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(3aS,6aR)-3-[2-(4-methoxyphenyl)ethyl]-5-(pyrazin-2-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-{1-[(3-methylphenyl)methyl]cyclopropyl}-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
2-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-3-carbonitrile
(4aS,7aR)-1-(2-methylpropyl)-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
butyl 2-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxylate
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]piperidin-3-amine
2-[4-(isoquinolin-5-ylmethyl)-1-(3-methylbutyl)piperazin-2-yl]ethan-1-ol
1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-methyl-1,4-diazepan-5-one
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-3-(2-oxopyrrolidin-1-yl)propanamide
2-hydroxy-1-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}propan-1-one
3-ethyl-1-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]-1H-pyrazole-5-carboxamide
8-[2-(1H-imidazol-1-yl)acetyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
1-[4-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
(3S,9aR)-8-(naphthalene-2-sulfonyl)-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-(4-methylphenyl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}propanamide
N1-(2-methoxy-5-phenylphenyl)piperidine-1,3-dicarboxamide
(4aS,7aR)-1-(4-methyl-2-oxopentanoyl)-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-2,4-dimethylpyrimidine-5-carboxamide
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-4-(pyridin-2-yl)pyrimidin-2-amine
N-[(5-chloro-1H-indol-2-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
1-(cyclopropylmethyl)-5-(2-methyl-1H-1,3-benzodiazole-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
4-({4-[3-(azocan-1-yl)-2-hydroxypropoxy]-3-methoxyphenyl}methyl)piperazin-2-one
[(2S,4R,5R)-5-(4-chlorophenyl)-4-({[(3,5-dimethoxyphenyl)methyl]amino}methyl)-1-ethyl-2-methylpyrrolidin-2-yl]methanol
N-(2-{7-[(2-fluoro-5-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-3-carboxamide
3-cyclohexyl-2-oxo-1-{[(oxolan-2-ylmethyl)carbamoyl]methyl}-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
5-{[(4-methoxynaphthalen-1-yl)oxy]methyl}-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1,2-oxazole-3-carboxamide
2-[3-(2-hydroxyethyl)-4-(2-phenylethyl)piperazine-1-carbonyl]-4-methylphenol
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylcyclobutanamine
N-{[7-fluoro-5-(3-fluoro-4-methylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}oxolane-2-carboxamide
2-methoxy-3-{thieno[3,2-d]pyrimidin-4-yl}pyridine
2-ethoxy-5-{2-[4-hydroxy-4-(hydroxymethyl)piperidin-1-yl]pyrimidin-4-yl}benzoic acid
6-methyl-2-(morpholin-4-yl)-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}pyrimidin-4-amine
6-(2-chlorophenyl)-2-{4-[(diethylamino)methyl]phenyl}-3,4-dihydropyrimidin-4-one
{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)[(5-phenyl-1,2-oxazol-3-yl)methyl]amine
3-[2-(propylsulfanyl)phenyl]-1-[1-(pyrazin-2-yl)piperidin-3-yl]urea
2-(ethanesulfonyl)-N-[2-(pyridin-2-yl)ethyl]-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-1H-indole-6-carboxamide
4-({4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
3-(2-methyl-1H-indol-1-yl)-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)propanamide
3-[(2R,3R,6R)-5-(pyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
2-[2-(1H-imidazol-4-yl)ethyl]-9-[2-(methylsulfanyl)pyrimidin-4-yl]-2,9-diazaspiro[5.5]undecan-3-one
3-[1-(1-benzofuran-2-ylmethyl)piperidin-4-yl]-N-(3-methoxyphenyl)propanamide
8-(1H-indol-2-ylmethyl)-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-[(diethylamino)methyl]-N-(oxan-3-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]pyrimidin-2-amine
5-[3-(diethylamino)pyrrolidine-1-carbonyl]-1-(3-methylbutyl)-N-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
methyl 1-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}piperidine-4-carboxylate
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(benzyloxy)-1-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]ethan-1-one
1-{[4-(5-methylpyridin-2-yl)piperidin-4-yl]methyl}-2-phenylpiperazine