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N-[(1-benzylpiperidin-4-yl)methyl]-4,4,4-trifluoro-N-methylbutanamide
N-(cyclohex-1-en-1-ylmethyl)-1-(pyridin-2-yl)piperidine-3-carboxamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-({1-[(4-methylphenyl)amino]cyclohexyl}formamido)acetic acid
N-[(2,5-difluorophenyl)methyl]-1-(6-fluoro-4-methylquinazolin-2-yl)azepan-4-amine
2-ethyl-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methylpyrimidine-5-carboxamide
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-4-methoxypiperidine-1-sulfonamide
(3R,4S)-4-({[6-(dimethylamino)pyridin-3-yl]methyl}(ethyl)amino)oxolan-3-ol
3-[1-(2,1,3-benzoxadiazol-5-ylmethyl)piperidin-3-yl]-N-[(2-chlorophenyl)methyl]propanamide
9-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{3-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-oxopropyl}methanesulfonamide
1-{2-[3-(hydroxymethyl)phenyl]pyrimidin-4-yl}pyrrolidin-3-ol
(3R,5S)-1-benzyl-5-(morpholin-4-ylmethyl)-N-(oxolan-2-ylmethyl)piperidine-3-carboxamide
5-[(4-fluoro-3-methoxyphenyl)methyl]-5-{3-[4-(6-methylpyridin-2-yl)piperazin-1-yl]-3-oxopropyl}pyrrolidin-2-one
2-amino-6-(3,4-dimethoxyphenyl)-4-(4-hydroxy-2-methoxyphenyl)pyridine-3-carbonitrile
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
(1R,5S,6R,7S)-N-{[2-(diethylamino)pyridin-3-yl]methyl}-3-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-butyl-2-(phenylamino)-N-(thiophen-3-ylmethyl)pyrimidine-5-carboxamide
1-{5-acetyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-phenoxypropan-1-one
2-(2-methoxyethyl)-6-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1,3-benzoxazole
2-(4-methoxy-3,5-dimethylphenyl)-5-(pyrrolidin-1-ylmethyl)pyridine
3-({4-[(2-hydroxyethyl)(methyl)amino]piperidin-1-yl}methyl)-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
1-(1,2-oxazolidin-2-yl)-3-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)propan-1-one
(1R,7S)-3-(pentan-3-yl)-6-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
N-(3-aminopropyl)-1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]piperidine-3-carboxamide
(3-{2-[1-(2,3-dihydro-1-benzofuran-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
7-[3-(1,2-oxazinan-2-yl)propanoyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
(1S,5R)-3-[2-(4-fluoro-2-methylphenyl)acetyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
5-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
(1S,5R)-6-(1-phenylcyclopropanecarbonyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-ethyl-5-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyrimidin-2-amine
1-ethyl-2,5-dimethyl-N-[(1S,2R)-2-[(oxan-4-yl)amino]cyclobutyl]-1H-pyrrole-3-carboxamide
N-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-3-cyclohexyl-1H-pyrazole-4-carboxamide
1-(2-aminoethyl)-N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
ethyl 3-benzyl-1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidine-3-carboxylate
3-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-N-methyl-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-1,2-oxazole-5-carboxamide
1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-2,3,4,9-tetrahydro-1H-carbazole
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-(1H-pyrazol-1-yl)benzamide
7-({4-[2-methyl-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}methyl)quinoline
N-[(1-ethyl-1H-imidazol-5-yl)methyl]-5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
2-[2-(4-fluorophenyl)ethyl]-4-{4-[3-(3-methoxyphenyl)propanoyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N-methyl-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1H-indazole-3-carboxamide
3-[5-(5-phenyl-1,2-oxazole-3-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]pyridine
N-methyl-5-[1-(1-methylpiperidin-4-yl)-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]pyrimidin-2-amine
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-4-(1H-imidazol-1-yl)benzamide
3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}-N-(2,3-dimethylphenyl)piperidine-1-carboxamide
2-[2-(3-fluorophenyl)pyrimidin-5-yl]-N,N,8-trimethylquinoline-4-carboxamide
(1S,5R)-6-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
7-fluoro-3-({[2-(2-methoxyphenyl)ethyl]amino}methyl)-N,N-dimethylquinolin-2-amine
4-{[2-(4-methoxyphenyl)ethyl]amino}-N,5-dimethyl-N-[1-(1,2-oxazol-3-yl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide