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1-(2-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-oxoethyl)-1,2-dihydropyridin-2-one
2-amino-6-(4-methyl-1,3-thiazol-5-yl)-4-[1-(pyridin-4-yl)-1H-pyrrol-2-yl]pyridine-3-carbonitrile
N-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-N-methyl-2,3-dihydro-1H-inden-2-amine
3-(3,4-difluorophenyl)-5-(3-methylfuran-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
8-[2-(3-chloro-2,6-difluorophenyl)acetyl]-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
(4aR,7aS)-4-[(4-fluoro-2-methylphenyl)methyl]-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
1'-(1H-pyrrole-2-carbonyl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
methyl[(2-methyl-1H-imidazol-4-yl)methyl][1-(pyridin-2-yl)ethyl]amine
1-(1-ethyl-1H-pyrazole-5-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
2-methyl-3-({4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}methyl)quinoxaline
1,3-dimethyl-N-[1-(pyrazin-2-yl)propan-2-yl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
methyl 3-cyclohexanecarbonyl-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
8-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
(1R,3S,5S)-8-(4-methylquinazolin-2-yl)-8-azabicyclo[3.2.1]octan-3-ol
1-(2-{3-[ethyl(pyridin-4-ylmethyl)amino]piperidin-1-yl}-2-oxoethyl)-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[2-(azepan-1-yl)-2-phenylethyl]-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-[3-(1H-imidazol-1-yl)propyl]-9-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
5-[1-(2H-1,3-benzodioxol-5-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-4-ethyl-1,2,3-thiadiazole
9-(6-aminopyrimidin-4-yl)-2-(cyclopropylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(3S,4S)-4-(morpholin-4-yl)-1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}pyrrolidin-3-ol
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-methyl-3-(pyrrolidin-1-yl)propanamide
(1-benzothiophen-2-ylmethyl)({[4-({1-[(5-chlorothiophen-2-yl)sulfonyl]piperidin-4-yl}oxy)phenyl]methyl})methylamine
N-{[3-methyl-7-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}thiophene-2-sulfonamide
2-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)phenol
1-{[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}-4-(4-methyl-1,2,5-oxadiazol-3-yl)piperazine
N,N-dimethyl-4-(2-phenylmorpholin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
3-(hydroxymethyl)-1-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-3-ol
1-[cyclohexyl(methyl)amino]-3-[2-methoxy-4-({methyl[(4-methyl-1,3-thiazol-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
5-{methyl[(3-methylpyridin-4-yl)methyl]amino}-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
1,3-dimethyl-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
1-methyl-4-({[4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}methyl)pyrrolidin-2-one
2-({[(3R,4R)-1-(4-chloro-2-methylbenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
6-(2-aminoethyl)-N-[furan-2-yl(phenyl)methyl]pyrimidin-4-amine
1-ethyl-N-[4-(furan-2-yl)butan-2-yl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl](methyl){[1-(piperidin-1-yl)cyclohexyl]methyl}amine
N-ethyl-N-{[6-(4-methyl-1,4-diazepane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}cyclopropanamine
N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)-2,1,3-benzothiadiazole-4-sulfonamide
1-{1-[(3,5-dimethoxyphenyl)methyl]piperidin-3-yl}-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide
3-[(propan-2-yl)sulfamoyl]-5-(pyridin-3-yl)benzoic acid
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperazine
{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
[(2S)-1-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl]methanol
4-{5-[3-(3-methoxyphenyl)-1H-pyrazol-5-yl]-1,2,4-oxadiazol-3-yl}pyridine
7-(2-hydroxyethyl)-2-{[5-(4-methylphenyl)-1,2,4-oxadiazol-3-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
5-(1-cyclopentylpyrrolidin-2-yl)-N-[2-(methylsulfamoyl)ethyl]thiophene-2-carboxamide
2-{2-[2-(2-methoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-2-cyclopropyl-4-methylpyrimidine-5-carboxamide
1-(cyclopropylmethyl)-N-(pyridin-2-ylmethyl)-5-[2-(thiophen-3-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
{3-[(2,4-difluorophenyl)methyl]-1-[(8-methoxyquinolin-2-yl)methyl]piperidin-3-yl}methanol