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5-(3-{1-[(6-methylpyridin-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)-2-(4H-1,2,4-triazol-4-yl)pyridine
1-methyl-N-{[5-methyl-2-(4-phenylmethanesulfonamidophenyl)-1,3-oxazol-4-yl]methyl}-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
1-(adamantan-1-yl)-4-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperazine
methyl 2-oxo-8-[(4-phenylphenyl)methyl]-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
2-[5-(1,7-dimethyl-1H-indol-3-yl)-4-phenyl-1H-imidazol-1-yl]ethan-1-amine
4'-(cyclopropylmethyl)-3'-oxo-N-pentyl-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-carboxamide
2-benzyl-4-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)morpholine
methyl 1-[(3R,5S)-1-[(3-methylthiophen-2-yl)methyl]-5-(4-phenylpiperazine-1-carbonyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
1-{1-[(2-chlorophenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
(2R,6R)-11-methoxy-4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
{3-[(4-fluorophenyl)methyl]-1-[(1-methyl-1H-indol-3-yl)methyl]piperidin-3-yl}methanol
[(2-chlorophenyl)methyl]({[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl})methylamine
6-methoxy-N-(2-methoxyethyl)-1-methyl-N-(pyridin-3-ylmethyl)-1H-indole-2-carboxamide
1-(benzyloxy)-8-(3-methylbutanoyl)-1,8-diazaspiro[4.5]decan-2-one
(4aS,7aR)-1-{[2-(benzylamino)pyrimidin-5-yl]methyl}-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-(methoxymethyl)-N-[4-(4-{[(2-methoxyphenyl)formamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]thiophene-2-carboxamide
7-methyl-2-{[4-(pyrimidin-2-yloxy)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
5-ethyl-2-{4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}pyrimidine
(2S,4R)-1-(2H-1,3-benzodioxol-5-ylmethyl)-N-[2-(dimethylamino)ethyl]-4-[(4-methylpyrimidin-2-yl)sulfanyl]pyrrolidine-2-carboxamide
N-[1-(4-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}phenyl)-1H-pyrazol-4-yl]oxane-4-carboxamide
1-(4-methoxy-3,5-dimethylphenyl)-3-[4-(pyrrolidin-1-yl)butyl]urea
methyl 2-{3-[3-(1,3-thiazol-2-yl)phenyl]-1H-pyrazol-1-yl}acetate
2-[methyl(piperidin-4-yl)amino]-N-{[2-(trifluoromethyl)phenyl]methyl}acetamide
1-[(4aS,8aS)-4a-hydroxy-decahydroisoquinolin-2-yl]-3-(benzenesulfonyl)propan-1-one
2-amino-4-(2-butyl-1H-imidazol-4-yl)-6-(3,5-dimethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
8-{[5-(4-chlorophenyl)furan-2-yl]methyl}-1-methoxy-1,8-diazaspiro[4.5]decan-2-one
{1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]azepan-2-yl}methanol
4-fluoro-3-{3-methyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decane-8-carbonyl}benzene-1-sulfonamide
2-(dimethylamino)-N-[2-(2-methoxyphenyl)ethyl]-2-(3-methylphenyl)acetamide
(2S)-2-amino-N-{5H,6H,7H,8H,9H,10H,11H-cycloocta[b]indol-2-ylmethyl}-4-hydroxybutanamide
N-[2-(1H-imidazol-1-yl)ethyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
4-(3-hydroxy-3-methylbutyl)-N-[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]benzamide
N-(6-hydroxy-6-methylheptan-2-yl)-3-{2-[(4-methylphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
4-(3-methylphenoxy)-1-(thiophene-3-carbonyl)piperidine-4-carboxylic acid
3-cyclobutyl-5-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}-1H-1,2,4-triazole
1-{1-[4-(1-benzofuran-2-yl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carbonyl}-4-methyl-1,4-diazepane
2,3-dimethyl-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}quinoxaline-6-carboxamide
3-[methyl({[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl})amino]propan-1-ol
N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
(1S,5R)-3-{2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-({1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]piperidin-3-yl}methyl)cyclopropanesulfonamide
3-{2-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]propanamide
9-(2-amino-5-butyl-6-methylpyrimidin-4-yl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
(2E)-N-[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-3-(thiophen-2-yl)prop-2-enamide
N-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-1-(pyridin-4-ylmethyl)piperidin-4-amine
N-benzyl-3-(1-methylpiperidin-2-yl)-N-[(3-methylpyridin-2-yl)methyl]propanamide
ethyl 1-({1-[(2-fluorophenyl)methyl]-7-methoxy-2-oxo-1,2-dihydroquinolin-3-yl}methyl)piperidine-3-carboxylate
(hexan-2-yl)({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)amine
9-methoxy-3-[(4-methoxy-3-methylphenyl)methyl]-7-oxo-N-(thiophen-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(4aS,7aR)-1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-4-(cyclopropylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione