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5-(1-butanoylpiperidin-4-yl)-5-(3-methylbutyl)-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
3-methyl-3-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]piperidine
8-[(6-chloropyridin-2-yl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
N-benzyl-3-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-N-methylpropanamide
N-cyclohexyl-3-(hydroxymethyl)-3-(3-methoxypropyl)piperidine-1-carboxamide
2-[4-(2-amino-6-methylpyrimidin-4-yl)-1-[(4-methylphenyl)methyl]piperazin-2-yl]ethan-1-ol
3-(2,3-dihydro-1-benzofuran-7-yl)-5-(pyrrolidine-1-sulfonyl)benzoic acid
2-methoxy-5-methyl-N-(1,4-oxazepan-6-ylmethyl)benzene-1-sulfonamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]benzamide
5-(2,1,3-benzoxadiazole-4-sulfonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
(5S,9aS,9bS)-2-[(2-methoxyphenyl)methyl]-5-[4-(trifluoromethyl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[2-methyl-5-(methylcarbamoyl)phenyl]-4-(pyridin-4-ylmethyl)-1,4-diazepane-1-carboxamide
N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]-2,3-dihydro-1,4-benzodioxine-2-carboxamide
2-(2-chloro-6-methoxyphenyl)-2-(4-propylpiperazin-1-yl)acetic acid
2-ethyl-8-(2-methyl-1,3-thiazole-5-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
2-(dimethyl-1,2-oxazol-4-yl)-1-[4-(2-methylphenyl)-1,4-diazepan-1-yl]ethan-1-one
5-ethyl-6-methyl-N4-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}pyrimidine-2,4-diamine
1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-3-{3-[(furan-2-ylmethyl)sulfanyl]propyl}urea
1-methyl-N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}azepane-2-carboxamide
N-methyl-N-[(4-methylphenyl)methyl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
15-methyl-12-[4-(propan-2-yl)piperazine-1-carbonyl]-9-(thiophen-3-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaen-13-one
N-ethyl-2-[(4-methoxyphenyl)methyl]-N-(pyridin-4-ylmethyl)-1,3-benzoxazole-6-carboxamide
2-(4-benzylmorpholin-2-yl)-6-(piperidin-4-yl)-3,4-dihydropyrimidin-4-one
1-ethyl-5-oxo-N-{2-[2-(trifluoromethoxy)phenyl]ethyl}pyrrolidine-3-carboxamide
N-[(4-fluorophenyl)methyl]-N-(2-hydroxyethyl)-6-methoxy-3-methyl-1-benzofuran-2-carboxamide
4-(2,3-dimethyl-1H-indole-7-carbonyl)-1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane
methyl 3-(4-methyl-2-oxopentanoyl)-9-[2-(morpholin-4-yl)ethoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-cyclopropyl-6-[4-(2-methoxyphenyl)-2-methylpiperazine-1-carbonyl]-1,3-benzoxazole
N-[3-(methylsulfanyl)propyl]-2-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)-1,3-oxazole-4-carboxamide
2-methyl-5-{2-[2-(thiophen-2-yl)ethyl]piperidine-1-carbonyl}-3,4-dihydropyrimidin-4-one
1-{2-hydroxy-3-[4-methoxy-2-({methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}methyl)phenoxy]propyl}piperidin-4-ol
4-benzyl-3-ethyl-1-({2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidin-5-yl}methyl)-1,4-diazepan-5-one
2-[(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)methyl]pyridine-3-carboxylic acid
1-(2-fluorophenyl)-3-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}urea
4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-N-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-1-carboxamide
2-cyclopropanecarbonyl-8-[(2-ethylpyrimidin-4-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-[4-hydroxy-4-(2-methylquinolin-6-yl)piperidin-1-yl]-3-(methylsulfanyl)propan-1-one
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-3-propanamidobenzamide
N2-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-5-fluoro-N4,N4-dimethylpyrimidine-2,4-diamine
{1-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]-3-(cyclopropylmethyl)piperidin-3-yl}methanol
2-methoxy-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
(2S)-1-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
5-ethyl-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}thiophene-3-carboxamide
1-methyl-4-[4-(piperidin-3-ylmethyl)benzoyl]-1,4-diazepane
6-(2-aminoethyl)-N-[(3-fluorophenyl)methyl]-2-methylpyrimidin-4-amine
(3R,4R)-4-(azepan-1-yl)-1-(8-methoxy-4-methylquinolin-2-yl)piperidin-3-ol
1-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}-3-(1-methylpiperidin-3-yl)propan-1-one
N-[2-(4-fluorobenzenesulfonyl)ethyl]-4-(1H-pyrazol-3-yl)benzamide
N-[2-(benzylsulfanyl)ethyl]-1-(methoxymethyl)cyclobutane-1-carboxamide
N-[1-(furan-2-yl)ethyl]-9-methoxy-N-methyl-3-(3-methylbutyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide