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ethyl 1-(2H-1,3-benzodioxol-4-ylmethyl)-3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylate
8-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
(2E)-1-[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]-3-(thiophen-2-yl)prop-2-en-1-one
1-(2-oxo-2-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethyl)imidazolidine-2,4-dione
6-[6-hydroxy-4-(1H-1,2,3-triazol-4-ylmethyl)-1,4-diazepan-1-yl]pyridine-3-carboxamide
2-[2,4-bis(prop-2-en-1-yloxy)phenyl]-1H-imidazole
N-[(3R,4S)-1-[4-(piperidine-1-carbonyl)pyridin-2-yl]-4-propylpyrrolidin-3-yl]acetamide
(2R)-2-amino-N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-phenylacetamide
N-{[1-(furan-2-ylmethyl)pyrrolidin-3-yl]methyl}quinoxaline-5-carboxamide
1-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]-3-[5-(thiophen-2-yl)furan-2-yl]propan-1-one
5-(3-chloro-5-fluorobenzoyl)-2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
5-{4-[(2-aminopyridin-3-yl)methyl]-6-hydroxy-1,4-diazepane-1-carbonyl}-1H-pyrrole-3-carbonitrile
4-(2H-1,3-benzodioxol-5-yloxy)-1-(pyrazin-2-yl)piperidine-4-carboxylic acid
4-hydroxy-2-{[4-(2-methoxyethyl)piperazin-1-yl]methyl}quinoline-6-carboxamide
2-[3-(furan-2-yl)-5-oxo-1-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-[(5-methylfuran-2-yl)methyl]acetamide
N4-{[2-(dimethylamino)pyridin-3-yl]methyl}-N1,N1-dimethylpiperidine-1,4-dicarboxamide
2-(2,4-dimethoxy-3-methylphenyl)-4-{[2-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-5-methyl-1,3-oxazole
N-(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)-2-(1H-1,2,3,4-tetrazol-5-yl)acetamide
3-[(1-{5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carbonyl}piperidin-4-yl)oxy]pyridine
N-[2-(dimethylamino)ethyl]-4-(pyrimidin-2-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
1-{7-methyl-12-oxo-3,7,11-triazaspiro[5.6]dodecan-3-yl}-2-phenylethane-1,2-dione
7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decane
N-({3-methyl-7-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(thiophen-3-yl)acetamide
3-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-1-[4-(3-hydroxypiperidin-1-yl)piperidin-1-yl]propan-1-one
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}acetamide
[(3-ethyl-1,2-oxazol-5-yl)methyl]({4-[5-(pyrrolidin-1-yl)pyridazin-3-yl]phenyl}methyl)amine
N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-4-methyl-N-(pyridin-4-ylmethyl)benzamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-3-(1,2-oxazolidin-2-yl)propanamide
N-({7-[(4-methoxy-2,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine-4-carboxamide
3-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-1-(furan-2-ylmethyl)urea
1-[4-(1H-1,3-benzodiazol-1-yl)phenyl]-N-(1-methyl-1H-1,2,3-triazol-4-yl)piperidin-4-amine
2-(2-fluoro-5-methoxyphenyl)-2-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]acetic acid
3-[(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amino]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
2-methoxy-6-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-5-oxo-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
(2S,4S)-4-amino-N-ethyl-1-[2-(1,1,2,2-tetrafluoroethoxy)benzoyl]pyrrolidine-2-carboxamide
N-{[4-(2-methylphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-2-(trifluoromethyl)benzene-1-sulfonamide
{[1-(cyclohexylmethyl)-2-methanesulfonyl-1H-imidazol-5-yl]methyl}[1-(dimethyl-1,3-thiazol-4-yl)ethyl]methylamine
1-[2-(morpholin-4-ylmethyl)piperidin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
1-(cyclopropylmethyl)-5-[(3-phenyl-1H-pyrazol-4-yl)methyl]-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
[(3R,4R)-4-(azepan-1-ylmethyl)-1-[1-(4-methylphenyl)cyclopropanecarbonyl]pyrrolidin-3-yl]methanol
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-[3-(ethoxymethyl)-5-[4-(1H-pyrazol-1-yl)phenyl]-1H-1,2,4-triazol-1-yl]-1-methylpiperidine
5-ethyl-5-(1-{[3-(2-hydroxyethoxy)phenyl]methyl}piperidin-4-yl)-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]imidazolidine-2,4-dione
2,6-difluoro-N-[1-(2-phenylethyl)piperidin-3-yl]benzamide
2-[ethyl({[(3R,4R)-4-(hydroxymethyl)-1-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]pyrrolidin-3-yl]methyl})amino]ethan-1-ol
1-(4-{1-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenyl)-1H-1,2,4-triazole
1-[(3,4-difluorophenyl)methyl]-4-ethyl-1,4-diazepan-5-one
1-(2-{[4-(2,4-dioxoimidazolidin-1-yl)phenyl]formamido}ethyl)piperidine-3-carboxamide
N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-2-(2,2,3,3-tetrafluoropropoxy)acetamide
4-benzyl-3-[1-(1,2-oxazole-3-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one