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5-ethanesulfonamido-N-[(1-ethylpyrrolidin-2-yl)methyl]-1-methyl-2-phenyl-1H-1,3-benzodiazole-7-carboxamide
1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-4-[2-(methylsulfanyl)ethyl]piperazine
N-methyl-5-(1-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}pyrrolidin-2-yl)thiophene-2-carboxamide
4-(2-fluorophenyl)-2-{4-[4-(piperidin-1-yl)piperidine-1-carbonyl]-5-(propan-2-yl)-1H-pyrazol-1-yl}pyrimidine
1-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-1H-indazole-3-carboxylic acid
N-benzyl-7-cyclobutaneamido-N-ethyl-1-methyl-2-(pyridin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
2-{[2-amino-6-(5-methylpyridin-3-yl)pyrimidin-4-yl]amino}ethan-1-ol
6-(2,5-dimethylfuran-3-yl)-7-methyl-2-[(3R)-3-methylpiperazine-1-carbonyl]-7H,8H-imidazo[1,2-a]pyrazin-8-one
methyl 2-[ethyl(2-methylprop-2-en-1-yl)sulfamoyl]-6-[(2-fluoro-5-methoxyphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-cyclopropyl-2-{4-[(3-fluorophenyl)methyl]-3-oxopiperazin-1-yl}pyridine-4-carboxamide
4-{[3-(2-ethylphenoxy)azetidin-1-yl]methyl}-1-methyl-1H-pyrrole-2-carbonitrile
1-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}-2-(1H-indol-3-yl)ethan-1-one
4-[(dimethylsulfamoyl)amino]-1-[2-(4-methoxyphenyl)ethyl]pyrrolidin-2-one
2-methyl-1-{4-[(4-methylphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}propan-1-ol
4-(1-ethyl-1H-imidazol-2-yl)-1-(oxolane-2-carbonyl)piperidine
2-[1-(3-methoxypropyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]-N-methyl-N-(propan-2-yl)acetamide
7-(cyclohex-3-ene-1-carbonyl)-N,N-dimethyl-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
6-{3-oxo-3-[4-(2-phenoxyethyl)piperazin-1-yl]propyl}-2,3-dihydropyridazin-3-one
1-(7-methoxy-4-methylquinazolin-2-yl)-N-[(1R)-1-(4-methoxyphenyl)ethyl]piperidine-3-carboxamide
(1R,3S)-3-(2-hydroxyethoxy)-7-(2-methyl-1H-pyrrole-3-carbonyl)-7-azaspiro[3.5]nonan-1-ol
methyl (2S,4S)-4-({[(1R)-1-(4-chlorophenyl)ethyl]carbamoyl}amino)-1-methylpyrrolidine-2-carboxylate
N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-1-(propan-2-yl)piperidine-4-carboxamide
5-({spiro[indene-1,4'-piperidine]-1'-yl}carbonyl)-7H-[1,3]thiazolo[3,2-a]pyrimidin-7-one
2-[cyclopentyl(methyl)amino]-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
N-{[3-(3-fluorophenyl)-1,2-oxazol-5-yl]methyl}-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propanamide
4-hydroxy-N-methyl-2-(4-methylphenyl)-N-[1-(pyridin-2-yl)propyl]pyrimidine-5-carboxamide
(3aR,6aS)-5-({2-[2-(dimethylamino)ethoxy]phenyl}methyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{4-[3-oxo-3-(4-phenylpiperazin-1-yl)propyl]piperidin-1-yl}pyridine-3-carbonitrile
2-{[2-methanesulfonyl-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}-1,2,3,4-tetrahydroisoquinoline
2-chloro-4-({4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}methyl)phenol
2-(dimethyl-1,2-oxazole-4-carbonyl)-7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decane
{9-[(3-methyl-1,2-oxazol-5-yl)methyl]-3-(1,3-thiazol-4-ylmethyl)-3,9-diazaspiro[5.5]undecan-1-yl}methanol
6-(4-cyclopentyl-1,4-diazepane-1-carbonyl)pyridin-2-amine
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N-methyl-2-(morpholin-4-yl)pyridine-3-carboxamide
(1R,3S,5S)-8-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}-8-azabicyclo[3.2.1]octan-3-ol
1-[1-(cyclopropylmethyl)-1H-pyrazol-5-yl]-3-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}urea
(2R,6R)-4-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-[5-(morpholin-4-yl)pentyl]-3-(3,4,5-trifluorophenyl)urea
1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-4-(2,6-dimethylpyridin-4-yl)piperazine
1-tert-butyl-4-({methyl[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}methyl)pyrrolidin-2-one
3-[(3-methoxypropyl)sulfamoyl]-N-[(1-methylpiperidin-2-yl)methyl]benzamide
1-{3-[3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-3-oxopropyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
({1-[(2-fluorophenyl)methyl]-2-methanesulfonyl-1H-imidazol-5-yl}methyl)(methyl)(thiophen-2-ylmethyl)amine
3-({[1-(furan-2-yl)ethyl](methyl)amino}methyl)-7-methoxy-1,2-dihydroquinolin-2-one
N5-(2,3-dihydro-1H-inden-1-yl)-N6-(3-methoxypropyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
2-{1-[(4-fluorophenyl)methyl]-4-(2,2,3,3-tetramethylcyclopropanecarbonyl)piperazin-2-yl}ethan-1-ol
4-methyl-2-[1-(4-methylpyrimidine-5-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
N-(3-fluoro-2-methylphenyl)-2-{methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}acetamide
N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-amine
4-[2-(2-oxopiperidin-1-yl)acetyl]-1-(2-phenylethyl)piperazin-2-one