyl)-2-[4-(5-oxo-1,4-diazepan-1-yl)piperidin-1-yl]acetic acid
1-[(4S)-4-hydroxy-3,3,4-trimethylpiperidin-1-yl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
8-(6-methyl-4-oxo-1,4-dihydropyridine-3-carbonyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
3-{2-[(4-ethoxypyrimidin-2-yl)amino]ethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[benzyl(methyl)amino]-3-{4-[(4-ethylpiperazin-1-yl)methyl]phenoxy}propan-2-ol
N-{[5-(2,6-difluorophenyl)-1,2,4-oxadiazol-3-yl]methyl}-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
3-ethyl-8-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-{3-[(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]phenoxy}ethan-1-ol
3-(2-methoxyphenyl)-N-(2-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)propanamide
(2S,4S)-4-[2-(carbamoylamino)acetamido]-N-ethyl-1-(3-methylbenzoyl)pyrrolidine-2-carboxamide
N-({1-[(5-chlorofuran-2-yl)methyl]piperidin-3-yl}methyl)-1-phenylmethanesulfonamide
N-methyl-3-{methyl[(4-methyl-2-oxo-2H-chromen-7-yl)methyl]amino}butanamide
2-(1H-pyrazol-1-yl)-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]butanamide
1-(cyclopent-1-ene-1-carbonyl)-3-[4-(trifluoromethyl)benzoyl]piperidine
1-(2-methyl-1-benzofuran-5-carbonyl)-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
(2S)-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)-2-(1H-1,2,3,4-tetrazol-1-yl)propanamide
(1S,4S)-2-[2-(methylsulfanyl)phenyl]-5-(quinolin-6-ylmethyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
N-{3-[3-(hydroxymethyl)-3-propylpiperidin-1-yl]-3-oxopropyl}acetamide
2,3,5,6-tetramethyl-N-[2-(morpholin-4-yl)ethyl]benzamide
4-[3-(2-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]quinoline
4-[2-(2-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-1λ6-thiomorpholine-1,1-dione
N-butyl-N-methyl-3-({methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
6-(4-fluorophenyl)-N-methyl-N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
{2-[(2R,3S,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-1,3-thiazol-4-yl}methanol
(2S,4S)-N-ethyl-1-methyl-4-{2-[(4-methylphenyl)methyl]benzamido}pyrrolidine-2-carboxamide
3-{2-oxo-2-[4-(thiomorpholin-4-yl)piperidin-1-yl]ethyl}-3-phenyl-1-(pyridin-4-ylmethyl)pyrrolidine-2,5-dione
1-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]-2-(2-ethoxyphenyl)ethan-1-one
5-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-(oxan-4-yl)pyridin-2-amine
(1S,4S)-5-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-2-(4-chloro-2-methoxy-5-methylphenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
1-(oxolan-3-ylmethyl)-4-{[1,2,4]triazolo[4,3-a]pyrimidin-5-yl}piperazine
2-{1-[(1-{5-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}propan-2-ol
4-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-sulfonyl]-5-methyl-2,1,3-benzothiadiazole
1-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]-2-(1H-imidazol-1-yl)ethan-1-one
5-{[4-(2,3-dihydro-1H-inden-2-yl)piperazin-1-yl]methyl}-N,N-dimethylpyridin-2-amine
N-methyl-4-oxo-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-4H-chromene-2-carboxamide
N-cyclopropyl-1,1-dioxo-N-(thiophen-3-ylmethyl)-1λ6-thiolane-3-carboxamide
3-(3-fluorophenyl)-5-[(2E)-3-phenylprop-2-en-1-yl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
7-methyl-3-[2-(oxan-2-yl)ethyl]-3,4-dihydroquinazolin-4-one
[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl](methyl)[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]amine
2-(3-phenylpropyl)-N-[2-(pyridin-4-yl)ethyl]-1,3-benzoxazole-5-carboxamide
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(2-oxopiperidin-1-yl)acetamide
4-{[3-oxo-3-(pyrrolidin-1-yl)propyl]amino}-N-(pyridin-2-ylmethyl)pyridine-2-carboxamide
1-[(3-fluorophenyl)methyl]-4-[(trimethyl-1H-pyrazol-4-yl)methyl]piperazine
4-benzyl-3-ethyl-1-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}-1,4-diazepan-5-one
3-(2H-1,3-benzodioxol-5-yl)-N-(2-methylpropyl)-N-(pyridin-2-ylmethyl)propanamide
5-[methyl(2-phenylethyl)amino]-2-[2-(pyrrolidin-1-yl)ethyl]-2,3-dihydropyridazin-3-one