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5-benzyl-5-[1-(2-methylbenzoyl)piperidin-4-yl]-3-[2-(pyrrolidin-1-yl)ethyl]imidazolidine-2,4-dione
N-cyclopentyl-N'-{2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}butanediamide
3-(2-methylpropyl)-N-(pyridin-3-ylmethyl)-N-(thiophen-3-ylmethyl)-1,2-oxazole-5-carboxamide
[(2-ethoxyphenyl)methyl](methyl)[1-(pyrazin-2-yl)propan-2-yl]amine
1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-8-[(1-methyl-1H-indol-3-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-(3-fluorobenzenesulfonyl)-3,6-diazabicyclo[3.2.2]nonane
8-methoxy-N-[3-(pyridin-3-yloxy)propyl]-3,4-dihydro-2H-1-benzopyran-3-amine
3-(4-methyl-1,3-thiazol-5-yl)-N-{[3-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}propanamide
N,N,4,5-tetramethyl-6-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]pyrimidin-2-amine
(3R,4S)-1-[2-(benzyloxy)benzoyl]-4-cyclopropylpyrrolidin-3-amine
4-[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]pyrimidin-2-amine
2-(3-fluoro-4-methoxyphenyl)-2-[4-(pyridin-2-ylmethoxy)piperidin-1-yl]acetic acid
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-6-methoxypyrimidin-4-amine
8-[2-(methylsulfanyl)pyrimidin-4-yl]-2-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
5-benzyl-5-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}imidazolidine-2,4-dione
5-methyl-N-(2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)-1-propyl-1H-pyrazole-4-carboxamide
3-(2-fluorophenyl)-N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylpropanamide
5-{[methyl({3-[2-(4-{4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}piperazin-1-yl)ethoxy]phenyl}methyl)amino]methyl}pyrrolidin-2-one
(4aR,8aR)-2-(dimethyl-1,3-oxazole-5-carbonyl)-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
N-(butan-2-yl)-2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carboxamide
(1S,4S)-2-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-2-azabicyclo[2.2.1]heptane
N-[2-(1-methylpyrrolidin-2-yl)ethyl]-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
methyl 2-{5-methyl-2-[(oxolan-2-ylformamido)methyl]-2,3-dihydro-1-benzofuran-7-yl}benzoate
4-phenyl-3-[1-(pyridin-3-ylmethyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-1-(2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}morpholin-4-yl)ethan-1-one
N-ethyl-5-{2-[2-(1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}pyrimidin-2-amine
4-hydroxy-N-[2-(1H-imidazol-4-yl)ethyl]-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxamide
2-(3-chlorophenoxy)-N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methylpropanamide
N-[2-(2,4-dimethoxyphenyl)ethyl]-5-phenyl-1,2,4-triazin-3-amine
N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-N-(prop-2-en-1-yl)-2-{[1,2,4]triazolo[4,3-b]pyridazin-6-yloxy}acetamide
(2S,4S)-4-amino-1-methyl-N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]pyrrolidine-2-carboxamide
2-(4-fluorophenyl)-N-[(3R,4R)-3-hydroxypiperidin-4-yl]benzamide
1-(3-methoxy-5-methylthiophene-2-carbonyl)-4-phenylpiperidin-4-ol
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-5-(methoxymethyl)furan-2-carboxamide
N-methyl-3-[methyl(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)amino]butanamide
methyl 2-[(4-chlorophenyl)sulfamoyl]-6-cyclohexanecarbonyl-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
methyl 4-[5-methyl-4-({methyl[1-(1,2-oxazol-3-yl)ethyl]amino}methyl)-1,3-oxazol-2-yl]benzoate
4-(2-methylpiperidin-1-yl)-N-[3-(morpholin-4-yl)propyl]pyridine-2-carboxamide
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-(3-ethyl-4-methyl-1-phenyl-1H-pyrazol-5-yl)acetamide
1-(5-cyclopropyl-1-{8-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-1H-pyrazole-4-carbonyl)-N,N-dimethylpyrrolidin-3-amine
2-{3-[(4-butyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}-5-methylpyrazine
N-[2-(5-cyano-2-methyl-1H-indol-3-yl)ethyl]-3-(pyridin-2-yl)-1H-pyrazole-5-carboxamide
1-{1-[(4-chlorophenyl)methyl]pyrrolidin-3-yl}piperidine
(3S,4S)-1-(2,1,3-benzothiadiazol-5-ylmethyl)-4-(morpholin-4-yl)pyrrolidin-3-ol
N,N-bis(1,3-oxazol-4-ylmethyl)-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]acetamide
N-cyclopentyl-1-(diphenylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-{3-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decane-4-sulfonyl]-4-methoxyphenyl}acetic acid
1-[(4-chlorophenyl)methyl]-N-[2-(3-phenylpiperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}-N-[(5-methylpyrazin-2-yl)methyl]benzamide
1-(benzyloxy)-8-[3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanoyl]-1,8-diazaspiro[4.5]decan-2-one