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6-[(2S)-4-methyl-2-(propan-2-yl)piperazin-1-yl]-N-(thiophen-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
2-(2-{[(furan-2-ylmethyl)(3-methylbutan-2-yl)amino]methyl}phenoxy)ethan-1-ol
7-(propan-2-yl)-N-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
2-phenoxy-1-{3-[1-(pyrimidin-2-yl)piperidin-4-yl]pyrrolidin-1-yl}ethan-1-one
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-2-(4-methyl-1,4-diazepan-1-yl)acetamide
N-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-methyl-6-oxo-1-(pyridin-2-ylmethyl)-N-(thiophen-3-ylmethyl)piperidine-3-carboxamide
4-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-1-(2-phenylethyl)piperazin-2-one
4-{[({6-chloro-2-methylimidazo[1,2-a]pyridin-3-yl}methyl)(methyl)amino]methyl}-1-cyclopentylpyrrolidin-2-one
1-[(1-methyl-1H-imidazol-5-yl)methyl]-4-[1-(naphthalen-1-yl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridine
2-[4-(5,6-dimethylpyrazin-2-yl)phenyl]-2-methylpropanenitrile
3-(1,2-dihydroacenaphthylene-5-carbonyl)-1-(1,3-thiazole-5-carbonyl)piperidine
2-(dimethylamino)-2-(2-fluorophenyl)-N-{2-[methyl(phenyl)amino]ethyl}acetamide
4-(4-methyl-1H-pyrazol-1-yl)-1-(pyridine-3-sulfonyl)piperidine-4-carboxylic acid
3-(1-methyl-1H-pyrazol-4-yl)-1-[2-(thiophen-2-yl)azetidin-1-yl]propan-1-one
N-(1-{2-[4-(3-methoxyphenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-3-phenoxypropanamide
(2E)-3-(3,4-dimethoxyphenyl)-N-{[7-(6-methoxypyridazin-3-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}prop-2-enamide
2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]-1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]ethan-1-one
5-[(3R,4S)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidine-1-carbonyl]pyrazin-2-ol
2,5-dimethoxy-N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]benzamide
3-[(2-fluoro-4-methoxyphenyl)methyl]-9-methoxy-10-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
1-(1-methylpiperidin-4-yl)-N-[(2-methylpyridin-4-yl)methyl]piperidine-3-carboxamide
(3aR,7aS)-2-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
N-[1-(4-fluorophenyl)propyl]-1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
4-[4-(2-methylpropyl)phenyl]-7-(2-oxoimidazolidin-1-yl)-1,2,3,4-tetrahydroquinolin-2-one
4-[1-(propan-2-yl)-1H-imidazol-2-yl]-1-[2-(trifluoromethyl)benzoyl]piperidine
1-cycloheptyl-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N-methyl-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
(3S,5R)-5-[(pyridin-3-ylmethyl)carbamoyl]-1-(pyrimidin-2-yl)piperidine-3-carboxylic acid
3-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-3-methyl-1-[4-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]urea
1-[(2,4-difluorophenyl)methyl]-4-{imidazo[1,2-b]pyridazin-6-yl}piperazine
4-(4-chlorophenyl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}butanamide
1-(3-{[methyl(oxan-4-yl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
N-[3-(furan-2-yl)phenyl]-1-(5-methyl-1,3-oxazole-4-carbonyl)piperidine-4-carboxamide
4-methoxy-2-({4-[5-(3-methylphenyl)-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}methyl)phenol
N-[(1S,2R)-2-[(1-ethylpiperidin-4-yl)amino]cyclobutyl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
1-(4-{3-[2-(3-methoxyphenyl)ethyl]piperidine-1-carbonyl}piperidin-1-yl)ethan-1-one
1-{4-[3-(3-methoxyphenoxy)azetidin-1-yl]-4-oxobutyl}pyrrolidin-2-one
1,2-dimethyl-3-(3-phenylpiperazine-1-carbonyl)-1H-indol-5-ol
N-{2-[5-(hydroxymethyl)-1,2,4-oxadiazol-3-yl]ethyl}-3-methylthiophene-2-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-6-(piperidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
1-[3-(1H-imidazol-2-yl)piperidin-1-yl]-2-{2-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-{[4-(2-methylphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}benzamide
2-hydroxy-N-[3-(2-methyl-1H-imidazol-1-yl)propyl]-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
(4aR,7aS)-1-(2-hydroxyethyl)-4-[2-(1H-indol-1-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(1-cyclohexyl-1H-1,2,4-triazol-5-yl)-N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)propanamide
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(thiophene-2-carbonyl)piperazine
3-{[(2,2-dimethylpropyl)amino]methyl}-3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
N-(dimethyl-1,2-oxazol-4-yl)-4-({3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)benzamide
9-butyl-3,9-diazaspiro[5.6]dodecane