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2-[1-cyclopentyl-3-(3-fluorophenyl)-2,5-dioxopyrrolidin-3-yl]-N-[2-(diethylamino)ethyl]-N-ethylacetamide
N-methyl-N-(quinolin-5-ylmethyl)cyclohex-3-ene-1-carboxamide
{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}({[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl})amine
N-[(6-chloropyridin-3-yl)methyl]-N,1-dimethyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-benzyl-8-(2,3-dihydro-1H-inden-2-yl)-3-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3R,4R)-1-[(4,5-dimethylfuran-2-yl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-ol
(3R,4R)-4-(azepan-1-yl)-1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidin-3-ol
2-chloro-N-{[5-(5-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
3-{1-[2-(2H-1,3-benzodioxol-5-yloxy)acetyl]piperidin-4-yl}-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{[4-(2-methoxyphenyl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}ethan-1-ol
2-(4-fluorophenyl)-2-hydroxy-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
4-[1-(2-ethoxyacetyl)piperidin-3-yl]benzoic acid
4-ethyl-1-[(3-phenyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
N-[(1-cyclohexylpiperidin-3-yl)methyl]-1-phenyl-N-(pyridin-3-ylmethyl)cyclopropane-1-carboxamide
(1S,5R)-3-{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}-3,9-diazabicyclo[3.3.2]decan-10-one
1-[2-methoxy-5-({[(2-methylphenyl)methyl]amino}methyl)phenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
[(2S,4R,5R)-5-(2-fluorophenyl)-1-methyl-4-[({trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)methyl]pyrrolidin-2-yl]methanol
2-{[3-(hydroxymethyl)pyrrolidin-1-yl]sulfonyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
5-(2-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-oxoethyl)-3-propylimidazolidine-2,4-dione
3-fluoro-N-{2-[3-(thiomorpholin-4-ylmethyl)phenoxy]propyl}benzamide
4-(1-{[4-(1H-imidazol-1-yl)phenyl]methyl}pyrrolidin-2-yl)-3,5-dimethyl-1,2-oxazole
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[(1-ethyl-1H-imidazol-5-yl)methyl]-1H-pyrazole-3-carboxamide
3-(1-benzyl-1H-imidazol-2-yl)-1-[3-(2-methyl-1H-imidazol-1-yl)propyl]piperidine
3-(2H-1,3-benzodioxole-5-carbonyl)-1-[(2,3,6-trifluorophenyl)methyl]piperidine
8-(1,3-benzothiazol-2-ylmethyl)-1-[2-(4-methoxyphenyl)ethyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[1-cyclopentyl-3-(3-fluorophenyl)-2,5-dioxopyrrolidin-3-yl]-N,N-bis(prop-2-en-1-yl)acetamide
7-methoxy-2-{3-[3-(methoxymethyl)piperidine-1-carbonyl]piperidin-1-yl}-4-methylquinazoline
1-(2-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}pyrimidin-4-yl)pyrrolidin-3-ol
3-[2-(propan-2-ylsulfanyl)phenyl]-1-{3-[(pyridin-3-yl)amino]propyl}urea
5-{1-[(2-butyl-1H-imidazol-4-yl)methyl]piperidin-4-yl}-3-cyclopentyl-5-[(4-fluorophenyl)methyl]imidazolidine-2,4-dione
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-3-(3-methyl-1H-pyrazol-1-yl)propanamide
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(pyridin-3-yloxy)propyl]acetamide
3-(1H-1,3-benzodiazol-1-yl)-N-[(3R,4R)-3-hydroxypiperidin-4-yl]propanamide
4-({[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)-2,6-dimethoxyphenol
3-(3-methylphenyl)-5-{2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1,2,4-oxadiazole
N-[2-(benzylsulfanyl)ethyl]-6-fluoro-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
3-{1-[(5-chlorofuran-2-yl)methyl]piperidin-2-yl}propanoic acid
methyl({[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl})(pyrimidin-4-ylmethyl)amine
ethyl 4-[(4-chlorophenyl)methyl]-1-[(3-ethoxy-3-oxopropyl)carbamoyl]piperidine-4-carboxylate
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-3-(pyridin-2-yl)propanamide
2-{4-[(5-ethylfuran-2-yl)methyl]-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N4-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N2,N2-dimethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
2-(furan-3-carbonyl)-1-(2-methylpropyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
3-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-4,5,6,7-tetrahydro-1-benzofuran-4-one
2-{2-[(3-ethylmorpholin-4-yl)methyl]-4-(pyridin-2-yl)phenoxy}acetic acid
5-(2-{4-[5-(oxan-2-yl)thiophen-2-yl]-1H-1,2,3-triazol-1-yl}ethyl)-1,3,4-thiadiazol-2-amine
[(3,5-dichloropyridin-4-yl)methyl](methyl)[1-(4-methylpyridin-2-yl)propan-2-yl]amine
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
ethyl 4-[1-(thiophen-3-ylmethyl)piperidin-3-yl]piperazine-1-carboxylate