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N-ethyl-2-[3-(2-methylphenoxymethyl)piperidin-1-yl]pyridine-4-carboxamide
(2R)-3-(benzyloxy)-2-[4-phenyl-5-(pyridin-4-yl)-1H-imidazol-1-yl]propan-1-ol
1-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]azocane
N-[1-(7-{[3-(benzyloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]pyridine-3-carboxamide
3-cyclohexyl-5-{[2-(oxolan-3-yl)-1H-imidazol-1-yl]methyl}-1,2,4-oxadiazole
3-(2H-1,3-benzodioxol-5-yl)-N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-3-phenylpropanamide
1-(4-{[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
5-methoxy-4-(1-methyl-1H-pyrazol-5-yl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}pyrimidin-2-amine
(2R,3S,6R)-5-(4-methyl-1H-pyrrole-2-carbonyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(furan-2-carbonyl)piperazine
2-(4-fluorophenyl)-4-[4-(pyridin-3-yl)pyrimidin-2-yl]morpholine
N-({3-methyl-7-[3-(2-oxopyrrolidin-1-yl)benzoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-3-carboxamide
{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)methylamine
4-[2-(2,5-dioxoimidazolidin-1-yl)acetyl]-1-phenylpiperazine-2-carboxylic acid
(2S)-2-amino-1-(4-cyclopentyl-1,4-diazepan-1-yl)-3-(4-hydroxyphenyl)propan-1-one
2-amino-6-(2,2-dimethylcyclopropyl)-4-(2-methoxypyrimidin-5-yl)-5-methylpyridine-3-carbonitrile
N-({7-[2-(2,6-difluorophenyl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)oxane-4-carboxamide
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-(propane-1-sulfonyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}(methyl)(thiophen-2-ylmethyl)amine
(4aS,7aR)-1-[3-(1H-imidazol-2-yl)benzoyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[(4-fluorophenyl)methyl]-1-(2-methoxyethyl)-3-(propan-2-yl)-1,4-diazepan-5-one
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-5-methylpyrazolo[1,5-a]pyrimidin-7-amine
5-ethyl-N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
6-(2-aminoethyl)-2-methyl-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyrimidin-4-amine
2-(2H-1,3-benzodioxole-5-carbonyl)-1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
1-(3-cyclohexylpropanoyl)-4-ethyl-1,4-diazepan-5-one
2-{3-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-3-oxopropyl}-2,3-dihydro-1H-isoindol-1-one
2-cyclopentyl-N-(2-methoxyethyl)-N-{[6-methyl-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}acetamide
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-(2-methyl-1H-imidazol-1-yl)butanamide
2-[2,5-dioxo-3-phenyl-1-(thiophen-2-ylmethyl)pyrrolidin-3-yl]-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
4-(1-hydroxy-3-phenylpropyl)-N-(5-methyl-1,3,4-thiadiazol-2-yl)piperidine-1-carboxamide
9-[1-(benzenesulfonyl)cyclopropanecarbonyl]-3-oxa-9-azaspiro[5.5]undecane
1-benzoyl-N-[2-methoxy-2-(thiophen-2-yl)ethyl]piperidin-4-amine
ethyl({[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]amine
methyl 1-({4-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidine-2-carboxylate
N-[3-methyl-1-(2-methylphenyl)-1H-pyrazol-5-yl]-2-[3-(3-methylpyrazin-2-yl)-1H-pyrazol-1-yl]acetamide
4-{[2-(pentan-3-yl)-1H-imidazol-1-yl]methyl}pyridine
2,8-dimethyl-4-(thiomorpholine-4-carbonyl)quinoline
4-ethyl-5-methyl-2-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidine
1-[2-(4-chlorophenyl)ethyl]-N-ethyl-6-oxo-N-(propan-2-yl)piperidine-3-carboxamide
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-4,6-dimethyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
2-amino-4-{4-[3-(dimethylamino)propoxy]phenyl}-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-{4-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]morpholin-3-yl}-N-propylacetamide
3-(5-chloro-2-methoxybenzoyl)-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidine
1-cyclopentyl-3-(2-methylphenyl)-3-[2-oxo-2-(piperidin-1-yl)ethyl]pyrrolidine-2,5-dione
1-cycloheptyl-N-(2-methoxy-2-methylpropyl)-6-oxopiperidine-3-carboxamide
1-cyclobutyl-N-(6-phenoxypyridin-3-yl)piperidine-2-carboxamide
(2S,4S)-4-amino-1-({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}sulfonyl)-N-methylpyrrolidine-2-carboxamide
N-{2-[4-(4-methylpiperazine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}-3-(trifluoromethyl)benzamide
1'-cycloheptyl-5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]