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7-(3,6-dimethylpyrazin-2-yl)-4-(5-propyl-1,2,4-oxadiazol-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(1-ethylpiperidin-4-yl)-N-[2-hydroxy-2-(naphthalen-2-yl)ethyl]acetamide
N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-N-(3-methoxypropyl)-5-(propan-2-yl)-1H-pyrazole-4-carboxamide
6-(cyclohexylmethyl)-N-(3-phenylpropyl)-6-azaspiro[2.5]octane-1-carboxamide
1-[7-(1,3-benzothiazol-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(3,4,5-trimethoxyphenyl)ethan-1-one
3-chloro-N-cyclopentyl-4-{[1-(3-methylbenzoyl)piperidin-4-yl]oxy}benzamide
1-{7-[(4-acetylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-(3,4-difluorophenyl)ethan-1-one
6-[(2E)-3-(2,5-difluorophenyl)prop-2-enoyl]-N-[3-(2-oxoimidazolidin-1-yl)phenyl]-6-azaspiro[2.5]octane-1-carboxamide
3-{1-[3-(ethylsulfanyl)propanoyl]piperidin-3-yl}-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[1'-(oxolane-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
1-[(2-fluorophenyl)methyl]-6-oxo-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]piperidine-3-carboxamide
N-butyl-5-(methoxymethyl)-N-methyl-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
2-{1-[3-(trifluoromethyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}pyridine
4-[6-(2-hydroxyethyl)pyrazolo[1,5-a]pyrimidine-3-carbonyl]-1-(4-methylphenyl)piperazin-2-one
3-({3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)pyridine
(3R,4R)-3-cyclobutyl-1-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]-4-methylpyrrolidin-3-ol
N-(1-{1-[2-(2-methoxyphenyl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methylbenzamide
3-(1-cyclopentanecarbonylpiperidin-4-yl)-1-(4-phenylpiperazin-1-yl)propan-1-one
N-[(3R,4S)-4-cyclopropyl-1-methanesulfonylpyrrolidin-3-yl]-2-methoxypyridine-3-carboxamide
4-{6-[4-(2-methoxyphenoxy)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}morpholine
2,2-dimethyl-N-{1-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}propanamide
4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)-1-[(2,4-dimethoxyphenyl)methyl]piperidine
N-(furan-2-ylmethyl)-N,1-dimethyl-5-[methyl(2-phenylethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
methyl 4-({[(3R,5S)-1-[(3-chlorophenyl)methyl]-5-(ethylcarbamoyl)pyrrolidin-3-yl]amino}methyl)benzoate
2-{[2-(2-hydroxyethyl)pyrrolidin-1-yl]methyl}-6,8-dimethylquinolin-4-ol
4-(3-fluorophenoxy)-1-(oxolan-3-ylmethyl)piperidine-4-carboxylic acid
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-2-(4-methylphenoxymethyl)furan-3-carboxamide
2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
2-amino-6-(1H-pyrrol-2-yl)-4-[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]pyridine-3-carbonitrile
1-{1-[2-(4-fluorophenoxy)ethanesulfonyl]piperidin-4-yl}pyrrolidin-2-one
N-[1-(pyrimidin-2-yl)piperidin-3-yl]-1-benzofuran-2-carboxamide
N-(3-chloro-2,6-dimethylphenyl)-3-acetamidopyrrolidine-1-carboxamide
3-(5-methyl-1H-1,2,4-triazol-3-yl)-1-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]propan-1-one
2-({[4-(dimethylamino)-5-methylpyrimidin-2-yl]amino}methyl)-3,5-dimethylpyridin-4-ol
N-{1-[7-(2-chloropyridine-4-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-2-methylpropyl}furan-3-carboxamide
5-ethyl-5-{1-[(2E)-3-(4-fluorophenyl)prop-2-enoyl]piperidin-4-yl}-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]imidazolidine-2,4-dione
4-{[2-(cyclopropylmethyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]methyl}benzonitrile
2-(dimethylamino)-N-[3-({[(3S,4S)-4-hydroxy-1-(propan-2-yl)pyrrolidin-3-yl]carbamoyl}amino)phenyl]acetamide
1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-4-(thian-4-yl)piperazine
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]acetamide
methyl 3-(1,3-dimethyl-1H-pyrazole-5-amido)-6-{[methyl(2-phenylethyl)amino]methyl}thieno[2,3-b]pyridine-2-carboxylate
1-cyclopropanecarbonyl-N-[4-(3-methoxyphenyl)phenyl]pyrrolidine-2-carboxamide
3,7-dimethyl-2-[4-(thian-4-yl)piperazin-1-yl]quinoline
4-(3-chloropyridin-4-yl)-3-ethyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-[1-(1-methylpiperidin-4-yl)-4-{[2-(2-phenylethynyl)phenyl]methyl}piperazin-2-yl]ethan-1-ol
6-fluoro-2-oxo-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-methyl-2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}acetamide
3-[(4-cyclohexyl-1,4-diazepan-1-yl)methyl]-1-(cyclopropylmethyl)-3-hydroxypiperidin-2-one
{[2-(difluoromethoxy)phenyl]methyl}(methyl)({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine