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1-{3-[(pyridin-3-yl)amino]propyl}-3-(5,6,7,8-tetrahydronaphthalen-1-yl)urea
3-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-5,6-dimethyl-1,2-dihydropyridin-2-one
6-[4-(thiomorpholin-4-yl)piperidin-1-yl]-N-(thiophen-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
2-(3-fluorophenoxymethyl)-N-[(3S,4S)-4-hydroxy-1-(propan-2-yl)pyrrolidin-3-yl]-1,3-oxazole-4-carboxamide
(2S)-N-(3-chloro-2-ethoxyphenyl)-2-(morpholine-4-carbonyl)pyrrolidine-1-carboxamide
2-(4-methyl-1H-imidazol-5-yl)-1-[2-(thiophen-2-yl)ethyl]-1H-imidazole
1-(4-{[(cyclopropylmethyl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
(3aR,6aS)-2-ethyl-1-oxo-5-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-amino-8-{3-methoxy-4-[(3-methylbut-2-en-1-yl)oxy]phenyl}-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
3-(2-methoxybenzoyl)-N-[4-(trifluoromethyl)phenyl]piperidine-1-carboxamide
ethyl 4-{[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}piperazine-1-carboxylate
2-(cyclopropylmethyl)-8-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
3-[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-3-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-3-[(oxolan-3-yl)sulfamoyl]benzamide
3-methyl-N-{2-[(4-methylpyridin-2-yl)amino]ethyl}-4-oxo-3,4-dihydrophthalazine-1-carboxamide
1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine
methyl 2-(azocane-1-sulfonyl)-6-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-[2-methoxy-4-({methyl[(4-methyl-1,3-thiazol-2-yl)methyl]amino}methyl)phenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
4-({4-[(2-fluoro-4-methoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenol
methyl({[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}){[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}amine
4-ethyl-1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-{5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carbonyl]pyrimidin-2-yl}morpholine
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-5-(pyrrolidine-1-carbonyl)pyridin-2-amine
N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-(2H-1,3-benzodioxol-5-yl)-7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
2-cyclopropyl-8-(4-methylquinolin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
3-phenyl-N-(1-propyl-1H-1,2,3-triazol-4-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carboxamide
3-[methyl({2-methylpyrido[2,3-d]pyrimidin-4-yl})amino]-1-phenylpropan-1-ol
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N,3,6-trimethyl-1-benzofuran-2-carboxamide
4-[3-(2-methoxyethyl)-1-methyl-1H-1,2,4-triazol-5-yl]-N,N-dimethylpiperidine-1-carboxamide
1-[3-(2H-1,3-benzodioxol-5-yl)-2-methylpropyl]-4-[(2-fluorophenyl)methyl]-1,4-diazepan-5-one
3-[1-(4-cyano-1-methyl-1H-pyrrole-2-carbonyl)piperidin-3-yl]-N-[(5-methylfuran-2-yl)methyl]propanamide
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperazine
3-[1-(cyclohex-3-en-1-ylmethyl)-1H-pyrazol-5-yl]-1-(2-hydroxyethyl)-1-[(5-methylthiophen-2-yl)methyl]urea
[(3S,5R)-1-(5-chlorothiophene-2-carbonyl)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]piperidin-3-yl]methanol
1-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-methoxyethan-1-one
(2S,4S)-4-amino-N-ethyl-1-[2-hydroxy-4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]pyrrolidine-2-carboxamide
N-methyl-2-[1-methyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]-N-(1,2-oxazol-3-ylmethyl)acetamide
N-(2,4-difluorophenyl)-3-{[methyl(1,2-oxazol-5-ylmethyl)amino]methyl}benzamide
ethyl 5-{imidazo[1,2-a]pyridine-2-carbonyl}-1-(2-methoxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
4-[(4-butyl-1H-1,2,3-triazol-1-yl)methyl]-1-{imidazo[1,2-a]pyridine-2-carbonyl}piperidine
N-{4-[(3S,4S)-3,4-dihydroxy-4-methylpiperidine-1-carbonyl]phenyl}ethane-1-sulfonamide
methyl({[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl})[2-(piperidin-1-yl)ethyl]amine
N-(6-phenoxypyridin-3-yl)-1-(2-phenylethyl)piperidine-4-carboxamide
4-{[4-(2-methyl-1-benzofuran-5-carbonyl)piperazin-1-yl]sulfonyl}morpholine
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-3-methylbutanamide
2,6-difluoro-N-(2-hydroxyethyl)-3-methoxy-N-[(2E)-3-phenylprop-2-en-1-yl]benzamide
4-ethyl-N-methyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)piperazine-1-sulfonamide
4-{[2-(3-chlorophenyl)-8-methylquinolin-3-yl]methyl}-3-methylpiperazin-2-one
1-{4-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]thiophen-2-yl}ethan-1-one