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2-{[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]methyl}phenol
3-(2-chlorophenyl)-1-methyl-6-(thiophene-3-carbonyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
2-{3-[4-(4-chlorophenoxy)piperidine-1-carbonyl]piperidin-1-yl}acetamide
N-{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N,1-dimethyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
2-(3-{1-ethyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenoxymethyl)pyridine
2-(dimethylamino)-N-(1H-indol-2-ylmethyl)benzamide
3-{5-[1-(5-propyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]-1,2,4-oxadiazol-3-yl}pyridine
5-(1-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1H-1,2,3-triazol-4-yl)-2-methoxypyridine
(1S,6R)-3-methyl-9-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
1-[(4-chlorophenyl)methyl]-6-oxo-N-{[4-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
5-{3-oxo-3-[4-(pyridin-2-ylmethoxy)piperidin-1-yl]propyl}imidazolidine-2,4-dione
2-(2-methoxyethyl)-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]-1,3-benzoxazole-6-carboxamide
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-2-(pyridin-2-ylsulfanyl)acetamide
5-methyl-1-(oxan-4-ylmethyl)-5-phenylpiperidin-2-one
4-(1H-pyrazol-3-yl)-N-[1-(pyrrolidine-1-carbonyl)piperidin-4-yl]benzamide
4-{2-[4-(2,6-dimethylpyridine-4-carbonyl)piperazin-1-yl]ethyl}morpholine
N-(prop-2-en-1-yl)-N-(pyridin-3-ylmethyl)-4-(trifluoromethyl)benzamide
3-[(3R,4S)-1-(1-methyl-1H-pyrazole-4-carbonyl)-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
2-{4-[5-(2-fluorophenyl)-1,2,4-triazin-3-yl]piperazin-1-yl}ethan-1-ol
ethyl 2-{[4-(1,3-thiazol-2-yl)piperazin-1-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxylate
(2S)-2-acetamido-4-methyl-N-({5-[4-(methylsulfanyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)pentanamide
1-(2-methoxyethyl)-4-oxo-N-[(1-phenylcyclopentyl)methyl]-5-(pyrrolidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
1-[1'-(5-fluoro-2-methylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
2-methyl-4-{3-methyl-5-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazol-5-yl]-1H-1,2,4-triazol-1-yl}pyridine
1-[2-(5-methyl-1,2-oxazol-3-yl)pyrrolidin-1-yl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propan-1-one
4-{2-[1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidin-2-yl]ethyl}phenol
(4aS,7aR)-1-(1,5-dimethyl-1H-indole-2-carbonyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(5,6-dimethoxy-1-oxo-1,2-dihydroisoquinolin-2-yl)-N-methyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]acetamide
3-({4-[3-(4-ethylpiperazin-1-yl)-3-oxopropyl]piperidin-1-yl}methyl)-1,2,4-oxadiazole-5-carboxamide
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-3-(3-methoxyphenyl)-N-methyl-1H-pyrazole-4-carboxamide
4-({4-methyl-5-[1-(1H-pyrazole-3-carbonyl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
N-(3-methyl-1-{7-[(2E)-2-methylbut-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)furan-2-carboxamide
1-[(2-methoxyphenyl)methyl]-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
4-(4-chlorophenyl)-N-cyclopropyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]butanamide
(3R,5S)-1-[(3,4-dimethoxyphenyl)methyl]-3-(pyrrolidine-1-carbonyl)-5-[3-(trifluoromethyl)phenoxymethyl]piperidine
3-methyl-N-[(3R,4S)-1-[2-(2-oxopyrrolidin-1-yl)ethyl]-4-(propan-2-yl)pyrrolidin-3-yl]-1,2-oxazole-5-carboxamide
4-(1-butyl-1H-imidazol-2-yl)-1-(3-chloro-5-fluorobenzoyl)piperidine
2-(pyridin-2-ylsulfanyl)-1-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
(2S)-N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}pyrrolidine-2-carboxamide
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-3,5-dimethyl-1-benzofuran-2-carboxamide
3-(2-amino-1,3-thiazol-4-yl)-N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]propanamide
1-(cyclopropylmethyl)-4-(2-methoxy-5-methylbenzoyl)-2-(propan-2-yl)-1,4-diazepane
6-fluoro-N,N-dimethyl-2-(1-phenyl-1H-pyrazol-4-yl)quinoline-4-carboxamide
3-(1-{1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(2-methylphenyl)urea
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)propanamide
4-(2-fluorobenzenesulfonyl)-7-(2-methylphenyl)-9-(oxolan-3-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
[4-(3-phenylpropyl)-1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidin-4-yl]methanol
N,6-dimethyl-4-oxo-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1,4-dihydropyridine-3-carboxamide
1-ethyl-N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-[(3S)-1-benzylpyrrolidin-3-yl]-5-phenyl-1,2-oxazole-4-carboxamide