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4-[4-(2-amino-6-oxo-1,6-dihydropyrimidin-4-yl)piperazine-1-carbonyl]-1,2-dihydroquinolin-2-one
methyl 3-(4-chlorobenzoyl)-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-{2-[3-(3-methoxypropyl)piperidin-1-yl]-2-oxoethyl}-5,6-dimethyl-2,3-dihydropyridazin-3-one
methyl[2-(2-methylphenoxy)ethyl](oxolan-2-ylmethyl)amine
1-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]-2-(2-methyl-1H-imidazol-1-yl)ethan-1-one
8-{6-amino-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-2-benzyl-2,8-diazaspiro[4.5]decan-3-one
[1-({2,4-dimethyl-5-[(4-methylpiperazin-1-yl)methyl]phenyl}methyl)azepan-2-yl]methanol
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]acetamide
1-[4-(2-fluorophenyl)piperazin-1-yl]-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
5-[1-(furan-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-2-(2-methoxyphenyl)-1,3-thiazole
4-(1,3-dimethyl-1H-pyrazol-4-yl)-2-[4-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]pyrimidine
2-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]pyridine
2-methyl-4-{3-[3-(naphthalene-2-carbonyl)piperidine-1-carbonyl]phenyl}but-3-yn-2-ol
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-(oxolan-3-ylmethyl)-1H-pyrazole-3-carboxamide
5-cyclopropanecarbonyl-1'-[(2,4,5-trifluorophenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-methyl-2-(4-methylpiperazin-1-yl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}pyrimidine-5-carboxamide
4,5-dimethyl 1-[(3S,5S)-1-(2-ethylbutyl)-5-{[3-(methylsulfanyl)phenyl]carbamoyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4,5-dicarboxylate
1-[2-(4-chlorophenyl)-2-(pyrrolidin-1-yl)ethyl]-3-(1-ethyl-1H-pyrazol-4-yl)urea
1-phenoxy-2-[4-(quinolin-5-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]propan-2-ol
5-{2-[5-(1-ethyl-1H-1,2,4-triazol-5-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1H-1,2,3,4-tetrazole
1-[4-({[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]amino}methyl)-2-methoxyphenoxy]-3-(4-ethylpiperazin-1-yl)propan-2-ol
2-(2,5-dioxoimidazolidin-1-yl)-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]acetamide
[(3R,4R)-4-[(4-methylpiperazin-1-yl)methyl]-1-(pyrimidin-2-yl)pyrrolidin-3-yl]methanol
1-[(1R)-1-phenylpropyl]-3-(1,3,6-trimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)urea
diethyl[(1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl)methyl]amine
2-hydroxy-N-({1-[(4-methoxy-3-methylphenyl)methyl]piperidin-3-yl}methyl)acetamide
2-{4-[(2-methyl-1,3-oxazol-4-yl)methyl]piperazin-1-yl}-4-(propan-2-yl)-6-(trifluoromethyl)pyrimidine
1-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-5-(4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazole
4-[1-(1,1-dioxo-1λ6-thiolan-3-yl)-3-ethyl-1H-1,2,4-triazol-5-yl]benzene-1-sulfonamide
6-(5-cyclobutyl-1,3,4-oxadiazol-2-yl)-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
3-{3-[(1-methylpiperidin-4-yl)methyl]-5-(pyrazin-2-yl)-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
2-(morpholin-3-yl)-1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]ethan-1-one
2-amino-N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-4-methyl-1,3-thiazole-5-carboxamide
2-methyl-N-(2-phenylethyl)-N-(pyridin-3-ylmethyl)-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
3-({[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl](methyl)amino}methyl)-N-(4-methylpyridin-2-yl)benzamide
1-(3-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}-3-oxopropyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
(4aS,7aR)-1-{imidazo[1,2-a]pyridine-3-carbonyl}-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[2-(3-hydroxypropyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]-N-phenylpropanamide
6-[(diethylamino)methyl]-N-(1,3-thiazol-2-ylmethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
4-(azepan-1-yl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}butanamide
6-ethyl-4-[3-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
N-{1-[4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)phenyl]-1H-pyrazol-4-yl}furan-3-carboxamide
1-[3-(difluoromethoxy)benzoyl]-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-3-(3-hydroxy-3-methylbutyl)benzamide
1-{4-[(4aR,8aR)-octahydro-2H-1,4-benzoxazin-4-ylmethyl]thiophen-2-yl}ethan-1-one
1-(2-{1-[(2-chlorophenyl)methyl]-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-2-methylpropyl)-4-methylpiperazine
1-[4-(furan-2-yl)pyrimidin-2-yl]-5-(methoxymethyl)-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-1H-pyrazole-4-carboxamide
1,3-dimethyl-N-[2-(trimethyl-1H-pyrazol-1-yl)ethyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
(3S,4S)-4-(dimethylamino)-1-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}pyrrolidin-3-ol
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-3-(4-fluorophenyl)-N-methylpropanamide