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2-[(2-hydroxyethyl)({[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl})amino]ethan-1-ol
1-benzyl-8-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-N-[3-(pyridin-3-yl)propyl]propanamide
methyl 3-cyclohexyl-1-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylate
1-[4-(2-phenoxyethyl)piperazin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
2-ethyl-7-methoxy-4-[(3-phenyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-1-(piperazin-1-yl)ethan-1-one
1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-N-[4-(3-methylphenyl)phenyl]piperidine-4-carboxamide
6-methoxy-N-[(4-methylphenyl)(pyridin-4-yl)methyl]pyrimidin-4-amine
2-cyclopropyl-5-[4-(6-methylpyridin-2-yl)piperazine-1-carbonyl]-3,4-dihydropyrimidin-4-one
N-(1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)pyrimidin-2-amine
7-(2-hydroxyethyl)-2-(6-methyl-2-phenylpyrimidin-4-yl)-2,7-diazaspiro[4.5]decan-6-one
2-({4-methyl-5-[(trimethyl-1H-pyrazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}sulfanyl)acetic acid
5-(2-aminopropanoyl)-N-phenyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1-[3-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)propyl]-1H-1,2,3-benzotriazole
(3R,4S)-4-{4-[(2-chloro-4-fluorophenyl)methyl]-1,4-diazepan-1-yl}oxolan-3-ol
5-(1,5-dimethyl-1H-indazole-3-carbonyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-[(4-chlorophenyl)(phenyl)methyl]-6-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-1-(4,6-dimethylquinazolin-2-yl)piperidine-4-carboxamide
N-cyclopropyl-2-{4-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]piperidin-1-yl}acetamide
N-benzyl-1-ethyl-N-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(3R,4R)-1-[(4-fluoro-3-methoxyphenyl)methyl]-3-hydroxypiperidin-4-yl]pyridine-4-carboxamide
2-({methyl[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}methyl)-3,4-dihydroquinazolin-4-one
N-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]-5-[(isoquinolin-5-yloxy)methyl]-1,2-oxazole-3-carboxamide
1-[7-(6,8-dimethoxy-4-methylquinolin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(3,5-dimethyl-1H-pyrazol-1-yl)propan-1-one
N-methyl-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-(2,2,6,6-tetramethylpiperidin-4-yl)propanamide
2-cyclopentyl-4-{octahydropyrrolo[1,2-a]piperazin-2-yl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine
(4aS,8aR)-1-(3-methoxypropyl)-6-[2-(3-methylphenoxy)acetyl]-decahydro-1,6-naphthyridin-2-one
N-({2-[2-(2-cyclopentylacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-2-(4-fluorophenyl)acetamide
3-(5-{1-[2-(2-methoxyphenoxy)ethyl]piperidin-3-yl}-1,2,4-oxadiazol-3-yl)pyridine
N-[1-(furan-2-yl)ethyl]-9-methoxy-N-methyl-3-[2-(2-methylphenyl)acetyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
ethyl 1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-4-(2-phenylethyl)piperidine-4-carboxylate
1-{4-methyl-2-[4-(thiomorpholin-4-yl)piperidin-1-yl]pyrimidin-5-yl}ethan-1-one
N-(pyridin-3-yl)spiro[2.5]octane-1-carboxamide
1-(6-methoxy-1-methyl-1H-indole-2-carbonyl)-3-phenylpyrrolidin-3-ol
1-[2-(4-methoxyphenyl)ethyl]-3-methyl-8-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S)-4-{3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzoyl}-1-ethyl-3-methylpiperazin-2-one
5-{1-[(2-methyl-1H-imidazol-4-yl)methyl]pyrrolidin-2-yl}-N-(1-methyl-1H-pyrazol-4-yl)thiophene-2-carboxamide
N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-2,1-benzoxazole-3-carboxamide
N-[(3S,4R)-4-(4-methylphenyl)-1-(1,2-oxazole-3-carbonyl)pyrrolidin-3-yl]cyclopropanecarboxamide
2-(2-methyl-1H-imidazol-1-yl)-1-[(1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
1-(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-3-(2-methoxyphenoxy)azetidine
8-fluoro-2-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]-1,4-dihydroquinolin-4-one
3-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-1-(3-methyl-1-propyl-1H-pyrazol-5-yl)urea
(3R,5S)-1-[(3,4-dimethoxyphenyl)methyl]-N-[3-(dimethylamino)propyl]-5-{[(6-methylpyridin-3-yl)oxy]methyl}piperidine-3-carboxamide
2-(2-oxo-1,3-oxazolidin-3-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)acetamide
N-[1-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-4-yl)-2-(3-methoxyphenyl)ethyl]-N-methylpyridine-3-carboxamide
1-[4-(2-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}-2-oxoethyl)phenyl]imidazolidin-2-one
(4aS,7aR)-1-[4-(dimethylamino)benzoyl]-4-ethyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}-2-(2-phenylethyl)-1,3-benzoxazole