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5-(azepane-1-carbonyl)-1-(butan-2-yl)-N-methyl-N-(naphthalen-1-ylmethyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
3-methyl-5-{1-[(3-phenyl-1,2-oxazol-5-yl)methyl]pyrrolidin-2-yl}-1H-1,2,4-triazole
N-(1-propyl-1H-1,2,3-triazol-4-yl)-2-[4-(1,3-thiazol-2-yl)-1H-pyrazol-1-yl]acetamide
N-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propyl]-2,2-dimethylpyrrolidin-3-amine
5-hydroxy-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]pyrazine-2-carboxamide
1-(4-cyclopropanecarbonyl-1,4-diazepan-1-yl)-2-(2,4,7-trimethyl-1H-indol-3-yl)ethan-1-one
{2-[2-benzyl-5-oxo-4-(3-phenylphenyl)piperazin-1-yl]ethyl}urea
2-ethyl-N-[1-(1H-imidazol-1-yl)-3-methylbutan-2-yl]pyrimidine-5-carboxamide
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}-4-(methylsulfanyl)benzamide
2-butyl-1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-2,5-dihydro-1H-pyrrole
3-[2-(4-fluorophenyl)morpholine-4-carbonyl]-4-phenyl-1H-pyrazol-5-amine
N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
6-{[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]amino}-2-methylheptan-2-ol
1-[(3,5-dimethylphenyl)methyl]-4-(5-fluoro-2-methylbenzoyl)piperazin-2-one
(2E)-3-(3,4-dimethoxyphenyl)-1-(3-{5-methyl-2-[(pyridin-3-ylmethyl)sulfanyl]pyrimidin-4-yl}piperidin-1-yl)prop-2-en-1-one
5-{5-methylimidazo[1,2-a]pyridin-2-yl}-3-(2-methylpropyl)-1H-1,2,4-triazole
2-[4-(3,5-dimethylphenyl)-3-oxopiperazin-1-yl]quinoline-4-carboxylic acid
(1S,9aR)-1-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-octahydro-1H-quinolizine
(2S,4S)-4-amino-N-methyl-1-(piperidine-1-sulfonyl)pyrrolidine-2-carboxamide
2-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-5-(1H-imidazol-1-ylmethyl)pyridine
[1-(4-aminopyrimidin-2-yl)-3-[(4-fluorophenyl)methyl]piperidin-3-yl]methanol
2-(2-methoxyphenyl)-1-[1-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1H-imidazole
2-(5-{5H,6H,7H-cyclopenta[b]pyridin-3-yl}-1-[(4-fluorophenyl)methyl]-1H-1,2,4-triazol-3-yl)acetamide
(2S,4R)-1-[(2,5-difluorophenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
(1S,6R)-9-(oxan-4-yl)-3,9-diazabicyclo[4.2.1]nonan-4-one
{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[(1-methylpiperidin-3-yl)methyl]amine
(2,1,3-benzoxadiazol-4-ylmethyl)[(1-methyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)amine
1-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]-3-(4H-1,2,4-triazol-4-yl)propan-1-one
N-{[7-(cyclohex-3-en-1-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-2,5-dimethylfuran-3-carboxamide
(4aR,8aS)-1-(2H-1,3-benzodioxol-5-ylmethyl)-6-(2-methoxybenzoyl)-decahydro-1,6-naphthyridin-2-one
3-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-3,9-diazaspiro[5.6]dodecan-10-one
2,2-dimethyl-3-{[1-propyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}propan-1-ol
N-(1-{1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-phenoxypropanamide
4-{3-[4-(5-amino-3-methyl-1H-pyrazol-1-yl)phenyl]-1,2,4-oxadiazol-5-yl}-1-(propan-2-yl)pyrrolidin-2-one
1-benzyl-6-(cyclopropylmethoxy)-4-(1-ethylpiperidin-4-yl)-1,4-diazepan-2-one
2-[3-({methyl[1-(pyridin-3-yl)ethyl]amino}methyl)phenoxy]acetamide
2-[4-(1H-indol-5-yl)-1H-pyrazol-1-yl]-N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
1-[(2-butyl-1H-imidazol-4-yl)methyl]-N-(2,3-dihydro-1,4-benzodioxin-6-yl)piperidin-3-amine
2-amino-6-(1-methyl-1H-pyrrol-3-yl)-4-[3-(1H-pyrazol-1-ylmethyl)phenyl]pyridine-3-carbonitrile
(1S,5R)-3-[3-(2-methoxyphenyl)-1H-pyrazole-5-carbonyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl[(2-methyl-1,3-thiazol-4-yl)methyl]{[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}amine
2-({5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-yl}amino)acetamide
1-(cyclohexylmethyl)-3-hydroxy-3-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}piperidin-2-one
5-[8-(3-methylbutyl)-9-oxo-2,8-diazaspiro[5.5]undecane-2-carbonyl]pyridine-2-carbonitrile
2-hydroxy-6-methyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}pyridine-3-carboxamide
1-(cyclohexylmethyl)-3-hydroxy-3-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)piperidin-2-one
5-(1H-imidazol-2-ylmethyl)-N-phenyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
2,3,5-trimethyl-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
(3R,9R)-11-(4-methylbenzoyl)-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide