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N-[(3-ethoxyphenyl)methyl]-1-ethyl-N-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-(4-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperazin-1-yl)-N-(pyridin-3-yl)acetamide
2-(1-phenyl-5-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-1,2,4-triazol-3-yl)acetamide
(3aS,6aS)-N-{4-[ethyl(phenyl)carbamoyl]phenyl}-octahydropyrrolo[2,3-c]pyrrole-1-carboxamide
4-[4-({7-[cyclohexyl(hydroxy)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}methyl)phenyl]-2-methylbut-3-yn-2-ol
{[5-(5-fluoropyrimidin-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}(methyl)[2-(pyridin-2-yl)ethyl]amine
[1-(2-methylpyrimidine-5-carbonyl)piperidin-4-yl]diphenylmethanol
(2R)-2-hydroxy-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-phenylacetamide
N,3,6-trimethyl-N-[(2-methylpyridin-4-yl)methyl]-2-(1H-pyrazol-4-yl)quinoline-4-carboxamide
(1R,3s,6r,8S)-4-(2,6-dimethoxypyrimidine-4-carbonyl)-4-azatricyclo[4.3.1.13,8]undecane
3-chloro-4-[(1-cyclohexylpiperidin-4-yl)oxy]-N-[2-(dimethylamino)ethyl]benzamide
2-(2,5-dimethoxyphenyl)-N-[1-(pyrimidin-2-yl)piperidin-3-yl]acetamide
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-3-(3-methoxyphenyl)-N-methyl-1H-pyrazole-5-carboxamide
{5-fluoro-7-[4-(pyrrolidine-1-carbonyl)pyridin-2-yl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
8-(4-cyclobutyl-6-methylpyrimidin-2-yl)-2-methyl-1,3,8-triazaspiro[4.5]dec-1-en-4-one
N-[(3R,4R)-4-hydroxypyrrolidin-3-yl]-2-methyl-3-[(pyridin-3-ylmethyl)amino]benzamide
(2S,4S)-4-amino-N-ethyl-1-{2-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methoxy]acetyl}pyrrolidine-2-carboxamide
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-(1H-pyrazol-3-yl)benzamide
3-(4-hydroxyphenyl)-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-1H-pyrazole-5-carboxamide
2-methyl-N-{[4-(2-methylphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}propanamide
N-methyl-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
3-cyclopropyl-1-[(4-ethylphenyl)methyl]-5-[2-(1H-pyrazol-4-yl)ethyl]-1H-1,2,4-triazole
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(2-methoxypyridine-4-carbonyl)piperidin-3-ol
1-(cyclohexylmethyl)-4-{[(1-ethyl-1H-pyrazol-4-yl)methyl]amino}pyrrolidin-2-one
7-(cyclobutylmethyl)-2-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
2-(2-fluorophenoxymethyl)-N-[(5-methylthiophen-2-yl)methyl]-1,3-oxazole-4-carboxamide
N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1-(propan-2-yl)piperidine-4-carboxamide
2,5-dimethyl-N-[(1-methyl-4-phenylpiperidin-4-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-(dimethyl-1H-1,2,4-triazol-3-yl)-4-(4-fluorophenyl)-1,4-diazepane-1-carboxamide
N-(2,4-dimethylphenyl)-N'-methyl-N'-[1-(pyridin-3-yl)ethyl]ethanediamide
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]propanamide
N-(2,5-difluorophenyl)-3-[(2-hydroxy-3-phenylpropyl)amino]propanamide
N-{2-[3-(4-methoxybenzenesulfonamidomethyl)piperidin-1-yl]-2-oxoethyl}acetamide
N,N-diethyl-9-methyl-10-oxo-3,9-diazaspiro[5.6]dodecane-3-sulfonamide
1-[(2,6-difluorophenyl)methyl]-4-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}-1H-1,2,3-triazole
2-(3-methoxyphenyl)-1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidine
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1H-1,2,3-triazole-5-carboxamide
1-[2-(3,4-dichlorophenyl)morpholin-4-yl]-2-(pyridin-3-yloxy)ethan-1-one
3-(2H-1,3-benzodioxol-5-yl)-N-[(3-methylpyridin-4-yl)methyl]-3-phenylpropanamide
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-2-(dimethylamino)-2-(4-fluorophenyl)acetamide
5-fluoro-2-{[3-(methanesulfonylmethyl)piperidin-1-yl]methyl}-3-methyl-1H-indole
N-[(3-propyl-1,2-oxazol-5-yl)methyl]-6-[3-(1H-pyrazol-1-yl)azetidin-1-yl]pyridine-3-carboxamide
N-ethyl-2-(4-{1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)acetamide
3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-(prop-2-en-1-yl)propanamide
1-(2-methoxyethyl)-6-oxo-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]piperidine-3-carboxamide
2-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-5-fluoro-4-methoxypyrimidine
N-(furan-2-ylmethyl)-3-{4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazin-1-yl}propanamide
1-phenyl-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1H-1,2,3-triazole-4-carboxamide
5-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[2-(dimethylamino)ethyl]-3-(2-fluorophenyl)-3-{2-[4-(2-fluorophenyl)piperazin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione