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3-({2-[1-(2,5-dimethylfuran-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
(2S)-2-amino-1-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}-3-(4-methoxyphenyl)propan-1-one
3,3-dimethyl-1-{2-oxo-2-[3-oxo-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-9-yl]ethyl}urea
N,N-diethyl-3-oxo-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-butyl-2-{[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl](methyl)amino}acetamide
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-3,5-dimethyladamantane-1-carboxamide
1-cyclopentanecarbonyl-N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide
3-[(3-methylpiperidin-1-yl)methyl]-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrimidin-3-yl}benzamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(3,4-difluorophenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
2-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-N-(propan-2-yl)acetamide
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
N-[2-(3-ethylphenoxy)ethyl]-N-methyl-2-{3-oxo-2-azaspiro[4.4]nonan-2-yl}acetamide
3-(2-methylpropyl)-5-[3-(1H-pyrazol-4-yl)phenyl]-1H-1,2,4-triazole
N-benzyl-N-butyl-2,8-diazaspiro[4.5]decane-3-carboxamide
N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
1-[(1-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)methyl]pyrrolidin-2-one
(2S)-2-({6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidin-3-yl}formamido)-3-methylbutanamide
3-{[1-(4-carbamoylpyridin-2-yl)piperidin-4-yl]methyl}benzoic acid
1-{4-[5-(3-fluorophenyl)-2-[(2-methoxyethyl)sulfanyl]pyrimidin-4-yl]piperidin-1-yl}-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
(2R)-2-amino-1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-methylbutan-1-one
1-[3-(3-fluorophenyl)propyl]-4-(3-methylpyridin-4-yl)piperazine
2-(5-{[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]methyl}-1,2,4-oxadiazol-3-yl)pyridine
N-[4-(1H-indol-2-yl)phenyl]-1-(oxan-4-yl)pyrrolidine-2-carboxamide
N-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
2-[3-(dimethylamino)propyl]-9-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}-2,9-diazaspiro[5.5]undecan-3-one
1-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-phenyl-1,4-diazepane
1-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
1-[(3aR,6aR)-2-cyclopentyl-octahydropyrrolo[3,4-c]pyrrole-3a-carbonyl]piperidine-4-carboxamide
7-[2-(methylamino)-1,3-thiazole-4-carbonyl]-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-(6,8-difluoroquinolin-4-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}[3-(1H-pyrazol-1-yl)propyl]amine
1-{[2-cyclohexylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-2-methylpiperidine
3-(cyclopropylsulfamoyl)-5-(2,4-dimethoxyphenyl)benzoic acid
2-ethyl-8-[2-(3-methyl-6-oxo-1,6-dihydropyridazin-1-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
[(3R,4R)-4-(piperidin-1-ylmethyl)-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl]methanol
6-[(4aS,8aR)-1-[2-(methylamino)ethyl]-2-oxo-decahydro-1,6-naphthyridin-6-yl]-N-ethylpyridine-3-carboxamide
1-(2-phenylethyl)-N-[4-(pyridin-3-yloxy)phenyl]piperidine-2-carboxamide
1-[(2-chlorophenyl)methyl]-N-[(2-methyl-1H-indol-5-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-cyclohexyl-3-[(6-ethyl-2-methylquinolin-4-yl)formamido]propanamide
N1-{1-[3-(furan-2-yl)phenyl]piperidin-4-yl}propane-1,3-diamine
3-hydroxy-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]pyridine-2-carboxamide
7-fluoro-3-methyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1-benzofuran-2-carboxamide
(5-{1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}furan-2-yl)methanol
N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
2-cyclopentyl-9-({7-oxo-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)-2,9-diazaspiro[5.5]undecan-3-one
2-{[3-(2,3-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1-ethyl-1H-imidazole
[(3R,4R)-1-(6-methyl-2-phenylpyrimidin-4-yl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
2-chloro-4-[({[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]phenol
5-ethyl-1'-[6-(methoxymethyl)pyridine-2-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-(3-hydroxy-3-methylbutyl)-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}benzamide