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4-methyl-2-[4-(pyridin-4-yl)piperidin-1-yl]pyrimidine
4-(2-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-5-fluoropyrimidin-4-yl)morpholine
1,3-dimethyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
1-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(1,3-thiazol-2-yl)piperidine
N-methyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}-2-(oxan-4-yl)acetamide
3-cyclohexyl-1-[2-(diethylamino)ethyl]-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
5-(3,5-dimethyladamantane-1-carbonyl)-4H,5H,6H,7H-thieno[3,2-c]pyridine
1-{4-[6-(benzylamino)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]-1,4-diazepan-1-yl}ethan-1-one
3-({[1-(7-chloro-3,5-dimethyl-1-benzofuran-2-carbonyl)piperidin-3-yl]oxy}methyl)pyridine
N-[(1R,3R)-3-aminocyclopentyl]-2-methyl-5-(2-methyl-1,3-oxazol-5-yl)benzene-1-sulfonamide
(3S,4S)-1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(3-methoxyphenyl)piperidin-3-ol
N-{2-[7-(2-phenylpropyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}pyridine-3-carboxamide
1-(diethylamino)-3-(2-methoxy-5-{[(2-methoxyethyl)(methyl)amino]methyl}phenoxy)propan-2-ol
5-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
6-{[methyl(thian-4-yl)amino]methyl}naphthalen-2-ol
2-[4-({[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl](methyl)amino}methyl)phenyl]-3H,4H,5H,6H,7H-cyclopenta[d]pyrimidin-4-one
4-[4-({3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)phenyl]-2-methylbutan-2-ol
2-{4-[benzyl(methyl)amino]-6-oxo-1,6-dihydropyridazin-1-yl}-N-(thiophen-2-ylmethyl)acetamide
(4-methyl-5-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methanol
1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(4H-1,2,4-triazol-4-yl)ethan-1-one
N-[4-(3-acetamidopropanamido)-2-methoxyphenyl]-3-methylbutanamide
(3aR,6aS)-5-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[(1-methyl-1H-imidazol-5-yl)methyl]-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
1-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
(3S,9aR)-3-[(4-chlorophenyl)methyl]-8-(2,3-difluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(1-ethyl-1H-pyrazol-4-yl)-N,8-dimethyl-N-(propan-2-yl)quinoline-4-carboxamide
N-cyclobutyl-3-{ethyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]sulfamoyl}benzamide
4-(4-aminopyridine-2-carbonyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-({[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)-N-methylacetamide
2-[(3-fluorophenyl)methyl]-6-methyl-1-[3-(morpholin-4-yl)propyl]-3-(thiomorpholine-4-carbonyl)-1,4-dihydropyridin-4-one
methyl(2-phenylethyl)[1-(pyrazin-2-yl)propan-2-yl]amine
1-[(2S)-2-amino-3-cyclohexylpropanoyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}benzamide
3-(5-cyclobutyl-1,3,4-thiadiazol-2-yl)-1-methyl-1-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)urea
3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-[2-(1H-indol-1-yl)ethyl]propanamide
8-(cyclopropylmethyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-[4-(3-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-yl]azocane
1-methyl-N-[(5-methylfuran-2-yl)methyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}-1,3-oxazole-4-carboxamide
3-{3-[3-(6-phenylpyridazin-3-yl)phenyl]-1H-pyrazol-1-yl}propan-1-ol
(1R,3S)-7-(2,2-diphenylethyl)-7-azaspiro[3.5]nonane-1,3-diol
[(3R,4R)-1-(4-methoxy-2-methylbenzoyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
(2R)-2-amino-1-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-phenylethan-1-one
N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-(2-methyl-1,3-thiazol-4-yl)acetamide
N-(3-hydroxypropyl)-N-[(5-methylthiophen-2-yl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-({3-[(1-propylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}methyl)morpholine
2,2-dimethylpropyl 4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxylate
2-[4-(2H-1,3-benzodioxol-5-yl)-2-[(diethylamino)methyl]phenoxy]-N-(3-fluoro-2-methylphenyl)acetamide
N-butyl-4'-ethyl-3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-carboxamide
(3aS,6aS)-2-(ethanesulfonyl)-5-(9H-purin-6-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid