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3-acetamido-N-[3-(trifluoromethyl)phenyl]pyrrolidine-1-carboxamide
4-{[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]amino}-N-(propan-2-yl)pyridine-2-carboxamide
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]acetamide
methyl 4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
propyl 4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
2,5-dimethoxy-N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)benzene-1-sulfonamide
5-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-4-phenyl-1H-imidazole
3-phenyl-1-[1-(pyrrolidine-1-carbonyl)piperidin-3-yl]propan-1-one
2-{3-[1-(4-fluorophenyl)-1H-pyrazol-4-yl]-1H-pyrazol-1-yl}-N-(1-methyl-1H-pyrazol-5-yl)acetamide
2-[(cyclopentylamino)methyl]-4-(pyrazin-2-yl)phenol
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)pyridin-2-amine
ethyl 4-{[(2-methylpropyl)(pyridin-2-ylmethyl)amino]methyl}-1H-pyrazole-3-carboxylate
1-(4,7-dimethylquinazolin-2-yl)-N-(oxolan-3-yl)piperidine-4-carboxamide
(4aS,8aR)-1-(2-aminoethyl)-6-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}-decahydro-1,6-naphthyridin-2-one
4-[3-(propoxymethyl)pyrrolidin-1-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
1-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(thiophen-2-yl)propan-1-one
5-{[1-(2-methoxyphenyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-1H-1,2,3,4-tetrazole
N-cyclooctyl-1-[(2-fluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
2-[(4aR,8aR)-4a-hydroxy-7-methanesulfonyl-decahydro-2,7-naphthyridin-2-yl]-N-[(2-methylphenyl)methyl]acetamide
N-[4-({[(2,3-dimethylphenyl)methyl]carbamoyl}methoxy)phenyl]propanamide
2-cyclopentyl-9-(2,5-difluorobenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-2-methyl-1H-pyrrole-3-carboxamide
[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-[(3-methoxyphenyl)methyl]piperidin-4-yl]methanol
1-[3-(pyridin-3-yl)azetidin-1-yl]-3-(4H-1,2,4-triazol-4-yl)propan-1-one
[(6-chloropyridin-3-yl)methyl]({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})amine
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]-decahydro-1,6-naphthyridin-2-one
6-{4-[(3-methylphenyl)sulfanyl]piperidin-1-yl}pyridine-2-carboxylic acid
(2S,4S)-4-amino-N,N-diethyl-1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}pyrrolidine-2-carboxamide
7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-9-methoxy-4-[(5-methylfuran-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-4-(piperidin-1-ylmethyl)benzamide
(3S,4R)-3-benzyl-1-(3-cyclopropyl-1,2-oxazole-5-carbonyl)-4-methylpiperidin-4-ol
[(2S,4R,5R)-5-(2-fluorophenyl)-1-methyl-4-[({3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}amino)methyl]pyrrolidin-2-yl]methanol
2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)acetamide
3-({[1-(4-methyl-1,3-thiazol-2-yl)piperidin-3-yl]oxy}methyl)pyridine
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl][(5-methylthiophen-2-yl)methyl](pyridin-4-ylmethyl)amine
4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]benzamide
4-[3-(2-methoxyphenoxy)propyl]-6-methylpyrimidin-2-amine
(2E)-N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(pyridin-2-yl)prop-2-enamide
(3R,5S)-1-benzyl-N-[3-(dimethylamino)propyl]-5-(3-fluorophenoxymethyl)piperidine-3-carboxamide
3-[(dimethylamino)methyl]-1-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}pyrrolidin-3-ol
N-ethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1H-1,2,3-triazole-5-carboxamide
1-{6-[2-(pyridin-3-yl)-1H-imidazol-1-yl]-1,2,3,4-tetrahydroquinolin-1-yl}ethan-1-one
N-ethyl-5-(1-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}pyrrolidin-2-yl)thiophene-2-carboxamide
1-[(5-ethylpyridin-2-yl)methyl]-4-(naphthalen-2-yloxy)piperidine-4-carboxylic acid
{1-[2-(2-methoxy-4-methylphenyl)-1H-imidazol-1-yl]butan-2-yl}dimethylamine
1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-2-methyl-2-(methylamino)propan-1-one
5-(quinolin-8-yl)furan-2-carboxylic acid
(1H-1,3-benzodiazol-2-ylmethyl)(benzyl)(1,3-thiazol-2-ylmethyl)amine
(1R,5R)-6-(cyclopropylmethyl)-3-(5-fluoro-2-methoxybenzoyl)-3,6-diazabicyclo[3.2.2]nonane
3-(2-{1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}-2-oxoethyl)imidazolidine-2,4-dione