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(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-(9H-purin-6-yl)piperidin-3-ol
N-(6-chloropyridin-3-yl)-8-cyclopropyl-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
1-(2,3-dihydro-1H-indol-1-yl)-2-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
[(2-methoxypyrimidin-5-yl)methyl](methyl)[1-(pyridin-2-yl)ethyl]amine
{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[(3-methoxyphenyl)methyl]methylamine
5-(2,5-dimethylfuran-3-yl)-3-[3-(4-fluorophenyl)pyrrolidin-1-yl]-1,2,4-triazine
5-{[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]methyl}-3-(1-methyl-1H-imidazol-4-yl)-1,2,4-oxadiazole
3-{2-[2-(furan-2-yl)pyrrolidine-1-carbonyl]phenyl}-1H-1,2,4-triazole
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-{[4-(methylsulfanyl)phenyl]methyl}-decahydro-2,7-naphthyridine-2-sulfonamide
1-(4-{1-[methyl(pyridin-4-ylmethyl)amino]-2-phenylethyl}piperidin-1-yl)-2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]ethan-1-one
5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-1-[(3-methoxyphenyl)methyl]piperidin-2-one
1-cyclopentanecarbonyl-N-[cyclopropyl(6-methylpyridin-2-yl)methyl]piperidine-4-carboxamide
N-({1-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)acetamide
2-{4-[(benzylsulfamoyl)amino]-3,5-dimethyl-1H-pyrazol-1-yl}acetic acid
1-methyl-2-[3-(thiophen-3-ylmethyl)-1,2,4-oxadiazol-5-yl]piperidine
2-[(3,4-difluorophenyl)methyl]-8-(piperidin-3-yl)-2,8-diazaspiro[4.5]decan-3-one
2-(2,5-dimethylphenoxy)-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}propanamide
5-(3-fluorophenoxymethyl)-N-methyl-N-[(3-methylthiophen-2-yl)methyl]-1H-pyrazole-3-carboxamide
6-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidine-1-carbonyl]-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
(2R,3R,6R)-3-(4-methylphenyl)-5-(pyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-{[2-(furan-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}azepan-2-one
2-({3-[(2S)-2-(methoxymethyl)pyrrolidine-1-carbonyl]phenyl}amino)acetic acid
2-[2-({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)ethyl]-6-phenyl-2,3,4,5-tetrahydropyridazin-3-one
4-{[2-methanesulfonyl-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}thiomorpholine
2-[4-({[(1-cyclopentylpiperidin-3-yl)methyl][2-(piperidin-1-yl)ethyl]amino}methyl)phenoxy]ethan-1-ol
ethyl 2-[4-(2,2,6,6-tetramethylpiperidin-4-yl)piperazin-1-yl]pyridine-3-carboxylate
4-[(4-fluorophenyl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-[2-(3-chlorophenyl)ethyl]-2-(methoxymethyl)-6-methyl-3-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-1,4-dihydropyridin-4-one
3-phenyl-6-{1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-ylmethyl}pyrazolo[1,5-a]pyrimidine
N-cyclohexyl-1-{1,3-dioxo-2-[1-(thiophen-2-yl)ethyl]-2,3-dihydro-1H-isoindol-4-yl}-N-methylpiperidine-4-carboxamide
1-({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)piperidine-4-carboxamide
4-[1-cyclohexyl-5-(pyridin-3-ylmethyl)-1H-1,2,4-triazol-3-yl]pyridine
(4-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}phenyl)methanol
2-[(1-cyclopentylpiperidin-4-yl)methyl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-{[4-(furan-2-carbonyl)piperazin-1-yl]methyl}-8-methoxyquinoline
5-({[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl](methyl)amino}methyl)-N-(propan-2-yl)pyrimidin-2-amine
[(3R,4R)-1-[4-methyl-7-(methylsulfanyl)quinolin-2-yl]-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
1-{1-[2-(2-aminoethyl)quinazolin-4-yl]piperidin-4-yl}-3-methylbutan-1-ol
1-[(2-cyclohexylpyrimidin-5-yl)methyl]-2-methyl-1,4-diazepan-5-one
N-{3-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]-3-oxopropyl}methanesulfonamide
N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-N-methyl-3-{[(4-methylphenyl)methyl]amino}benzamide
1-(3-chlorophenyl)-4-[3-(4-methyl-1H-pyrazol-1-yl)propyl]piperazin-2-one
5-{[2-(5-tert-butyl-1H-pyrazol-3-yl)-1H-imidazol-1-yl]methyl}-3-phenyl-1,2,4-oxadiazole
(3aR,7aS)-2-(5-methoxypyrimidin-2-yl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole
3-{1-[2-(2,5,7-trimethyl-1H-indol-3-yl)acetyl]piperidin-4-yl}-1,3-oxazolidin-2-one
8-(1,3-benzothiazol-2-ylmethyl)-3-[2-(dimethylamino)ethyl]-1-ethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}-3-(trimethyl-1H-pyrazol-1-yl)propanamide
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-5-(phenoxymethyl)-1,2-oxazole-3-carboxamide
methyl 4-(2-{[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]carbamoyl}piperidin-1-yl)-4-oxobutanoate