Propranolol

• 产品号: Bio-0732
• CAS号: 525-66-6
• 分子式: C16H21NO2
• 分子量: 259.34344

产品别名

• 标题: Propranolol
• IUPAC标准名: [2-hydroxy-3-(naphthalen-1-yloxy)propyl](propan-2-yl)amine
• IUPAC传统名: [2-hydroxy-3-(naphthalen-1-yloxy)propyl](propan-2-yl)amine
• 别名: 1-[(1-Methylethyl)amino]-3-(1-naphthalenyloxy)-2-propanol; 1-Isopropylamino-3-(1-naphthyloxy)-2-propanol

产品登记号

• CAS号: 525-66-6

产品性质

• 应用领域: Antiarrhythmic agent
• 应用领域: Hypotensives
• 应用领域: Local anesthetic
• 生物活性机理: Beta-Adrenergic blocking agent
• 生物活性机理: It is a non-selective beta blocker, that is, it blocks the action of epinephrine on both beta1- and beta2-adrenergic receptors.
• 生物活性机理: It has little intrinsic sympathomimetic activity (ISA) but has strong membrane stabilizing activity (only at high blood concentrations, eg overdosage).
• 生物活性机理: Only L-propranolol is a powerful adrenoceptor antagonist, whereas D-propranolol is not

参考文献

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