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2-[(2S)-2-amino-4-methylpentanamido]-N-ethyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
2-(5-{[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)pyridine
(1S,5R)-6-(2,3-dihydro-1H-indene-5-carbonyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2,8-dimethyl-4-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidine-1-carbonyl]quinoline
2,6-difluoro-N-[2-(furan-2-ylmethoxy)phenyl]-4-methoxybenzamide
4-(7-chloroquinolin-4-yl)-2-[(3-methylpiperidin-1-yl)methyl]phenol
4-{[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]methyl}-N-methylbenzene-1-sulfonamide
4-(3-benzyl-1H-pyrazol-5-yl)-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-5-carbonyl}piperidine
4-(4-fluoro-2-methoxyphenyl)-2,5,6-trimethylpyrimidine
5-methyl-N-[(3-methylphenyl)methyl]-4-{[3-(2-oxopyrrolidin-1-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
2,4-dimethyl-N-[4-(4-{[(5-methylfuran-2-yl)methyl]amino}piperidin-1-yl)phenyl]benzamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-5-(2-fluorophenyl)-1,2,4-triazin-3-amine
N-phenyl-5-(thiomorpholine-4-carbonyl)pyrimidin-2-amine
(1R,9S)-5-amino-12-methyl-3-[4-(1H-pyrazol-1-yl)phenyl]-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
ethyl 1-{[3-(furan-3-amido)-2-(methoxycarbonyl)thieno[2,3-b]pyridin-6-yl]methyl}piperidine-4-carboxylate
1-({2-ethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)-3-(pyrrolidin-1-yl)propan-2-ol
5-(2H-1,3-benzodioxol-5-yl)-N-(pyridin-3-ylmethyl)-1,2,4-triazin-3-amine
2-methoxy-4-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]pyridine
2-{[3-(6-methoxynaphthalene-2-carbonyl)piperidin-1-yl]methyl}-6-methylpyridine
5-[2-(1-methyl-1H-imidazol-2-yl)phenyl]-3-(2-phenylethyl)-1H-1,2,4-triazole
N-(2,4-dichloro-3-methylphenyl)-3-oxo-2-(propan-2-yl)piperazine-1-carboxamide
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N,5,7-trimethylpyrido[2,3-d]pyrimidin-4-amine
N-[2-(furan-2-yl)ethyl]-8-methyl-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
1-[2-(dimethylamino)ethyl]-4-ethyl-3-[1-(6-methylpyridine-2-carbonyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
(1R,5R)-6-[3-(difluoromethoxy)benzoyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-[4-(1H-1,3-benzodiazol-2-ylmethyl)-1-(propan-2-yl)piperazin-2-yl]ethan-1-ol
4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]-N-[1-(thiophen-3-yl)propan-2-yl]benzamide
3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}-N-[2-(propan-2-yloxy)ethyl]propanamide
4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(4-methylpent-3-en-1-yl)piperidine
N-{[7-(3,6-dimethylpyrazin-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-ethyl-1-methyl-1H-pyrazole-5-carboxamide
N-(2-hydroxyethyl)-2-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)-N-(propan-2-yl)-1,3-oxazole-4-carboxamide
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]acetamide
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-6-methylpyridine-3-carboxamide
6-(benzyloxy)-4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
1-{3-[4-(3-{[methyl(quinolin-5-ylmethyl)amino]methyl}phenoxy)piperidine-1-carbonyl]phenyl}imidazolidin-2-one
1-[2-(2-hydroxyethyl)piperidin-1-yl]-3-{5-[(3-methylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propan-1-one
2-(1-ethyl-1H-pyrazole-4-carbonyl)-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decane
N-(2-{[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]amino}ethyl)acetamide
methyl 4-[2-amino-3-cyano-6-(2,5-dimethylphenyl)pyridin-4-yl]-1H-pyrazole-3-carboxylate
(2S)-1-{3-[(4-fluorophenyl)methyl]-1,2-oxazole-5-carbonyl}-4-methyl-2-phenylpiperazine
2-(1-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)pyridine
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)acetamide
3-[5-(2,1,3-benzoxadiazole-5-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
1-{3-[(3,4-difluorophenyl)amino]piperidin-1-yl}-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethan-1-one
(3R,5S)-N-(4-fluorophenyl)-5-(piperidine-1-carbonyl)piperidine-3-carboxamide
3-[(1S,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]-4H-chromen-4-one
N-(3,3-dimethylbutyl)-5-(3-methoxyphenoxymethyl)-1H-pyrazole-3-carboxamide
{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[1-(2-methyl-1,3-thiazol-4-yl)ethyl]amine
2-methyl-N-{[4-(2-methylpropyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-1,3-thiazole-4-carboxamide
4-fluoro-N-({1-[3-(methylsulfanyl)propyl]piperidin-3-yl}methyl)benzamide