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N-{[7-(2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}acetyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(methylsulfanyl)benzamide
N-[(2R,3R)-2-methoxy-1'-[(2-methoxyphenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide
N-methyl-4-(morpholine-4-carbonyl)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}pyridin-2-amine
2-(1-propylpiperidin-4-yl)-1-[4-(pyrimidin-2-yloxy)piperidin-1-yl]ethan-1-one
2-(5-acetylthiophen-3-yl)-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]acetamide
N-(cyclopropylmethyl)-1-[(2-fluorophenyl)methyl]-N-propyl-1H-1,2,3-triazole-4-carboxamide
1,9-dimethyl-N-(naphthalen-1-yl)-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
4-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(3-fluorophenyl)piperazin-2-one
N-{[7-chloro-2-(4-methoxyphenyl)quinolin-3-yl]methyl}-3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(oxolan-2-ylmethyl)propanamide
N-[2-(3-fluorophenyl)ethyl]-3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]propanamide
5,7-dimethyl-N-{[5-(5-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}pyrazolo[1,5-a]pyrimidine-2-carboxamide
2-(azepan-1-yl)-1-[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]ethan-1-one
4-hydroxy-2-methyl-N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]pyrimidine-5-carboxamide
1-(1-benzoxepine-4-carbonyl)-4-phenyl-1,4-diazepane
N4-(furan-2-ylmethyl)-7-[(2R)-pyrrolidine-2-carbonyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
8-(1-ethyl-1H-pyrazole-3-carbonyl)-3-hexyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
7-{[4-(benzyloxy)piperidin-1-yl]methyl}-4-(3-fluorobenzoyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[3-(3-ethylphenoxy)azetidine-1-carbonyl]-1-methylazepane
N-[(3,4-difluorophenyl)methyl]-3-{1-[3-(1,2-oxazolidin-2-yl)propanoyl]piperidin-3-yl}propanamide
[3-benzyl-1-(2,3-dimethoxybenzoyl)piperidin-3-yl]methanol
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(4-methoxybenzoyl)pyrrolidin-3-yl]methanol
1-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl}-2-{[(3,5-dimethylphenyl)methyl]sulfanyl}ethan-1-one
5-ethyl-N-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
3-fluoro-2-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
1-methyl-N-(1-{7-[(2,4,5-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)piperidine-4-carboxamide
2-[2-(3-methoxyphenyl)piperidin-1-yl]-N-(1-methyl-1H-pyrazol-4-yl)acetamide
(1S,5R)-6-(2-propyl-1,3-thiazole-4-carbonyl)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
N-(3-carbamoyl-4-fluorophenyl)-4-(3,6-dimethylpyrazin-2-yl)piperazine-1-carboxamide
1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl}piperidin-4-amine
4-(cyclopropylmethyl)-1-(1H-indol-5-ylmethyl)-3-(propan-2-yl)-1,4-diazepan-5-one
5-methoxy-2-{[2-(trifluoromethyl)morpholin-4-yl]methyl}pyridin-4-ol
3-{2-[4-(2-hydroxyethyl)piperazin-1-yl]-2-oxoethyl}-3-phenyl-1-[3-(pyridin-3-yloxy)propyl]pyrrolidine-2,5-dione
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-2-(2,5-dioxoimidazolidin-4-yl)acetamide
4-{1-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1-(4-methylphenyl)-1H-pyrazole
1-methyl-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1,2-dihydroquinolin-2-one
5-chloro-N-(isoquinolin-5-ylmethyl)-N-methyl-2,3-dihydro-1H-indole-2-carboxamide
2-{1-cyclopropyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}-N-(furan-2-ylmethyl)-N-methylacetamide
N-[cyclopropyl(6-methylpyridin-2-yl)methyl]-2,7,8-trimethylquinoline-4-carboxamide
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,6-dimethoxybenzamide
1-(2H-1,3-benzodioxol-5-yl)-5-[4-(methoxymethyl)-5-methyl-1,2-oxazol-3-yl]-3-(2-methylpropyl)-1H-1,2,4-triazole
4-[2-(2-fluorophenyl)acetyl]-5-methyl-1-(4-methylphenyl)piperazin-2-one
N-(2,2-dimethyloxan-4-yl)-N-ethyl-2-methyl-1-benzofuran-5-carboxamide
1-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]urea
1-(2,2-dimethyloxan-4-yl)-1-ethyl-3-(4-ethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)urea
N-(3-{[(2-fluorophenyl)methyl]sulfanyl}propyl)-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
1-acetyl-N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]piperidine-4-carboxamide
1-(1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carbonyl)azocane
4-ethyl-5-methyl-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]thiophene-3-carboxamide
N-methyl-N-(2-phenyl-1-{1-[2-(1H-pyrazol-1-yl)benzoyl]piperidin-4-yl}ethyl)thiophene-3-carboxamide