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2-(3-{[2-(3-methoxyphenyl)piperidin-1-yl]methyl}phenyl)-6-methyl-3,4-dihydropyrimidin-4-one
3-(4-{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}piperazin-1-yl)-2,5-dimethylpyrazine
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1-ethyl-3-methyl-1H-pyrazole-5-sulfonamide
2-(2,2-difluoroethyl)-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
(3S,4R)-3-benzyl-1-[(3-chloro-4-hydroxyphenyl)methyl]-4-methylpiperidin-4-ol
1-methyl-3-(propan-2-yl)-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazole-5-carboxamide
3-{[(cyclohexylmethyl)amino]methyl}-5,6,7-trimethoxy-N,N-dimethylquinolin-2-amine
1-(3-chloro-5-fluorobenzoyl)-4-[1-(pyrrolidin-1-yl)ethyl]piperidine
4-(3-methyl-5-propyl-1-benzofuran-2-carbonyl)piperazin-2-one
4-(1-ethyl-5-oxopyrrolidine-3-carbonyl)-1-[(2-fluorophenyl)methyl]piperazin-2-one
N-(3,4-dimethoxyphenyl)-1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidin-3-amine
methyl 6-({[(1S,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]carbamoyl}amino)-1,2,3,4-tetrahydroquinoline-1-carboxylate
N-[3-(2-fluorophenyl)propyl]-2-(morpholin-3-yl)acetamide
N-benzyl-3-{[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl}-N-methylimidazo[1,2-a]pyridine-2-carboxamide
[(3R,4R)-4-[(dimethylamino)methyl]-1-{6-methylthieno[2,3-d]pyrimidin-4-yl}pyrrolidin-3-yl]methanol
1-(3-{3-[(2-fluorophenyl)methoxy]azetidine-1-carbonyl}phenyl)-1H-pyrazole
4-{3-[2-(methylamino)ethoxy]phenyl}benzonitrile
1-(2-{7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-oxoethyl)pyrrolidin-2-one
(4aR,7aS)-1-(3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-(2-ethylbenzoyl)-2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
N-[2-(1H-indol-1-yl)ethyl]-2-oxo-1-phenylpyrrolidine-3-carboxamide
8-(1-ethyl-1H-pyrazole-5-carbonyl)-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-{3-[methyl(2-phenylethyl)amino]piperidine-1-carbonyl}pyridin-1-ium-1-olate
2-{6-[(3S)-3-(3-methoxyphenyl)piperidin-1-yl]-2-methylpyrimidin-4-yl}ethan-1-amine
(2E)-N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-3-(3-fluorophenyl)prop-2-enamide
N-methyl-2-(1,2-oxazole-3-carbonyl)-N-(1,3-thiazol-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
4-(1-ethyl-3-methyl-1H-pyrazole-4-carbonyl)-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-(1-butyl-1H-imidazol-2-yl)-1-(5-methylthiophene-2-carbonyl)piperidine
(3S,4R)-1-(cyclohexylcarbamoyl)-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
(1S,5R)-3-[(1-propyl-1H-imidazol-2-yl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-(2-methyl-1-benzofuran-7-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-[(3-methylpyridin-2-yl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
5-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]phenyl}-3-ethyl-1,2,4-oxadiazole
(2S,4R)-1-[(2,4-dimethoxyphenyl)methyl]-4-[(4-fluorophenyl)sulfanyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-(piperidin-4-yl)piperidine-3-carboxamide
8-(1H-indol-3-ylmethyl)-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[3-(1,3-thiazol-4-yl)phenyl]quinoxaline-6-carboxamide
4-{[3-(pyridin-2-yl)phenyl]methyl}morpholine-2-carboxylic acid
(1S,5R)-6-(cyclobutylmethyl)-3-[2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-acetyl-8-(2-methyl-6-propylpyrimidin-4-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-4-ol
2-methyl-5-{[3-(3-{pyrazolo[1,5-a]pyrimidin-3-yl}phenyl)-1H-pyrazol-1-yl]methyl}-1,3,4-oxadiazole
2-({3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl}sulfanyl)-1-(4-phenylazepan-1-yl)ethan-1-one
1-ethyl-6-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}-1H-indole
N-[2-methoxy-4-(2-propyl-1H-imidazol-1-yl)phenyl]acetamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-1-[2-(2,2-dimethyloxan-4-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]piperidine-3-carboxamide
ethyl 2-[1-(quinolin-4-ylmethyl)piperidin-2-yl]acetate
1-{2-[1-(2-ethylphenyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-1,2,3,4-tetrazole
N-[1-(2-methoxyphenyl)ethyl]-N-methyl-5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
(1R,3S,5S)-8-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octane