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2-(ethylamino)-4-methyl-N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-1,3-thiazole-5-carboxamide
(2E)-1-[4-(3-{[4-(furan-2-carbonyl)piperazin-1-yl]methyl}phenoxy)piperidin-1-yl]-3-(4-methoxyphenyl)prop-2-en-1-one
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
3-(2-methylphenyl)-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidine
(3S,4R)-N,N-dimethyl-1-[(3-methyl-1H-indol-2-yl)methyl]-4-propylpyrrolidin-3-amine
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-(oxane-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(1S,2R)-2-{[1-(2-chlorophenyl)piperidin-4-yl]amino}cyclobutyl]-1-methyl-1H-pyrrole-2-carboxamide
N-[1-(1H-indol-1-yl)propan-2-yl]-5-(2-methylphenyl)-1,2,4-triazin-3-amine
4-(3-{[2-(pyridin-3-yl)piperidin-1-yl]methyl}imidazo[1,2-a]pyridine-2-carbonyl)morpholine
(1S,5R)-3-[3-(1H-imidazol-1-yl)propyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{1-[1-(2,6-dimethoxypyridine-3-carbonyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}-N-methylcyclopropanecarboxamide
7-oxo-N,N-bis(prop-2-en-1-yl)-2-propanamido-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
4-({methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}methyl)-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraen-2-one
1-(1-methylpiperidin-4-yl)-N-[2-(1,3-thiazol-4-yl)ethyl]piperidine-3-carboxamide
methyl({2-phenyl-1-[1-(3-phenyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]ethyl})(pyridin-3-ylmethyl)amine
2-ethyl-1-[(1-ethylpyrrolidin-2-yl)methyl]-3-[4-(2-fluorophenyl)piperazine-1-carbonyl]-6-methyl-1,4-dihydropyridin-4-one
4-{1-[5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]piperidin-4-yl}thiomorpholine
2-methoxy-3-{1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-5H,6H,7H-cyclopenta[b]pyridine
(5S,9aS,9bS)-5-(3-methylthiophen-2-yl)-2-(pyridin-3-ylmethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-[(1S,5R)-6-(1H-imidazol-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
(1S,5R)-3-(4-aminopyrimidin-2-yl)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-(3-{[1-(1-methylcyclohexanecarbonyl)piperidin-4-yl]oxy}benzoyl)morpholine
5-phenyl-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]-1,2-oxazole-3-carboxamide
11-(4-hydroxy-3-methylphenyl)-4,6,10,12-tetraazatricyclo[7.3.0.03,7]dodeca-1,3(7),8,10-tetraen-5-one
methyl 3-cyclohexyl-2-oxo-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylate
5-[(2R)-2-amino-4-methylpentanoyl]-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N,N-dimethyl-5-({8-methyl-3-oxo-2,8-diazaspiro[4.5]decan-2-yl}methyl)furan-2-carboxamide
3-{4-[hydroxy(thiophen-2-yl)methyl]piperidine-1-carbonyl}-6-(propan-2-yl)-1,2-dihydropyridin-2-one
{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}[1-(pyrimidin-4-yl)ethyl]amine
2-{[1-(pyridin-4-ylmethyl)piperidin-3-yl]methyl}-1H-1,3-benzodiazole
3-chloro-N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzamide
3-[1-(4-methoxypyrimidin-2-yl)piperidin-3-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-acetyl-8-[3-(1H-imidazol-1-yl)propanoyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-{1-[3-(3-methylphenoxy)azetidine-1-carbonyl]cyclohexyl}morpholine
N-({1-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]piperidin-3-yl}methyl)-1-phenylmethanesulfonamide
2-[1-(2,3-dimethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-5-methylpyrazine
N-[3-(1H-imidazol-1-yl)butyl]-5,6-dimethylthieno[2,3-d]pyrimidin-4-amine
N-[2-(cyclohex-1-en-1-yl)ethyl]-2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-ethyl-2-[2-oxo-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]acetamide
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methyl-4-propylpyrimidine-5-carboxamide
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-2,4-difluorobenzene-1-sulfonamide
3-[4-hydroxy-4-(pyridin-3-yl)piperidine-1-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
N-({3,5-dimethoxy-4-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]pyridine-3-carboxamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carboxamide
N,N-dimethyl-4-[3-methyl-5-(pyrrolidin-1-ylmethyl)phenoxy]benzamide
1-methyl-9-(2-phenylbenzoyl)-1,4,9-triazaspiro[5.5]undecan-5-one
6-{[methyl(2-methylpropyl)amino]methyl}-2-oxo-N-[(4-sulfamoylphenyl)methyl]-1,2-dihydropyridine-3-carboxamide
1-(3-methoxyphenyl)-4-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperazine
2-{1-[(2-chloro-6-fluorophenyl)methyl]-5-(5-ethyl-1,2-oxazol-3-yl)-1H-1,2,4-triazol-3-yl}acetamide
2-(3-chlorobenzoyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one